大野 浩章

最終更新日時: 2018/06/13 12:57:01

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氏名(漢字/フリガナ/アルファベット表記)
大野 浩章/オオノ ヒロアキ/Hiroaki Ohno
所属部署・職名(部局/所属/講座等/職名)
国際高等教育院/化学教室/教授
学部兼担
部局 所属 講座等 職名
薬学部
学内兼務
部局 所属 講座等 職名
薬学研究科 医薬創成情報科学専攻 医薬創成情報科学 教授
連絡先住所
種別 住所(日本語) 住所(英語)
職場 〒606-8501 京都市左京区吉田下阿達町46-29 46-29 Yoshidashimoadachi-cho, Sakyo-ku, Kyoto 606-8501, JAPAN
連絡先電話番号
種別 番号
職場 075-753-4571
所属学会(国内)
学会名(日本語) 学会名(英語)
日本薬学会 The Pharmaceutical Society of Japan
有機合成化学協会 The Society of Synthetic Organic Chemistry, Japan
日本ペプチド学会 The Japanese Peptide Society
取得学位
学位名(日本語) 学位名(英語) 大学(日本語) 大学(英語) 取得区分
修士(薬学) 京都大学
博士(薬学) 京都大学
出身大学院・研究科等
大学名(日本語) 大学名(英語) 研究科名(日本語) 研究科名(英語) 専攻名(日本語) 専攻名(英語) 修了区分
京都大学 大学院薬学研究科修士課程薬学専攻 修了
出身学校・専攻等
大学名(日本語) 大学名(英語) 学部名(日本語) 学部名(英語) 学科名(日本語) 学科名(英語) 卒業区分
京都大学 薬学部製薬化学科 卒業
出身高等学校
高等学校名 ふりがな
函館ラ・サール高等学校 はこだてら・さーるこうとうがっこう
職歴
期間 組織名(日本語) 組織名(英語) 職名(日本語) 職名(英語)
1999/01/01〜1999/09/15 日本学術振興会 Japan Society for the Promotion of Science 特別研究員 JSPS Research Fellow
1999/09/16〜2005/06/30 大阪大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Osaka University 助手 Assistant Professor
2005/07/01〜2008/03/31 京都大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Kyoto University 助教授 Associate Professor
2008/04/01〜2014/11/30 京都大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Kyoto University 准教授 Associate Professor
2014/12/01〜 京都大学国際高等教育院/薬学部・薬学研究科 Institute for Liberal Arts and Sciences/Graduate School of Pharmaceutical Sciences, Kyoto University 教授 Professor
個人ホームページ
URL
http://www.pharm.kyoto-u.ac.jp//seizo/
ORCID ID
orcid.org/0000-0002-3246-4809
研究テーマ
(日本語)
連続反応及び高原子効率反応による有機合成の効率化
(英語)
Efficiency Improvement of Synthetic Organic Chemistry Based on Cascade and Atom-Economical Reactions
研究概要
(日本語)
高い原子効率を有する素反応の開発やその連続化を通じて有機合成の効率化を図るとともに、有用な物質の効率的合成法の開発と創薬展開を行う。
(英語)
Improvement of reaction efficiency by development of novel atom-economical cascade reactions, synthetic studies of bioactive compounds, and their medicinal application studies are conducted.
研究分野(キーワード)
キーワード(日本語) キーワード(英語)
カスケード反応 cascade reactions
反応集積化 Reaction Integration
遷移金属 Transitiom Metals
含窒素複素環 Nitrogen Heterocycles
天然物合成 Natural Product Syntheses
研究分野(科研費分類コード)
科研費分類コード
化学系薬学
有機化学
論文
著者 著者(日本語) 著者(英語) タイトル タイトル(日本語) タイトル(英語) 書誌情報等 書誌情報等(日本語) 書誌情報等(英語) 出版年月 査読の有無 記述言語 掲載種別 公開
Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 2018/05 公開
Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Inorganic chemistry Inorganic chemistry Inorganic chemistry 2018/04 公開
Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Journal of medicinal chemistry Journal of medicinal chemistry Journal of medicinal chemistry 2018/04 公開
Kaneda M, Inuki S, Ohno H, Oishi S Kaneda M, Inuki S, Ohno H, Oishi S Kaneda M, Inuki S, Ohno H, Oishi S Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. The Journal of organic chemistry, 83, 6, 3047-3060 The Journal of organic chemistry, 83, 6, 3047-3060 The Journal of organic chemistry, 83, 6, 3047-3060 2018/03/16 公開
Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 2017/10 公開
Hamada N, Yoshida Y, Oishi S, Ohno H Hamada N, Yoshida Y, Oishi S, Ohno H Hamada N, Yoshida Y, Oishi S, Ohno H Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Organic letters, 19, 14, 3875-3878 Organic letters, 19, 14, 3875-3878 Organic letters, 19, 14, 3875-3878 2017/07 公開
Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 2017/06 公開
Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Bioorganic & medicinal chemistry, 25, 12, 3046-3052 Bioorganic & medicinal chemistry, 25, 12, 3046-3052 Bioorganic & medicinal chemistry, 25, 12, 3046-3052 2017/06 公開
Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 2017/06 公開
Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Bioconjugate chemistry, 28, 2, 609-619 Bioconjugate chemistry, 28, 2, 609-619 Bioconjugate chemistry, 28, 2, 609-619 2017/02 公開
Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Organic & biomolecular chemistry, 14, 38, 9104 Organic & biomolecular chemistry, 14, 38, 9104 Organic & biomolecular chemistry, 14, 38, 9104 2016/09 公開
Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. The Journal of organic chemistry, 81, 13, 5698 The Journal of organic chemistry, 81, 13, 5698 The Journal of organic chemistry, 81, 13, 5698 2016/07 公開
Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Journal of liposome research, 1-10 Journal of liposome research, 1-10 Journal of liposome research, 1-10 2016/06 公開
Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Screening of a virtual mirror-image library of natural products. Screening of a virtual mirror-image library of natural products. Screening of a virtual mirror-image library of natural products. Chemical communications (Cambridge, England), 52, 49, 7656 Chemical communications (Cambridge, England), 52, 49, 7656 Chemical communications (Cambridge, England), 52, 49, 7656 2016/06 公開
Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Development of novel NK3 receptor antagonists with reduced environmental impact. Development of novel NK3 receptor antagonists with reduced environmental impact. Development of novel NK3 receptor antagonists with reduced environmental impact. Bioorganic & medicinal chemistry, 24, 16, 3500 Bioorganic & medicinal chemistry, 24, 16, 3500 Bioorganic & medicinal chemistry, 24, 16, 3500 2016/05 公開
Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Organic letters, 18, 7, 1673 Organic letters, 18, 7, 1673 Organic letters, 18, 7, 1673 2016/04 公開
Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Bioorganic & medicinal chemistry, 24, 5, 1141 Bioorganic & medicinal chemistry, 24, 5, 1141 Bioorganic & medicinal chemistry, 24, 5, 1141 2016/03 公開
Wagner B, Hiller W, Ohno H, Krause N Wagner B, Hiller W, Ohno H, Krause N Wagner B, Hiller W, Ohno H, Krause N Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Organic & biomolecular chemistry, 14, 5, 1583 Organic & biomolecular chemistry, 14, 5, 1583 Organic & biomolecular chemistry, 14, 5, 1583 2016/02 公開
Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Chemical & pharmaceutical bulletin, 64, 7, 1003 Chemical & pharmaceutical bulletin, 64, 7, 1003 Chemical & pharmaceutical bulletin, 64, 7, 1003 2016 公開
Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Organic letters, 17, 24, 6250-6253 Organic letters, 17, 24, 6250-6253 Organic letters, 17, 24, 6250-6253 2015/12 公開
Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Journal of medicinal chemistry, 58, 13, 5218-5225 Journal of medicinal chemistry, 58, 13, 5218-5225 Journal of medicinal chemistry, 58, 13, 5218-5225 2015/06 公開
Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 2015/05 公開
Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Organic & biomolecular chemistry, 13, 16, 4706-4713 Organic & biomolecular chemistry, 13, 16, 4706-4713 Organic & biomolecular chemistry, 13, 16, 4706-4713 2015/04 公開
Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Organic letters, 17, 7, 1774-1777 Organic letters, 17, 7, 1774-1777 Organic letters, 17, 7, 1774-1777 2015/04 公開
Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Bioorganic & medicinal chemistry, 23, 7, 1447-1452 Bioorganic & medicinal chemistry, 23, 7, 1447-1452 Bioorganic & medicinal chemistry, 23, 7, 1447-1452 2015/04 公開
Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Organic letters, 17, 3, 604-607 Organic letters, 17, 3, 604-607 Organic letters, 17, 3, 604-607 2015/02 公開
Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Bioorganic & medicinal chemistry letters, 25, 2, 302-306 Bioorganic & medicinal chemistry letters, 25, 2, 302-306 Bioorganic & medicinal chemistry letters, 25, 2, 302-306 2015/01 公開
Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 2015/01 公開
Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. Biological & pharmaceutical bulletin, 38, 1, 30-38 Biological & pharmaceutical bulletin, 38, 1, 30-38 Biological & pharmaceutical bulletin, 38, 1, 30-38 2015 公開
Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. Biological & pharmaceutical bulletin, 38, 9, 1345-1351 Biological & pharmaceutical bulletin, 38, 9, 1345-1351 Biological & pharmaceutical bulletin, 38, 9, 1345-1351 2015 公開
Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 2014/12 公開
Nabika R, Oishi S, Misu R, Ohno H, Fujii N Nabika R, Oishi S, Misu R, Ohno H, Fujii N Nabika R, Oishi S, Misu R, Ohno H, Fujii N Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Bioorganic & medicinal chemistry, 22, 21, 6156-6162 Bioorganic & medicinal chemistry, 22, 21, 6156-6162 Bioorganic & medicinal chemistry, 22, 21, 6156-6162 2014/11 公開
Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Journal of medicinal chemistry, 57, 20, 8646-8651 Journal of medicinal chemistry, 57, 20, 8646-8651 Journal of medicinal chemistry, 57, 20, 8646-8651 2014/10 公開
Ohno H Ohno H Ohno H Synthesis and applications of vinylaziridines and ethynylaziridines. Synthesis and applications of vinylaziridines and ethynylaziridines. Synthesis and applications of vinylaziridines and ethynylaziridines. Chemical reviews, 114, 16, 7784-7814 Chemical reviews, 114, 16, 7784-7814 Chemical reviews, 114, 16, 7784-7814 2014/08 公開
Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Chemistry, an Asian journal, 9, 7, 1841-1846 Chemistry, an Asian journal, 9, 7, 1841-1846 Chemistry, an Asian journal, 9, 7, 1841-1846 2014/07 公開
Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Design and synthesis of fluorescent probes for GPR54. Design and synthesis of fluorescent probes for GPR54. Design and synthesis of fluorescent probes for GPR54. Bioorganic & medicinal chemistry, 22, 13, 3325-3330 Bioorganic & medicinal chemistry, 22, 13, 3325-3330 Bioorganic & medicinal chemistry, 22, 13, 3325-3330 2014/07 公開
Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Organic letters, 16, 11, 3138-3141 Organic letters, 16, 11, 3138-3141 Organic letters, 16, 11, 3138-3141 2014/06 公開
Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Bioorganic & medicinal chemistry, 22, 12, 3171-3179 Bioorganic & medicinal chemistry, 22, 12, 3171-3179 Bioorganic & medicinal chemistry, 22, 12, 3171-3179 2014/06 公開
Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. ACS medicinal chemistry letters, 5, 5, 566-571 ACS medicinal chemistry letters, 5, 5, 566-571 ACS medicinal chemistry letters, 5, 5, 566-571 2014/05 公開
Iwata A, Inuki S, Oishi S, Fujii N, Ohno H Iwata A, Inuki S, Oishi S, Fujii N, Ohno H A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation. Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation. Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Chemical communications (Cambridge, England), 50, 3, 298-300 Chemical communications (Cambridge, England), 50, 3, 298-300 Chemical Communications, 50, 3, 298-300 2014/01 英語 公開
Mizuhara T, Kato T, Hirai A, Kurihara H, Shimada Y, Taniguchi M, Maeta H, Togami H, Shimura K, Matsuoka M, Okazaki S, Takeuchi T, Ohno H, Oishi S, Fujii N Mizuhara T, Kato T, Hirai A, Kurihara H, Shimada Y, Taniguchi M, Maeta H, Togami H, Shimura K, Matsuoka M, Okazaki S, Takeuchi T, Ohno H, Oishi S, Fujii N T. Mizuhara; T. Kato; A. Hirai; H. Kurihara; Y. Shimada; M. Taniguchi; H. Maeta; H. Togami; K. Shimura; M. Matsuoka; S. Okazaki; T. Takeuchi; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents. Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents. Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents Bioorganic & medicinal chemistry letters, 23, 16, 4557-4561 Bioorganic & medicinal chemistry letters, 23, 16, 4557-4561 Bioorganic and Medicinal Chemistry Letters, 23, 16, 4557-4561 2013/08 英語 公開
Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Kubo T, Kaneda M, Ohno H, Osada H, Fujii N Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Kubo T, Kaneda M, Ohno H, Osada H, Fujii N T. Noguchi; S. Oishi; K. Honda; Y. Kondoh; T. Saito; T. Kubo; M. Kaneda; H. Ohno; H. Osada; N. Fujii Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors. Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors. Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors Bioorganic & medicinal chemistry letters, 23, 13, 3802-3805 Bioorganic & medicinal chemistry letters, 23, 13, 3802-3805 Bioorganic and Medicinal Chemistry Letters, 23, 13, 3802-3805 2013/07 英語 公開
Kobayashi Y, Oishi S, Kobayashi K, Ohno H, Tsutsumi H, Hata Y, Fujii N Kobayashi Y, Oishi S, Kobayashi K, Ohno H, Tsutsumi H, Hata Y, Fujii N Y. Kobayashi; S. Oishi; K. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Synthesis and functional analysis of deferriferrichrysin derivatives: application to colorimetric pH indicators. Synthesis and functional analysis of deferriferrichrysin derivatives: application to colorimetric pH indicators. Synthesis and functional analysis of deferriferrichrysin derivatives: Application to colorimetric pH indicators Bioorganic & medicinal chemistry, 21, 14, 4296-4300 Bioorganic & medicinal chemistry, 21, 14, 4296-4300 Bioorganic and Medicinal Chemistry, 21, 14, 4296-4300 2013/07 英語 公開
Chiba H, Sakai Y, Ohara A, Oishi S, Fujii N, Ohno H Chiba H, Sakai Y, Ohara A, Oishi S, Fujii N, Ohno H H. Chiba; Y. Sakai; A. Ohara; S. Oishi; N. Fujii; H. Ohno Convergent synthesis of (-)-quinocarcin based on the combination of Sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination. Convergent synthesis of (-)-quinocarcin based on the combination of Sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination. Convergent synthesis of (-)-quinocarcin based on the combination of sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination Chemistry (Weinheim an der Bergstrasse, Germany), 19, 27, 8875-8883 Chemistry (Weinheim an der Bergstrasse, Germany), 19, 27, 8875-8883 Chemistry - A European Journal, 19, 27, 8875-8883 2013/07 英語 公開
Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: synthetic study of laurendecumallene B. Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: synthetic study of laurendecumallene B. Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: Synthetic study of laurendecumallene B Organic letters, 15, 12, 3046-3049 Organic letters, 15, 12, 3046-3049 Organic Letters, 15, 12, 3046-3049 2013/06 英語 公開
Hou Z, Oishi S, Suzuki Y, Kure T, Nakanishi I, Hirasawa A, Tsujimoto G, Ohno H, Fujii N Hou Z, Oishi S, Suzuki Y, Kure T, Nakanishi I, Hirasawa A, Tsujimoto G, Ohno H, Fujii N Z. Hou; S. Oishi; Y. Suzuki; T. Kure; I. Nakanishi; A. Hirasawa; G. Tsujimoto; H. Ohno; N. Fujii Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors. Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors. Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: Application to the development of a new class of CK2 inhibitors Organic & biomolecular chemistry, 11, 20, 3288-3296 Organic & biomolecular chemistry, 11, 20, 3288-3296 Organic and Biomolecular Chemistry, 11, 20, 3288-3296 2013/05 英語 公開
Misu R, Oishi S, Setsuda S, Noguchi T, Kaneda M, Ohno H, Evans B, Navenot JM, Peiper SC, Fujii N Misu R, Oishi S, Setsuda S, Noguchi T, Kaneda M, Ohno H, Evans B, Navenot JM, Peiper SC, Fujii N R. Misu; S. Oishi; S. Setsuda; T. Noguchi; M. Kaneda; H. Ohno; B. Evans; J.-M. Navenot; S.C. Peiper; N. Fujii Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes. Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes. Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes Bioorganic & medicinal chemistry letters, 23, 9, 2628-2631 Bioorganic & medicinal chemistry letters, 23, 9, 2628-2631 Bioorganic and Medicinal Chemistry Letters, 23, 9, 2628-2631 2013/05 英語 公開
Misu R, Noguchi T, Ohno H, Oishi S, Fujii N Misu R, Noguchi T, Ohno H, Oishi S, Fujii N R. Misu; T. Noguchi; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists. Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists. Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists Bioorganic & medicinal chemistry, 21, 8, 2413-2417 Bioorganic & medicinal chemistry, 21, 8, 2413-2417 Bioorganic and Medicinal Chemistry, 21, 8, 2413-2417 2013/04 英語 公開
Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182. Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182. Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182 Bioorganic & medicinal chemistry, 21, 7, 2079-2087 Bioorganic & medicinal chemistry, 21, 7, 2079-2087 Bioorganic and Medicinal Chemistry, 21, 7, 2079-2087 2013/04 英語 公開
Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani siRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine. siRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine. SiRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine International journal of pharmaceutics, 443, 1-2, 221-229 International journal of pharmaceutics, 443, 1-2, 221-229 International Journal of Pharmaceutics, 443, 1-2, 221-229 2013/02 英語 公開
Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine. Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine. Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine Biological & pharmaceutical bulletin, 36, 5, 856-860 Biological & pharmaceutical bulletin, 36, 5, 856-860 Biological and Pharmaceutical Bulletin, 36, 5, 856-860 2013 英語 公開
Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents. Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents. Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin- 6-imine derivatives for potent anti-HIV agents Bioorganic & medicinal chemistry, 20, 21, 6434-6441 Bioorganic & medicinal chemistry, 20, 21, 6434-6441 Bioorganic and Medicinal Chemistry, 20, 21, 6434-6441 2012/11 英語 公開
Chiba H, Oishi S, Fujii N, Ohno H Chiba H, Oishi S, Fujii N, Ohno H H. Chiba; S. Oishi; N. Fujii; H. Ohno Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination. Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination. Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination Angewandte Chemie (International ed. in English), 51, 36, 9169-9172 Angewandte Chemie (International ed. in English), 51, 36, 9169-9172 Angewandte Chemie - International Edition, 51, 36, 9169-9172 2012/09 英語 公開
Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles. Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles. Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3] benzothiazin-6-imines and related tricyclic heterocycles Organic & biomolecular chemistry, 10, 33, 6792-6802 Organic & biomolecular chemistry, 10, 33, 6792-6802 Organic and Biomolecular Chemistry, 10, 33, 6792-6802 2012/09 英語 公開
Suzuki Y, Oishi S, Takei Y, Yasue M, Misu R, Naoe S, Hou Z, Kure T, Nakanishi I, Ohno H, Hirasawa A, Tsujimoto G, Fujii N Suzuki Y, Oishi S, Takei Y, Yasue M, Misu R, Naoe S, Hou Z, Kure T, Nakanishi I, Ohno H, Hirasawa A, Tsujimoto G, Fujii N Y. Suzuki; S. Oishi; Y. Takei; M. Yasue; R. Misu; S. Naoe; Z. Hou; T. Kure; I. Nakanishi; H. Ohno; A. Hirasawa; G. Tsujimoto; N. Fujii Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles. Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles. Design and synthesis of a novel class of CK2 inhibitors: Application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles Organic & biomolecular chemistry, 10, 25, 4907-4915 Organic & biomolecular chemistry, 10, 25, 4907-4915 Organic and Biomolecular Chemistry, 10, 25, 4907-4915 2012/07 英語 公開
Naoe S, Suzuki Y, Hirano K, Inaba Y, Oishi S, Fujii N, Ohno H Naoe S, Suzuki Y, Hirano K, Inaba Y, Oishi S, Fujii N, Ohno H S. Naoe; Y. Suzuki; K. Hirano; Y. Inaba; S. Oishi; N. Fujii; H. Ohno Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes. Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes. Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes The Journal of organic chemistry, 77, 11, 4907-4916 The Journal of organic chemistry, 77, 11, 4907-4916 Journal of Organic Chemistry, 77, 11, 4907-4916 2012/06 英語 公開
Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot JM, Peiper SC, Fujii N Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot JM, Peiper SC, Fujii N R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; Y. Yano; K. Matsuzaki; J.-M. Navenot; S.C. Peiper; N. Fujii Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists. Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists. Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists Bioconjugate chemistry, 23, 6, 1259-1265 Bioconjugate chemistry, 23, 6, 1259-1265 Bioconjugate Chemistry, 23, 6, 1259-1265 2012/06 英語 公開
Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Development and application of fluorescent SDF-1 derivatives. Development and application of fluorescent SDF-1 derivatives. Development and application of fluorescent SDF-1 derivatives. Future medicinal chemistry, 4, 7, 837-844 Future medicinal chemistry, 4, 7, 837-844 Future medicinal chemistry, 4, 7, 837-844 2012/05 公開
Ohno H, Iuchi M, Kojima N, Yoshimitsu T, Fujii N, Tanaka T Ohno H, Iuchi M, Kojima N, Yoshimitsu T, Fujii N, Tanaka T H. Ohno; M. Iuchi; N. Kojima; T. Yoshimitsu; N. Fujii; T. Tanaka Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade. Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade. Double C-H functionalization in sequential order: Direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade Chemistry (Weinheim an der Bergstrasse, Germany), 18, 17, 5352-5360 Chemistry (Weinheim an der Bergstrasse, Germany), 18, 17, 5352-5360 Chemistry - A European Journal, 18, 17, 5352-5360 2012/04 英語 公開
Kobayashi K, Oishi S, Kobayashi Y, Ohno H, Tsutsumi H, Hata Y, Fujii N Kobayashi K, Oishi S, Kobayashi Y, Ohno H, Tsutsumi H, Hata Y, Fujii N K. Kobayashi; S. Oishi; Y. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Synthesis and application of an Nδ-acetyl-Nδ-hydroxyornithine analog: identification of novel metal complexes of deferriferrichrysin. Synthesis and application of an Nδ-acetyl-Nδ-hydroxyornithine analog: identification of novel metal complexes of deferriferrichrysin. Synthesis and application of an N <sup>δ</sup>-acetyl-N <sup>δ</sup>-hydroxyornithine analog: Identification of novel metal complexes of deferriferrichrysin Bioorganic & medicinal chemistry, 20, 8, 2651-2655 Bioorganic & medicinal chemistry, 20, 8, 2651-2655 Bioorganic and Medicinal Chemistry, 20, 8, 2651-2655 2012/04 英語 公開
Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Yoshikawa Y, Furuya T, Hoshino M, Fujii N Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Yoshikawa Y, Furuya T, Hoshino M, Fujii N K. Kobayashi; S. Oishi; R. Hayashi; K. Tomita; T. Kubo; N. Tanahara; H. Ohno; Y. Yoshikawa; T. Furuya; M. Hoshino; N. Fujii Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres. Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres. Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres Journal of medicinal chemistry, 55, 6, 2746-2757 Journal of medicinal chemistry, 55, 6, 2746-2757 Journal of Medicinal Chemistry, 55, 6, 2746-2757 2012/03 英語 公開
Hou Z, Nakanishi I, Kinoshita T, Takei Y, Yasue M, Misu R, Suzuki Y, Nakamura S, Kure T, Ohno H, Murata K, Kitaura K, Hirasawa A, Tsujimoto G, Oishi S, Fujii N Hou Z, Nakanishi I, Kinoshita T, Takei Y, Yasue M, Misu R, Suzuki Y, Nakamura S, Kure T, Ohno H, Murata K, Kitaura K, Hirasawa A, Tsujimoto G, Oishi S, Fujii N Z. Hou; I. Nakanishi; T. Kinoshita; Y. Takei; M. Yasue; R. Misu; Y. Suzuki; S. Nakamura; T. Kure; H. Ohno; K. Murata; K. Kitaura; A. Hirasawa; G. Tsujimoto; S. Oishi; N. Fujii Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds. Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds. Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds Journal of medicinal chemistry, 55, 6, 2899-2903 Journal of medicinal chemistry, 55, 6, 2899-2903 Journal of Medicinal Chemistry, 55, 6, 2899-2903 2012/03 英語 公開
Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Organic letters, 14, 1, 326-329 Organic letters, 14, 1, 326-329 Organic letters, 14, 1, 326-329 2012/01 公開
Hirano K, Inaba Y, Takasu K, Oishi S, Takemoto Y, Fujii N, Ohno H Hirano K, Inaba Y, Takasu K, Oishi S, Takemoto Y, Fujii N, Ohno H K. Hirano; Y. Inaba; K. Takasu; S. Oishi; Y. Takemoto; N. Fujii; H. Ohno Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade. Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade. Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade The Journal of organic chemistry, 76, 21, 9068-9080 The Journal of organic chemistry, 76, 21, 9068-9080 Journal of Organic Chemistry, 76, 21, 9068-9080 2011/11 英語 公開
Kinoshita T, Sekiguchi Y, Fukada H, Nakaniwa T, Tada T, Nakamura S, Kitaura K, Ohno H, Suzuki Y, Hirasawa A, Nakanishi I, Tsujimoto G Kinoshita T, Sekiguchi Y, Fukada H, Nakaniwa T, Tada T, Nakamura S, Kitaura K, Ohno H, Suzuki Y, Hirasawa A, Nakanishi I, Tsujimoto G T. Kinoshita; Y. Sekiguchi; H. Fukada; T. Nakaniwa; T. Tada; S. Nakamura; K. Kitaura; H. Ohno; Y. Suzuki; A. Hirasawa; I. Nakanishi; G. Tsujimoto A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase. A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase. A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase Molecular and cellular biochemistry, 356, 1-2, 97-105 Molecular and cellular biochemistry, 356, 1-2, 97-105 Molecular and Cellular Biochemistry, 356, 1-2, 97-105 2011/10 英語 公開
Yoshimitsu Y, Oishi S, Miyagaki J, Inuki S, Ohno H, Fujii N Yoshimitsu Y, Oishi S, Miyagaki J, Inuki S, Ohno H, Fujii N Y. Yoshimitsu; S. Oishi; J. Miyagaki; S. Inuki; H. Ohno; N. Fujii Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C. Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C. Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Bioorganic & medicinal chemistry, 19, 18, 5402-5408 Bioorganic & medicinal chemistry, 19, 18, 5402-5408 Bioorganic and Medicinal Chemistry, 19, 18, 5402-5408 2011/09 英語 公開
Takeuchi T, Oishi S, Watanabe T, Ohno H, Sawada J, Matsuno K, Asai A, Asada N, Kitaura K, Fujii N Takeuchi T, Oishi S, Watanabe T, Ohno H, Sawada J, Matsuno K, Asai A, Asada N, Kitaura K, Fujii N T. Takeuchi; S. Oishi; T. Watanabe; H. Ohno; J.-I. Sawada; K. Matsuno; A. Asai; N. Asada; K. Kitaura; N. Fujii Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors. Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors. Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors Journal of medicinal chemistry, 54, 13, 4839-4846 Journal of medicinal chemistry, 54, 13, 4839-4846 Journal of Medicinal Chemistry, 54, 13, 4839-4846 2011/07 英語 公開
Iwata A, Inuki S, Oishi S, Fujii N, Ohno H Iwata A, Inuki S, Oishi S, Fujii N, Ohno H A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane. Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane. Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane The Journal of organic chemistry, 76, 13, 5506-5512 The Journal of organic chemistry, 76, 13, 5506-5512 Journal of Organic Chemistry, 76, 13, 5506-5512 2011/07 英語 公開
Inokuchi E, Oishi S, Kubo T, Ohno H, Shimura K, Matsuoka M, Fujii N Inokuchi E, Oishi S, Kubo T, Ohno H, Shimura K, Matsuoka M, Fujii N E. Inokuchi; S. Oishi; T. Kubo; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Potent CXCR4 antagonists containing amidine type Peptide bond isosteres. Potent CXCR4 antagonists containing amidine type Peptide bond isosteres. Potent CXCR4 antagonists containing amidine type peptide bond isosteres ACS medicinal chemistry letters, 2, 6, 477-480 ACS medicinal chemistry letters, 2, 6, 477-480 ACS Medicinal Chemistry Letters, 2, 6, 477-480 2011/06 英語 公開
Masuda R, Oishi S, Ohno H, Kimura H, Saji H, Fujii N Masuda R, Oishi S, Ohno H, Kimura H, Saji H, Fujii N R. Masuda; S. Oishi; H. Ohno; H. Kimura; H. Saji; N. Fujii Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR4. Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR4. Concise site-specific synthesis of DTPA-peptide conjugates: Application to imaging probes for the chemokine receptor CXCR4 Bioorganic & medicinal chemistry, 19, 10, 3216-3220 Bioorganic & medicinal chemistry, 19, 10, 3216-3220 Bioorganic and Medicinal Chemistry, 19, 10, 3216-3220 2011/05 英語 公開
Inokuchi E, Yamada A, Hozumi K, Tomita K, Oishi S, Ohno H, Nomizu M, Fujii N Inokuchi E, Yamada A, Hozumi K, Tomita K, Oishi S, Ohno H, Nomizu M, Fujii N E. Inokuchi; A. Yamada; K. Hozumi; K. Tomita; S. Oishi; H. Ohno; M. Nomizu; N. Fujii Design and synthesis of amidine-type peptide bond isosteres: application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis. Design and synthesis of amidine-type peptide bond isosteres: application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis. Design and synthesis of amidine-type peptide bond isosteres: Application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis Organic & biomolecular chemistry, 9, 9, 3421-3427 Organic & biomolecular chemistry, 9, 9, 3421-3427 Organic and Biomolecular Chemistry, 9, 9, 3421-3427 2011/05 英語 公開
Inuki S, Iwata A, Oishi S, Fujii N, Ohno H Inuki S, Iwata A, Oishi S, Fujii N, Ohno H S. Inuki; A. Iwata; S. Oishi; N. Fujii; H. Ohno Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups. Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups. Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups The Journal of organic chemistry, 76, 7, 2072-2083 The Journal of organic chemistry, 76, 7, 2072-2083 Journal of Organic Chemistry, 76, 7, 2072-2083 2011/04 英語 公開
Hirano K, Inaba Y, Takahashi N, Shimano M, Oishi S, Fujii N, Ohno H Hirano K, Inaba Y, Takahashi N, Shimano M, Oishi S, Fujii N, Ohno H K. Hirano; Y. Inaba; N. Takahashi; M. Shimano; S. Oishi; N. Fujii; H. Ohno Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes. Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes. Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes The Journal of organic chemistry, 76, 5, 1212-1227 The Journal of organic chemistry, 76, 5, 1212-1227 Journal of Organic Chemistry, 76, 5, 1212-1227 2011/03 英語 公開
Oishi S, Misu R, Tomita K, Setsuda S, Masuda R, Ohno H, Naniwa Y, Ieda N, Inoue N, Ohkura S, Uenoyama Y, Tsukamura H, Maeda K, Hirasawa A, Tsujimoto G, Fujii N Oishi S, Misu R, Tomita K, Setsuda S, Masuda R, Ohno H, Naniwa Y, Ieda N, Inoue N, Ohkura S, Uenoyama Y, Tsukamura H, Maeda K, Hirasawa A, Tsujimoto G, Fujii N S. Oishi; R. Misu; K. Tomita; S. Setsuda; R. Masuda; H. Ohno; Y. Naniwa; N. Ieda; N. Inoue; S. Ohkura; Y. Uenoyama; H. Tsukamura; K.-I. Maeda; A. Hirasawa; G. Tsujimoto; N. Fujii Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands. Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands. Activation of neuropeptide FF receptors by kisspeptin receptor ligands ACS medicinal chemistry letters, 2, 1, 53-57 ACS medicinal chemistry letters, 2, 1, 53-57 ACS Medicinal Chemistry Letters, 2, 1, 53-57 2011/01 英語 公開
Ohta Y, Tokimizu Y, Oishi S, Fujii N, Ohno H Ohta Y, Tokimizu Y, Oishi S, Fujii N, Ohno H Y. Ohta; Y. Tokimizu; S. Oishi; N. Fujii; H. Ohno Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines. Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines. Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines Organic letters, 12, 17, 3963-3965 Organic letters, 12, 17, 3963-3965 Organic Letters, 12, 17, 3963-3965 2010/09 英語 公開
Okano A, Tsukamoto K, Kosaka S, Maeda H, Oishi S, Tanaka T, Fujii N, Ohno H Okano A, Tsukamoto K, Kosaka S, Maeda H, Oishi S, Tanaka T, Fujii N, Ohno H A. Okano; K. Tsukamoto; S. Kosaka; H. Maeda; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Synthesis of fused and linked bicyclic nitrogen heterocycles by palladiumcatalyzed domino cyclization of propargyl bromides Chemistry (Weinheim an der Bergstrasse, Germany), 16, 28, 8410-8418 Chemistry (Weinheim an der Bergstrasse, Germany), 16, 28, 8410-8418 Chemistry - A European Journal, 16, 28, 8410-8418 2010/07 英語 公開
Oishi S, Watanabe T, Sawada J, Asai A, Ohno H, Fujii N Oishi S, Watanabe T, Sawada J, Asai A, Ohno H, Fujii N S. Oishi; T. Watanabe; J.-I. Sawada; A. Asai; H. Ohno; N. Fujii Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds. Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds. Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds Journal of medicinal chemistry, 53, 13, 5054-5058 Journal of medicinal chemistry, 53, 13, 5054-5058 Journal of Medicinal Chemistry, 53, 13, 5054-5058 2010/07 英語 公開
Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H S. Inuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates. Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates. Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (Jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates The Journal of organic chemistry, 75, 11, 3831-3842 The Journal of organic chemistry, 75, 11, 3831-3842 Journal of Organic Chemistry, 75, 11, 3831-3842 2010/06 英語 公開
Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B). Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B). Stereoselective divergent synthesis of four diastereomers of pachastrissamine (Jaspine B) The Journal of organic chemistry, 75, 11, 3843-3846 The Journal of organic chemistry, 75, 11, 3843-3846 Journal of Organic Chemistry, 75, 11, 3843-3846 2010/06 英語 公開
Okano A, Oishi S, Tanaka T, Fujii N, Ohno H Okano A, Oishi S, Tanaka T, Fujii N, Ohno H A. Okano; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with isocyanate. Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with isocyanate. Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with Isocyanate The Journal of organic chemistry, 75, 10, 3396-3400 The Journal of organic chemistry, 75, 10, 3396-3400 Journal of Organic Chemistry, 75, 10, 3396-3400 2010/05 英語 公開
Narumi T, Hayashi R, Tomita K, Kobayashi K, Tanahara N, Ohno H, Naito T, Kodama E, Matsuoka M, Oishi S, Fujii N Narumi T, Hayashi R, Tomita K, Kobayashi K, Tanahara N, Ohno H, Naito T, Kodama E, Matsuoka M, Oishi S, Fujii N T. Narumi; R. Hayashi; K. Tomita; K. Kobayashi; N. Tanahara; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres. Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres. Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres Organic & biomolecular chemistry, 8, 3, 616-621 Organic & biomolecular chemistry, 8, 3, 616-621 Organic and Biomolecular Chemistry, 8, 3, 616-621 2010/02 英語 公開
Mizuhara T, Oishi S, Fujii N, Ohno H Mizuhara T, Oishi S, Fujii N, Ohno H T. Mizuhara; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S(N)Ar-type C-S, C-N, or C-O bond formation with heterocumulenes. Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S(N)Ar-type C-S, C-N, or C-O bond formation with heterocumulenes. Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S<sub>N</sub>Ar-type C-S, C-N, or C-O bond formation with heterocumulenes The Journal of organic chemistry, 75, 1, 265-268 The Journal of organic chemistry, 75, 1, 265-268 Journal of Organic Chemistry, 75, 1, 265-268 2010/01 英語 公開
Kajiwara K, Watanabe K, Tokiwa R, Kurose T, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N Kajiwara K, Watanabe K, Tokiwa R, Kurose T, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N K. Kajiwara; K. Watanabe; R. Tokiwa; T. Kurose; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group. Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group. Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group Bioorganic & medicinal chemistry, 17, 23, 7964-7970 Bioorganic & medicinal chemistry, 17, 23, 7964-7970 Bioorganic and Medicinal Chemistry, 17, 23, 7964-7970 2009/12 英語 公開
Tanaka M, Kajiwara K, Tokiwa R, Watanabe K, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N Tanaka M, Kajiwara K, Tokiwa R, Watanabe K, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N M. Tanaka; K. Kajiwara; R. Tokiwa; K. Watanabe; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins. Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins. Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins Bioorganic & medicinal chemistry, 17, 21, 7487-7492 Bioorganic & medicinal chemistry, 17, 21, 7487-7492 Bioorganic and Medicinal Chemistry, 17, 21, 7487-7492 2009/11 英語 公開
Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H S. Lnuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes. Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes. Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes Organic letters, 11, 19, 4478-4481 Organic letters, 11, 19, 4478-4481 Organic Letters, 11, 19, 4478-4481 2009/10 英語 公開
Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization. Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization. Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization The Journal of organic chemistry, 74, 18, 7052-7058 The Journal of organic chemistry, 74, 18, 7052-7058 Journal of Organic Chemistry, 74, 18, 7052-7058 2009/09 英語 公開
Watabe T, Terakawa Y, Watanabe K, Ohno H, Nakano H, Nakatsu T, Kato H, Izumi K, Kodama E, Matsuoka M, Kitaura K, Oishi S, Fujii N Watabe T, Terakawa Y, Watanabe K, Ohno H, Nakano H, Nakatsu T, Kato H, Izumi K, Kodama E, Matsuoka M, Kitaura K, Oishi S, Fujii N T. Watabe; Y. Terakawa; K. Watanabe; H. Ohno; H. Nakano; T. Nakatsu; H. Kato; K. Izumi; E. Kodama; M. Matsuoka; K. Kitaura; S. Oishi; N. Fujii X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution. X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution. X-ray Crystallographic Study of an HIV-1 Fusion Inhibitor with the gp41 S138A Substitution Journal of molecular biology, 392, 3, 657-665 Journal of molecular biology, 392, 3, 657-665 Journal of Molecular Biology, 392, 3, 657-665 2009/09 英語 公開
Ohta Y, Kubota Y, Watabe T, Chiba H, Oishi S, Fujii N, Ohno H Ohta Y, Kubota Y, Watabe T, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; Y. Kubota; T. Watabe; H. Chiba; S. Oishi; N. Fujii; H. Ohno Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation. Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation. Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation The Journal of organic chemistry, 74, 16, 6299-6302 The Journal of organic chemistry, 74, 16, 6299-6302 Journal of Organic Chemistry, 74, 16, 6299-6302 2009/08 英語 公開
Oishi S, Kamitani H, Kodera Y, Watanabe K, Kobayashi K, Narumi T, Tomita K, Ohno H, Naito T, Kodama E, Matsuoka M, Fujii N Oishi S, Kamitani H, Kodera Y, Watanabe K, Kobayashi K, Narumi T, Tomita K, Ohno H, Naito T, Kodama E, Matsuoka M, Fujii N S. Oishi; H. Kamitani; Y. Kodera; K. Watanabe; K. Kobayashi; T. Narumi; K. Tomita; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues. Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues. Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: Synthesis and bioevaluation of α-helical anti-HIV peptide analogues Organic & biomolecular chemistry, 7, 14, 2872-2877 Organic & biomolecular chemistry, 7, 14, 2872-2877 Organic and Biomolecular Chemistry, 7, 14, 2872-2877 2009/07 英語 公開
Oishi S, Kodera Y, Nishikawa H, Kamitani H, Watabe T, Ohno H, Tochikura T, Shimane K, Kodama E, Matsuoka M, Mizukoshi F, Tsujimoto H, Fujii N Oishi S, Kodera Y, Nishikawa H, Kamitani H, Watabe T, Ohno H, Tochikura T, Shimane K, Kodama E, Matsuoka M, Mizukoshi F, Tsujimoto H, Fujii N S. Oishi; Y. Kodera; H. Nishikawa; H. Kamitani; T. Watabe; H. Ohno; T. Tochikura; K. Shimane; E. Kodama; M. Matsuoka; F. Mizukoshi; H. Tsujimoto; N. Fujii Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus. Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus. Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus Bioorganic & medicinal chemistry, 17, 14, 4916-4920 Bioorganic & medicinal chemistry, 17, 14, 4916-4920 Bioorganic and Medicinal Chemistry, 17, 14, 4916-4920 2009/07 英語 公開
Watanabe T, Oishi S, Fujii N, Ohno H Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: synthesis and mechanistic study. Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: synthesis and mechanistic study. Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: Synthesis and mechanistic study The Journal of organic chemistry, 74, 13, 4720-4726 The Journal of organic chemistry, 74, 13, 4720-4726 Journal of Organic Chemistry, 74, 13, 4720-4726 2009/07 英語 公開
Mizuhara T, Inuki S, Oishi S, Fujii N, Ohno H Mizuhara T, Inuki S, Oishi S, Fujii N, Ohno H T. Mizuhara; S. Inuki; S. Oishi; N. Fujii; H. Ohno Cu(II)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group. Cu(II)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group. Cu(ii)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group Chemical communications (Cambridge, England), 23, 3413-3415 Chemical communications (Cambridge, England), 23, 3413-3415 Chemical Communications, 23, 3413-3415 2009/06 英語 公開
Kobayashi K, Narumi T, Oishi S, Ohno H, Fujii N Kobayashi K, Narumi T, Oishi S, Ohno H, Fujii N K. Kobayashi; T. Narumi; S. Oishi; H. Ohno; N. Fujii Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper-mediated S(N)2' alkylation. Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper-mediated S(N)2' alkylation. Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper- mediated S<sub>N</sub>2′ alkylation The Journal of organic chemistry, 74, 12, 4626-4629 The Journal of organic chemistry, 74, 12, 4626-4629 Journal of Organic Chemistry, 74, 12, 4626-4629 2009/06 英語 公開
Suzuki Y, Ohta Y, Oishi S, Fujii N, Ohno H Suzuki Y, Ohta Y, Oishi S, Fujii N, Ohno H Y. Suzuki; Y. Ohta; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization. Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization. Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization The Journal of organic chemistry, 74, 11, 4246-4251 The Journal of organic chemistry, 74, 11, 4246-4251 Journal of Organic Chemistry, 74, 11, 4246-4251 2009/06 英語 公開
Ohta Y, Oishi S, Fujii N, Ohno H Ohta Y, Oishi S, Fujii N, Ohno H Y. Ohta; S. Oishi; N. Fujii; H. Ohno Facile synthesis of 1,2,3,4-tetrahydro-beta-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization. Facile synthesis of 1,2,3,4-tetrahydro-beta-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization. Facile synthesis of 1,2,3,4-tetrahydro-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization Organic letters, 11, 9, 1979-1982 Organic letters, 11, 9, 1979-1982 Organic Letters, 11, 9, 1979-1982 2009/05 英語 公開
Nakaniwa T, Kinoshita T, Sekiguchi Y, Tada T, Nakanishi I, Kitaura K, Suzuki Y, Ohno H, Hirasawa A, Tsujimoto G Nakaniwa T, Kinoshita T, Sekiguchi Y, Tada T, Nakanishi I, Kitaura K, Suzuki Y, Ohno H, Hirasawa A, Tsujimoto G T. Nakaniwa; T. Kinoshita; Y. Sekiguchi; T. Tada; I. Nakanishi; K. Kitaura; Y. Suzuki; H. Ohno; A. Hirasawa; G. Tsujimoto Structure of human protein kinase CK2 alpha 2 with a potent indazole-derivative inhibitor. Structure of human protein kinase CK2 alpha 2 with a potent indazole-derivative inhibitor. Structure of human protein kinase CK2α2 with a potent indazole-derivative inhibitor Acta crystallographica. Section F, Structural biology and crystallization communications, 65, 75-79 Acta crystallographica. Section F, Structural biology and crystallization communications, 65, 75-79 Acta Crystallographica Section F: Structural Biology and Crystallization Communications, 65, 75-79 2009/02 英語 公開
Tomita K, Popiel HA, Nagai Y, Toda T, Yoshimitsu Y, Ohno H, Oishi S, Fujii N Tomita K, Popiel HA, Nagai Y, Toda T, Yoshimitsu Y, Ohno H, Oishi S, Fujii N K. Tomita; H.A. Popiel; Y. Nagai; T. Toda; Y. Yoshimitsu; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study on polyglutamine binding peptide QBP1. Structure-activity relationship study on polyglutamine binding peptide QBP1. Structure-activity relationship study on polyglutamine binding peptide QBP1 Bioorganic & medicinal chemistry, 17, 3, 1259-1263 Bioorganic & medicinal chemistry, 17, 3, 1259-1263 Bioorganic and Medicinal Chemistry, 17, 3, 1259-1263 2009/02 英語 公開
Oishi S, Ito S, Nishikawa H, Tanaka M, Ohno H, Otaka A, Izumi K, Kodama E, Matsuoka M, Fujii N Oishi S, Ito S, Nishikawa H, Tanaka M, Ohno H, Otaka A, Izumi K, Kodama E, Matsuoka M, Fujii N S. Oishi; S. Ito; H. Nishikawa; M. Tanaka; H. Ohno; A. Otaka; K. Izumi; E. Kodama; M. Matsuoka; N. Fujii Development of a novel fusion inhibitor against T-20-resistant HIV-1. Development of a novel fusion inhibitor against T-20-resistant HIV-1. Development of a novel fusion inhibitor against T-20-resistant HIV-1. Advances in experimental medicine and biology, 611, 389-391 Advances in experimental medicine and biology, 611, 389-391 Advances in experimental medicine and biology, 611, 389-391 2009 英語 公開
Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Advances in experimental medicine and biology, 611, 365-366 Advances in experimental medicine and biology, 611, 365-366 Advances in experimental medicine and biology, 611, 365-366 2009 英語 公開
Tomita K, Oishi S, Ohno H, Peiper SC, Fujii N Tomita K, Oishi S, Ohno H, Peiper SC, Fujii N K. Tomita; S. Oishi; H. Ohno; S.C. Peiper; N. Fujii Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase. Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase. Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase Journal of medicinal chemistry, 51, 23, 7645-7649 Journal of medicinal chemistry, 51, 23, 7645-7649 Journal of Medicinal Chemistry, 51, 23, 7645-7649 2008/12 英語 公開
Inuki S, Oishi S, Fujii N, Ohno H Inuki S, Oishi S, Fujii N, Ohno H S. Inuki; S. Oishi; N. Fujii; H. Ohno Total synthesis of (+/-)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group. Total synthesis of (+/-)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group. Total synthesis of (±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group Organic letters, 10, 22, 5239-5242 Organic letters, 10, 22, 5239-5242 Organic Letters, 10, 22, 5239-5242 2008/11 英語 公開
Nishikawa H, Oishi S, Fujita M, Watanabe K, Tokiwa R, Ohno H, Kodama E, Izumi K, Kajiwara K, Naitoh T, Matsuoka M, Otaka A, Fujii N Nishikawa H, Oishi S, Fujita M, Watanabe K, Tokiwa R, Ohno H, Kodama E, Izumi K, Kajiwara K, Naitoh T, Matsuoka M, Otaka A, Fujii N H. Nishikawa; S. Oishi; M. Fujita; K. Watanabe; R. Tokiwa; H. Ohno; E. Kodama; K. Izumi; K. Kajiwara; T. Naitoh; M. Matsuoka; A. Otaka; N. Fujii Identification of minimal sequence for HIV-1 fusion inhibitors. Identification of minimal sequence for HIV-1 fusion inhibitors. Identification of minimal sequence for HIV-1 fusion inhibitors Bioorganic & medicinal chemistry, 16, 20, 9184-9187 Bioorganic & medicinal chemistry, 16, 20, 9184-9187 Bioorganic and Medicinal Chemistry, 16, 20, 9184-9187 2008/10 英語 公開
Suzuki Y, Cluzeau J, Hara T, Hirasawa A, Tsujimoto G, Oishi S, Ohno H, Fujii N Suzuki Y, Cluzeau J, Hara T, Hirasawa A, Tsujimoto G, Oishi S, Ohno H, Fujii N Y. Suzuki; J. Cluzeau; T. Hara; A. Hirasawa; G. Tsujimoto; S. Oishi; H. Ohno; N. Fujii Structure-activity relationships of pyrazine-based CK2 inhibitors: synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines. Structure-activity relationships of pyrazine-based CK2 inhibitors: synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines. Structure-activity relationships of pyrazine-based CK2 inhibitors: Synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines Archiv der Pharmazie, 341, 9, 554-561 Archiv der Pharmazie, 341, 9, 554-561 Archiv der Pharmazie, 341, 9, 554-561 2008/09 英語 公開
Iwasaki H, Eguchi T, Tsutsui N, Ohno H, Tanaka T Iwasaki H, Eguchi T, Tsutsui N, Ohno H, Tanaka T H. Iwasaki; T. Eguchi; N. Tsutsui; H. Ohno; T. Tanaka Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring. Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring. Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring The Journal of organic chemistry, 73, 18, 7145-7152 The Journal of organic chemistry, 73, 18, 7145-7152 Journal of Organic Chemistry, 73, 18, 7145-7152 2008/09 英語 公開
Okano A, Mizutani T, Oishi S, Tanaka T, Ohno H, Fujii N Okano A, Mizutani T, Oishi S, Tanaka T, Ohno H, Fujii N A. Okano; T. Mizutani; S. Oishi; T. Tanaka; H. Ohno; N. Fujii Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade. Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade. Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade Chemical communications (Cambridge, England), 30, 3534-3536 Chemical communications (Cambridge, England), 30, 3534-3536 Chemical Communications, 30, 3534-3536 2008/08 英語 公開
Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Concise synthesis of indole-fused 1,4-diazepines through copper(I)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation. Concise synthesis of indole-fused 1,4-diazepines through copper(I)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation. Concise synthesis of indole-fused 1,4-diazepines through copper(l)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation Organic letters, 10, 16, 3535-3538 Organic letters, 10, 16, 3535-3538 Organic Letters, 10, 16, 3535-3538 2008/08 英語 公開
Ueda S, Kato M, Inuki S, Ohno H, Evans B, Wang ZX, Peiper SC, Izumi K, Kodama E, Matsuoka M, Nagasawa H, Oishi S, Fujii N Ueda S, Kato M, Inuki S, Ohno H, Evans B, Wang ZX, Peiper SC, Izumi K, Kodama E, Matsuoka M, Nagasawa H, Oishi S, Fujii N S. Ueda; M. Kato; S. Inuki; H. Ohno; B. Evans; Z.-x. Wang; S.C. Peiper; K. Izumi; E. Kodama; M. Matsuoka; H. Nagasawa; S. Oishi; N. Fujii Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach. Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach. Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Bioorganic & medicinal chemistry letters, 18, 14, 4124-4129 Bioorganic & medicinal chemistry letters, 18, 14, 4124-4129 Bioorganic and Medicinal Chemistry Letters, 18, 14, 4124-4129 2008/07 英語 公開
Inokuchi E, Narumi T, Niida A, Kobayashi K, Tomita K, Oishi S, Ohno H, Fujii N Inokuchi E, Narumi T, Niida A, Kobayashi K, Tomita K, Oishi S, Ohno H, Fujii N E. Inokuchi; T. Narumi; A. Niida; K. Kobayashi; K. Tomita; S. Oishi; H. Ohno; N. Fujii Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates. Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates. Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates The Journal of organic chemistry, 73, 10, 3942-3945 The Journal of organic chemistry, 73, 10, 3942-3945 Journal of Organic Chemistry, 73, 10, 3942-3945 2008/05 英語 公開
Oishi S, Masuda R, Evans B, Ueda S, Goto Y, Ohno H, Hirasawa A, Tsujimoto G, Wang Z, Peiper SC, Naito T, Kodama E, Matsuoka M, Fujii N Oishi S, Masuda R, Evans B, Ueda S, Goto Y, Ohno H, Hirasawa A, Tsujimoto G, Wang Z, Peiper SC, Naito T, Kodama E, Matsuoka M, Fujii N S. Oishi; R. Masuda; B. Evans; S. Ueda; Y. Goto; H. Ohno; A. Hirasawa; G. Tsujimoto; Z. Wang; S.C. Peiper; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4. Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4. Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4 Chembiochem : a European journal of chemical biology, 9, 7, 1154-1158 Chembiochem : a European journal of chemical biology, 9, 7, 1154-1158 ChemBioChem, 9, 7, 1154-1158 2008/05 英語 公開
Watanabe T, Oishi S, Fujii N, Ohno H Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines. Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines. Palladium-catalyzed sp<sup>3</sup> C-H activation of simple alkyl groups: Direct preparation of indoline derivatives from N-alkyl-2-bromoanilines Organic letters, 10, 9, 1759-1762 Organic letters, 10, 9, 1759-1762 Organic Letters, 10, 9, 1759-1762 2008/05 英語 公開
Ohno H, Okano A, Kosaka S, Tsukamoto K, Ohata M, Ishihara K, Maeda H, Tanaka T, Fujii N Ohno H, Okano A, Kosaka S, Tsukamoto K, Ohata M, Ishihara K, Maeda H, Tanaka T, Fujii N H. Ohno; A. Okano; S. Kosaka; K. Tsukamoto; M. Ohata; K. Ishihara; H. Maeda; T. Tanaka; N. Fujii Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides Organic letters, 10, 6, 1171-1174 Organic letters, 10, 6, 1171-1174 Organic Letters, 10, 6, 1171-1174 2008/03 英語 公開
Ohta Y, Oishi S, Fujii N, Ohno H Ohta Y, Oishi S, Fujii N, Ohno H Y. Ohta; S. Oishi; N. Fujii; H. Ohno Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation. Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation. Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation Chemical communications (Cambridge, England), 7, 835-837 Chemical communications (Cambridge, England), 7, 835-837 Chemical Communications, 7, 835-837 2008/02 英語 公開
Oishi S, Ito S, Nishikawa H, Watanabe K, Tanaka M, Ohno H, Izumi K, Sakagami Y, Kodama E, Matsuoka M, Fujii N Oishi S, Ito S, Nishikawa H, Watanabe K, Tanaka M, Ohno H, Izumi K, Sakagami Y, Kodama E, Matsuoka M, Fujii N S. Oishi; S. Ito; H. Nishikawa; K. Watanabe; M. Tanaka; H. Ohno; K. Izumi; Y. Sakagami; E. Kodama; M. Matsuoka; N. Fujii Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity. Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity. Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity Journal of medicinal chemistry, 51, 3, 388-391 Journal of medicinal chemistry, 51, 3, 388-391 Journal of Medicinal Chemistry, 51, 3, 388-391 2008/02 英語 公開
S. Oishi; T. Narumi; H. Ohno; A. Otaka; N. Fujii S. Oishi; T. Narumi; H. Ohno; A. Otaka; N. Fujii Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry, 66, 9, 846-857 Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry, 66, 9, 846-857 , 66, 9, 846-857 2008 日本語 公開
Tomita K, Oishi S, Ohno H, Fujii N Tomita K, Oishi S, Ohno H, Fujii N K. Tomita; S. Oishi; H. Ohno; N. Fujii Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists. Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists. Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists Biopolymers, 90, 4, 503-511 Biopolymers, 90, 4, 503-511 Biopolymers - Peptide Science Section, 90, 4, 503-511 2008 英語 公開
Watanabe T, Ueda S, Inuki S, Oishi S, Fujii N, Ohno H Watanabe T, Ueda S, Inuki S, Oishi S, Fujii N, Ohno H T. Watanabe; S. Ueda; S. Inuki; S. Oishi; N. Fujii; H. Ohno One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling. One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling. One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling Chemical communications (Cambridge, England), 43, 4516-4518 Chemical communications (Cambridge, England), 43, 4516-4518 Chemical Communications, 43, 4516-4518 2007/11 英語 公開
Watanabe T, Oishi S, Fujii N, Ohno H Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed hydroarylation of allenes: a highly regioselective carbon-carbon bond formation producing six-membered rings. Gold-catalyzed hydroarylation of allenes: a highly regioselective carbon-carbon bond formation producing six-membered rings. Gold-catalyzed hydroarylation of allenes: A highly regioselective carbon-carbon bond formation producing six-membered rings Organic letters, 9, 23, 4821-4824 Organic letters, 9, 23, 4821-4824 Organic Letters, 9, 23, 4821-4824 2007/11 英語 公開
Ohno H, Iuchi M, Fujii N, Tanaka T Ohno H, Iuchi M, Fujii N, Tanaka T H. Ohno; M. Iuchi; N. Fujii; T. Tanaka Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems. Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems. Zipper-mode double C-H activation: Palladium-catalyzed direct construction of highly-fused heterocyclic systems Organic letters, 9, 23, 4813-4815 Organic letters, 9, 23, 4813-4815 Organic Letters, 9, 23, 4813-4815 2007/11 英語 公開
Narumi T, Tomita K, Inokuchi E, Kobayashi K, Oishi S, Ohno H, Fujii N Narumi T, Tomita K, Inokuchi E, Kobayashi K, Oishi S, Ohno H, Fujii N T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides. Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides. Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides Organic letters, 9, 17, 3465-3468 Organic letters, 9, 17, 3465-3468 Organic Letters, 9, 17, 3465-3468 2007/08 英語 公開
Tomita K, Oishi S, Cluzeau J, Ohno H, Navenot JM, Wang ZX, Peiper SC, Akamatsu M, Fujii N Tomita K, Oishi S, Cluzeau J, Ohno H, Navenot JM, Wang ZX, Peiper SC, Akamatsu M, Fujii N K. Tomita; S. Oishi; J. Cluzeau; H. Ohno; J.-M. Navenot; Z.-X. Wang; S.C. Peiper; M. Akamatsu; N. Fujii SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54. SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54. SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54 Journal of medicinal chemistry, 50, 14, 3222-3228 Journal of medicinal chemistry, 50, 14, 3222-3228 Journal of Medicinal Chemistry, 50, 14, 3222-3228 2007/07 英語 公開
Cluzeau J, Oishi S, Ohno H, Wang Z, Evans B, Peiper SC, Fujii N Cluzeau J, Oishi S, Ohno H, Wang Z, Evans B, Peiper SC, Fujii N J. Cluzeau; S. Oishi; H. Ohno; Z. Wang; B. Evans; S.C. Peiper; N. Fujii Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists. Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists. Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists Organic & biomolecular chemistry, 5, 12, 1915-1923 Organic & biomolecular chemistry, 5, 12, 1915-1923 Organic and Biomolecular Chemistry, 5, 12, 1915-1923 2007/06 英語 公開
Ohno H, Mizutani T, Kadoh Y, Aso A, Miyamura K, Fujii N, Tanaka T Ohno H, Mizutani T, Kadoh Y, Aso A, Miyamura K, Fujii N, Tanaka T H. Ohno; T. Mizutani; Y. Kadoh; A. Aso; K. Miyamura; N. Fujii; T. Tanaka A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes. A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes. A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes The Journal of organic chemistry, 72, 12, 4378-4389 The Journal of organic chemistry, 72, 12, 4378-4389 Journal of Organic Chemistry, 72, 12, 4378-4389 2007/06 英語 公開
Ueda S, Oishi S, Wang ZX, Araki T, Tamamura H, Cluzeau J, Ohno H, Kusano S, Nakashima H, Trent JO, Peiper SC, Fujii N Ueda S, Oishi S, Wang ZX, Araki T, Tamamura H, Cluzeau J, Ohno H, Kusano S, Nakashima H, Trent JO, Peiper SC, Fujii N S. Ueda; S. Oishi; Z.-X. Wang; T. Araki; H. Tamamura; J. Cluzeau; H. Ohno; S. Kusano; H. Nakashima; J.O. Trent; S.C. Peiper; N. Fujii Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities. Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities. Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: Disclosing the importance of side-chain and backbone functionalities Journal of medicinal chemistry, 50, 2, 192-198 Journal of medicinal chemistry, 50, 2, 192-198 Journal of Medicinal Chemistry, 50, 2, 192-198 2007/01 英語 公開
Ohno H, Aso A, Kadoh Y, Fujii N, Tanaka T Ohno H, Aso A, Kadoh Y, Fujii N, Tanaka T H. Ohno; A. Aso; Y. Kadoh; N. Fujii; T. Tanaka Heck-type cyclization of oxime ethers: stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes. Heck-type cyclization of oxime ethers: stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes. Heck-type cyclization of oxime ethers: Stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes Angewandte Chemie (International ed. in English), 46, 33, 6325-6328 Angewandte Chemie (International ed. in English), 46, 33, 6325-6328 Angewandte Chemie - International Edition, 46, 33, 6325-6328 2007 英語 公開
Ohno H, Ohta Y, Oishi S, Fujii N Ohno H, Ohta Y, Oishi S, Fujii N H. Ohno; Y. Ohta; S. Oishi; N. Fujii Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions. Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions. Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions Angewandte Chemie (International ed. in English), 46, 13, 2295-2298 Angewandte Chemie (International ed. in English), 46, 13, 2295-2298 Angewandte Chemie - International Edition, 46, 13, 2295-2298 2007 英語 公開
Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres. Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres. Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres Biopolymers, 88, 2, 272-278 Biopolymers, 88, 2, 272-278 Biopolymers - Peptide Science Section, 88, 2, 272-278 2007 英語 公開
Hamaguchi H, Kosaka S, Ohno H, Fujii N, Tanaka T Hamaguchi H, Kosaka S, Ohno H, Fujii N, Tanaka T H. Hamaguchi; S. Kosaka; H. Ohno; N. Fujii; T. Tanaka Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): Direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes Chemistry (Weinheim an der Bergstrasse, Germany), 13, 6, 1692-1708 Chemistry (Weinheim an der Bergstrasse, Germany), 13, 6, 1692-1708 Chemistry - A European Journal, 13, 6, 1692-1708 2007 英語 公開
Narumi T, Niida A, Tomita K, Oishi S, Otaka A, Ohno H, Fujii N Narumi T, Niida A, Tomita K, Oishi S, Otaka A, Ohno H, Fujii N T. Narumi; A. Niida; K. Tomita; S. Oishi; A. Otaka; H. Ohno; N. Fujii A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres. A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres. A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres Chemical communications (Cambridge, England), 45, 4720-4722 Chemical communications (Cambridge, England), 45, 4720-4722 Chemical Communications, 45, 4720-4722 2006/12 英語 公開
Tomita K, Niida A, Oishi S, Ohno H, Cluzeau J, Navenot JM, Wang ZX, Peiper SC, Fujii N Tomita K, Niida A, Oishi S, Ohno H, Cluzeau J, Navenot JM, Wang ZX, Peiper SC, Fujii N K. Tomita; A. Niida; S. Oishi; H. Ohno; J. Cluzeau; J.-M. Navenot; Z.-x. Wang; S.C. Peiper; N. Fujii Structure-activity relationship study on small peptidic GPR54 agonists. Structure-activity relationship study on small peptidic GPR54 agonists. Structure-activity relationship study on small peptidic GPR54 agonists Bioorganic & medicinal chemistry, 14, 22, 7595-7603 Bioorganic & medicinal chemistry, 14, 22, 7595-7603 Bioorganic and Medicinal Chemistry, 14, 22, 7595-7603 2006/11 英語 公開
Tanaka T, Yamamoto S, Hiramatsu K, Murakami K, Yoshino H, Patra D, Iwata C, Ohno H Tanaka T, Yamamoto S, Hiramatsu K, Murakami K, Yoshino H, Patra D, Iwata C, Ohno H T. Tanaka; S. Yamamoto; K. Hiramatsu; K. Murakami; H. Yoshino; D. Patra; C. Iwata; H. Ohno Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system. Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system. Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system Chemical & pharmaceutical bulletin, 54, 8, 1138-1143 Chemical & pharmaceutical bulletin, 54, 8, 1138-1143 Chemical and Pharmaceutical Bulletin, 54, 8, 1138-1143 2006/08 英語 公開
Niida A, Mizumoto M, Narumi T, Inokuchi E, Oishi S, Ohno H, Otaka A, Kitaura K, Fujii N Niida A, Mizumoto M, Narumi T, Inokuchi E, Oishi S, Ohno H, Otaka A, Kitaura K, Fujii N A. Niida; M. Mizumoto; T. Narumi; E. Inokuchi; S. Oishi; H. Ohno; A. Otaka; K. Kitaura; N. Fujii Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations. Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations. Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations The Journal of organic chemistry, 71, 11, 4118-4129 The Journal of organic chemistry, 71, 11, 4118-4129 Journal of Organic Chemistry, 71, 11, 4118-4129 2006/05 英語 公開
Niida A, Tanigaki H, Inokuchi E, Sasaki Y, Oishi S, Ohno H, Tamamura H, Wang Z, Peiper SC, Kitaura K, Otaka A, Fujii N Niida A, Tanigaki H, Inokuchi E, Sasaki Y, Oishi S, Ohno H, Tamamura H, Wang Z, Peiper SC, Kitaura K, Otaka A, Fujii N A. Niida; H. Tanigaki; E. Inokuchi; Y. Sasaki; S. Oishi; H. Ohno; H. Tamamura; Z. Wang; S.C. Peiper; K. Kitaura; A. Otaka; N. Fujii Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists. Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists. Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-S <sub>N</sub>2′ reactions and their use in the preparation of low-molecule CXCR4 antagonists The Journal of organic chemistry, 71, 10, 3942-3951 The Journal of organic chemistry, 71, 10, 3942-3951 Journal of Organic Chemistry, 71, 10, 3942-3951 2006/05 英語 公開
Ohno H, Kadoh Y, Fujii N, Tanaka T Ohno H, Kadoh Y, Fujii N, Tanaka T H. Ohno; Y. Kadoh; N. Fujii; T. Tanaka Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals. Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals. Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals Organic letters, 8, 5, 947-950 Organic letters, 8, 5, 947-950 Organic Letters, 8, 5, 947-950 2006/03 英語 公開
H. Ohno H. Ohno Ohno H Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations. Yakugaku Zasshi, 125, 12, 899-925 Yakugaku Zasshi, 125, 12, 899-925 Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 125, 12, 899-925 2005/12 日本語 公開
Ohno H Ohno H H. Ohno Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds. Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds. Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds Chemical & pharmaceutical bulletin, 53, 10, 1211-1226 Chemical & pharmaceutical bulletin, 53, 10, 1211-1226 Chemical and Pharmaceutical Bulletin, 53, 10, 1211-1226 2005/10 英語 公開
Ohno H, Mizutani T, Kadoh Y, Miyamura K, Tanaka T Ohno H, Mizutani T, Kadoh Y, Miyamura K, Tanaka T H. Ohno; T. Mizutani; Y. Kadoh; K. Miyamura; T. Tanaka Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: diastereoselective access to bicyclic nitrogen heterocycles. Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: diastereoselective access to bicyclic nitrogen heterocycles. Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: Diastereoselective access to bicyclic nitrogen heterocycles Angewandte Chemie (International ed. in English), 44, 32, 5113-5115 Angewandte Chemie (International ed. in English), 44, 32, 5113-5115 Angewandte Chemie - International Edition, 44, 32, 5113-5115 2005/08 英語 公開
Ohno H, Yamamoto M, Iuchi M, Tanaka T Ohno H, Yamamoto M, Iuchi M, Tanaka T H. Ohno; M. Yamamoto; M. Iuchi; T. Tanaka Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization. Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization. Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization Angewandte Chemie (International ed. in English), 44, 32, 5103-5106 Angewandte Chemie (International ed. in English), 44, 32, 5103-5106 Angewandte Chemie - International Edition, 44, 32, 5103-5106 2005/08 英語 公開
Ohno H, Miyamura K, Mizutani T, Kadoh Y, Takeoka Y, Hamaguchi H, Tanaka T Ohno H, Miyamura K, Mizutani T, Kadoh Y, Takeoka Y, Hamaguchi H, Tanaka T H. Ohno; K. Miyamura; T. Mizutani; Y. Kadoh; Y. Takeoka; H. Hamaguchi; T. Tanaka Palladium(0)-catalyzed tandem cyclization of allenenes: direct construction of tricyclic heterocycles through aromatic C--H activation. Palladium(0)-catalyzed tandem cyclization of allenenes: direct construction of tricyclic heterocycles through aromatic C--H activation. Palladium(0)-catalyzed tandem cyclization of alleneues: Direct construction of tricyclic heterocycles through aromatic C-H activation Chemistry (Weinheim an der Bergstrasse, Germany), 11, 12, 3728-3741 Chemistry (Weinheim an der Bergstrasse, Germany), 11, 12, 3728-3741 Chemistry - A European Journal, 11, 12, 3728-3741 2005/06 英語 公開
Hamaguchi H, Kosaka S, Ohno H, Tanaka T Hamaguchi H, Kosaka S, Ohno H, Tanaka T H. Hamaguchi; S. Kosaka; H. Ohno; T. Tanaka Bromoallenes as allyl dication equivalents in the absence of palladium(0): synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the absence of palladium(0): synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the absence of palladium(0): Synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes Angewandte Chemie (International ed. in English), 44, 10, 1513-1517 Angewandte Chemie (International ed. in English), 44, 10, 1513-1517 Angewandte Chemie - International Edition, 44, 10, 1513-1517 2005/02 英語 公開
Ohno H, Iwasaki H, Eguchi T, Tanaka T Ohno H, Iwasaki H, Eguchi T, Tanaka T H. Ohno; H. Iwasaki; T. Eguchi; T. Tanaka The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring. The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring. The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring Chemical communications (Cambridge, England), 19, 2228-2229 Chemical communications (Cambridge, England), 19, 2228-2229 Chemical Communications, 19, 2228-2229 2004/10 英語 公開
Hayashi K, Rahman SM, Ohno H, Tanaka T, Toyooka N, Nemoto H, Hayashi T Hayashi K, Rahman SM, Ohno H, Tanaka T, Toyooka N, Nemoto H, Hayashi T K. Hayashi; S.M.A. Rahman; H. Ohno; T. Tanaka; N. Toyooka; H. Nemoto; T. Hayashi Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against Herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells. Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against Herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells. Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells Chemical & pharmaceutical bulletin, 52, 8, 1015-1017 Chemical & pharmaceutical bulletin, 52, 8, 1015-1017 Chemical and Pharmaceutical Bulletin, 52, 8, 1015-1017 2004/08 英語 公開
Ohno H, Hamaguchi H, Ohata M, Kosaka S, Tanaka T Ohno H, Hamaguchi H, Ohata M, Kosaka S, Tanaka T H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent. Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent. Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent Journal of the American Chemical Society, 126, 28, 8744-8754 Journal of the American Chemical Society, 126, 28, 8744-8754 Journal of the American Chemical Society, 126, 28, 8744-8754 2004/07 英語 公開
Ohno H, Takeoka Y, Kadoh Y, Miyamura K, Tanaka T Ohno H, Takeoka Y, Kadoh Y, Miyamura K, Tanaka T H. Ohno; Y. Takeoka; Y. Kadoh; K. Miyamura; T. Tanaka Palladium(0)-catalyzed stereoselective cyclization of allenenes: divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes. Palladium(0)-catalyzed stereoselective cyclization of allenenes: divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes. Palladium(0)-catalyzed stereoselective cyclization of allenenes: Divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes The Journal of organic chemistry, 69, 13, 4541-4544 The Journal of organic chemistry, 69, 13, 4541-4544 Journal of Organic Chemistry, 69, 13, 4541-4544 2004/06 英語 公開
Ohno H, Takemoto Y, Fujii N, Tanaka T, Ibuka T Ohno H, Takemoto Y, Fujii N, Tanaka T, Ibuka T H. Ohno; Y. Takemoto; N. Fujii; T. Tanaka; T. Ibukab Stereodivergent synthesis of chiral 2-alkenylaziridines: palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination. Stereodivergent synthesis of chiral 2-alkenylaziridines: palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination. Stereodivergent synthesis of chiral 2-alkenylaziridines: Palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination Chemical & pharmaceutical bulletin, 52, 1, 111-119 Chemical & pharmaceutical bulletin, 52, 1, 111-119 Chemical and Pharmaceutical Bulletin, 52, 1, 111-119 2004/01 英語 公開
Ohno H, Takeoka Y, Miyamura K, Kadoh Y, Tanaka T Ohno H, Takeoka Y, Miyamura K, Kadoh Y, Tanaka T H. Ohno; Y. Takeoka; K. Miyamura; Y. Kadoh; T. Tanaka Novel synthesis of 3-azabicyclo[3.1.0]hexanes by unusual palladium(0)-catalyzed cyclopropanation of allenenes. Novel synthesis of 3-azabicyclo[3.1.0]hexanes by unusual palladium(0)-catalyzed cyclopropanation of allenenes. Novel Synthesis of 3-Azabicyclo[3.1.0]hexanes by Unusual Palladium(0)-Catalyzed Cyclopropanation of Allenenes Organic letters, 5, 25, 4763-4766 Organic letters, 5, 25, 4763-4766 Organic Letters, 5, 25, 4763-4766 2003/12 英語 公開
Ohno H, Miyamura K, Tanaka T, Oishi S, Toda A, Takemoto Y, Fujii N, Ibuka T Ohno H, Miyamura K, Tanaka T, Oishi S, Toda A, Takemoto Y, Fujii N, Ibuka T H. Ohno; K. Miyamura; T. Tanaka; S. Oishi; A. Toda; Y. Takemoto; N. Fujii; T. Ibuka Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system. Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system. Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system The Journal of organic chemistry, 67, 4, 1359-1367 The Journal of organic chemistry, 67, 4, 1359-1367 Journal of Organic Chemistry, 67, 4, 1359-1367 2002/02 英語 公開
H. Ohno H. Ohno Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst Yakugaku Zasshi, 121, 10, 733-741 Yakugaku Zasshi, 121, 10, 733-741 , 121, 10, 733-741 2001 日本語 公開
K. Graf; P.D. Hindenberg; Y. Tokimizu; S. Naoe; M. Rudolph; F. Rominger; H. Ohno; A.S.K. Hashmi K. Graf; P.D. Hindenberg; Y. Tokimizu; S. Naoe; M. Rudolph; F. Rominger; H. Ohno; A.S.K. Hashmi The role of acetylides in dual gold catalysis: A mechanistic investigation of the selectivity difference in the naphthalene synthesis from diynes The role of acetylides in dual gold catalysis: A mechanistic investigation of the selectivity difference in the naphthalene synthesis from diynes ChemCatChem, 6, 1, 199-204 , 6, 1, 199-204 ChemCatChem, 6, 1, 199-204 2014 英語 公開
H. Ohno; H. Chiba; S. Inuki; S. Oishi; N. Fujii H. Ohno; H. Chiba; S. Inuki; S. Oishi; N. Fujii The synthesis of alkaloids using transition-metal-catalyzed intramolecular amination reactions The synthesis of alkaloids using transition-metal-catalyzed intramolecular amination reactions Synlett, 25, 2, 179-192 , 25, 2, 179-192 Synlett, 25, 2, 179-192 2014 英語 公開
Y. Yoshimitsu; J. Miyagaki; S. Oishi; N. Fujii; H. Ohno Y. Yoshimitsu; J. Miyagaki; S. Oishi; N. Fujii; H. Ohno Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis Tetrahedron, 69, 21, 4211-4220 , 69, 21, 4211-4220 Tetrahedron, 69, 21, 4211-4220 2013/05/27 英語 公開
T. Suzuki; Y. Tokimizu; Y. Sakano; R. Katoono; K. Fujiwara; S. Naoe; N. Fujii; H. Ohno T. Suzuki; Y. Tokimizu; Y. Sakano; R. Katoono; K. Fujiwara; S. Naoe; N. Fujii; H. Ohno 5,10-Dihydrobenzo[a]indolo[2,3-c]carbazole: A highly fluorescent disk-shaped electron donor exhibiting dual UVvisNIR and fluorescence spectral changes upon electrolysis 5,10-Dihydrobenzo[a]indolo[2,3-c]carbazole: A highly fluorescent disk-shaped electron donor exhibiting dual UVvisNIR and fluorescence spectral changes upon electrolysis Chemistry Letters, 42, 9, 1001-1003 , 42, 9, 1001-1003 Chemistry Letters, 42, 9, 1001-1003 2013 英語 公開
H. Ohno H. Ohno Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds Israel Journal of Chemistry, 53, 11-12, 869-882 , 53, 11-12, 869-882 Israel Journal of Chemistry, 53, 11-12, 869-882 2013 英語 公開
H. Chiba; Y. Sakai; S. Oishi; N. Fujii; H. Ohno H. Chiba; Y. Sakai; S. Oishi; N. Fujii; H. Ohno Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (-)-quinocarcinamide Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (-)-quinocarcinamide Tetrahedron Letters, 53, 46, 6273-6276 , 53, 46, 6273-6276 Tetrahedron Letters, 53, 46, 6273-6276 2012/11/14 英語 公開
R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; E. Kodama; M. Matsuoka; N. Fujii R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; E. Kodama; M. Matsuoka; N. Fujii Development and application of fluorescent SDF-1 derivatives Development and application of fluorescent SDF-1 derivatives Future Medicinal Chemistry, 4, 7, 837-844 , 4, 7, 837-844 Future Medicinal Chemistry, 4, 7, 837-844 2012/05 英語 公開
Z. Hou; Y. Suzuki; S. Oishi; N. Fujii; H. Ohno Z. Hou; Y. Suzuki; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of aminomethylated azaindoles and corresponding pyrrole-fused derivatives by copper-catalyzed domino multicomponent coupling and cyclization Efficient synthesis of aminomethylated azaindoles and corresponding pyrrole-fused derivatives by copper-catalyzed domino multicomponent coupling and cyclization Tetrahedron, 68, 6, 1695-1703 , 68, 6, 1695-1703 Tetrahedron, 68, 6, 1695-1703 2012/02/11 英語 公開
Y. Suzuki; S. Naoe; S. Oishi; N. Fujii; H. Ohno Y. Suzuki; S. Naoe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed three-component annulation: Efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones Gold-catalyzed three-component annulation: Efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones Organic Letters, 14, 1, 326-329 , 14, 1, 326-329 Organic Letters, 14, 1, 326-329 2012/01/06 英語 公開
H. Ohno; M. Yamamoto; M. Iuchi; N. Fujii; T. Tanaka H. Ohno; M. Yamamoto; M. Iuchi; N. Fujii; T. Tanaka Palladium-catalyzed construction of polycyclic heterocycles by an alkyne insertion and direct arylation cascade Palladium-catalyzed construction of polycyclic heterocycles by an alkyne insertion and direct arylation cascade Synthesis, 16, 2567-2578 , 16, 2567-2578 Synthesis, 16, 2567-2578 2011/08 英語 公開
Y. Tokimizu; Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Y. Tokimizu; Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Direct synthesis of highly fused perimidines by copper(I)-catalyzed hydroamination of 2-ethynylbenzaldehydes Direct synthesis of highly fused perimidines by copper(I)-catalyzed hydroamination of 2-ethynylbenzaldehydes Tetrahedron, 67, 29, 5168-5175 , 67, 29, 5168-5175 Tetrahedron, 67, 29, 5168-5175 2011/07/22 英語 公開
H. Iwasaki; N. Tsutsui; T. Eguchi; H. Ohno; M. Yamashita; T. Tanaka H. Iwasaki; N. Tsutsui; T. Eguchi; H. Ohno; M. Yamashita; T. Tanaka A novel samarium(II)-mediated tandem spirocyclization onto an aromatic ring A novel samarium(II)-mediated tandem spirocyclization onto an aromatic ring Tetrahedron Letters, 52, 15, 1770-1772 , 52, 15, 1770-1772 Tetrahedron Letters, 52, 15, 1770-1772 2011 英語 公開
S. Inuki; S. Oishi; N. Fujii; H. Ohno S. Inuki; S. Oishi; N. Fujii; H. Ohno Total synthesis of ((±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group (Oroganic Letters (2008) 10 (5239)) Total synthesis of ((±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group (Oroganic Letters (2008) 10 (5239)) Organic Letters, 13, 8, 2145- , 13, 8, 2145- Organic Letters, 13, 8, 2145- 2011 英語 公開
S. Oishi; K. Watanabe; S. Ito; M. Tanaka; H. Nishikawa; H. Ohno; K. Shimane; K. Izumi; Y. Sakagami; E.N. Kodama; M. Matsuoka; A. Asai; N. Fujii S. Oishi; K. Watanabe; S. Ito; M. Tanaka; H. Nishikawa; H. Ohno; K. Shimane; K. Izumi; Y. Sakagami; E.N. Kodama; M. Matsuoka; A. Asai; N. Fujii Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants MedChemComm, 1, 4, 276-281 , 1, 4, 276-281 MedChemComm, 1, 4, 276-281 2010/10 英語 公開
K. Hirano; Y. Inaba; T. Watanabe; S. Oishi; N. Fujii; H. Ohno K. Hirano; Y. Inaba; T. Watanabe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed intramolecular alkyne cycloisomerization cascade: Direct synthesis of aryl-annulated[a]carbazoles from aniline-substituted diethynylarenes Gold-catalyzed intramolecular alkyne cycloisomerization cascade: Direct synthesis of aryl-annulated[a]carbazoles from aniline-substituted diethynylarenes Advanced Synthesis and Catalysis, 352, 2/3, 368-372 , 352, 2/3, 368-372 Advanced Synthesis and Catalysis, 352, 2/3, 368-372 2010/02 英語 公開
T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic Tetrahedron, 64, 19, 4332-4346 , 64, 19, 4332-4346 Tetrahedron, 64, 19, 4332-4346 2008/05/05 英語 公開
M. Tanaka; S. Oishi; H. Ohno; N. Fujii M. Tanaka; S. Oishi; H. Ohno; N. Fujii A novel oxazolidine linker for the synthesis of peptide aldehydes A novel oxazolidine linker for the synthesis of peptide aldehydes International Journal of Peptide Research and Therapeutics, 13, 1-2, 271-279 , 13, 1-2, 271-279 International Journal of Peptide Research and Therapeutics, 13, 1-2, 271-279 2007/06 英語 公開
H. Ohno; Y. Ohta; S. Oishi; N. Fujii H. Ohno; Y. Ohta; S. Oishi; N. Fujii Erratum: Direct synthesis of 2-(aminomethyl)-indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions (Angewandte Chemie - International Edition (2007) 46, (2295-2298) DOI: 10.1002/anie.200604342) Erratum: Direct synthesis of 2-(aminomethyl)-indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions (Angewandte Chemie - International Edition (2007) 46, (2295-2298) DOI: 10.1002/anie.200604342) Angewandte Chemie - International Edition, 46, 18, 3173- , 46, 18, 3173- Angewandte Chemie - International Edition, 46, 18, 3173- 2007 英語 公開
H. Ohno H. Ohno Vinylaziridines in Organic Synthesis Vinylaziridines in Organic Synthesis Aziridines and Epoxides in Organic Synthesis, 37-71 , 37-71 Aziridines and Epoxides in Organic Synthesis, 37-71 2006 英語 公開
T. Tanaka; K. Hiramatsu; Y. Kobayashi; H. Ohno T. Tanaka; K. Hiramatsu; Y. Kobayashi; H. Ohno Chemo- and stereoselectivity in titanium-mediated regioselective ring-opening reaction of epoxides at the more substituted carbon Chemo- and stereoselectivity in titanium-mediated regioselective ring-opening reaction of epoxides at the more substituted carbon Tetrahedron, 61, 28, 6726-6742 , 61, 28, 6726-6742 Tetrahedron, 61, 28, 6726-6742 2005 英語 公開
大野 浩章 大野 浩章 Asymmetric construction of quaternary carbon centers by allyltitanium-mediated stereospecific ring-opening reaction of 2,3-epoxy alcohols. Asymmetric construction of quaternary carbon centers by allyltitanium-mediated stereospecific ring-opening reaction of 2,3-epoxy alcohols. Tetrahedron Lett. 45/1, 75–78, 45, 1, 75-78 , 45, 1, 75-78 Tetrahedron Lett. 45/1, 75–78, 45, 1, 75-78 2004 英語 公開
H. Ohno; K. Hiramatsu; T. Tanaka H. Ohno; K. Hiramatsu; T. Tanaka Asymmetric construction of quaternary carbon centers by titanium-mediated stereospecific allylation of 2,3-epoxy alcohol derivatives Asymmetric construction of quaternary carbon centers by titanium-mediated stereospecific allylation of 2,3-epoxy alcohol derivatives Tetrahedron Letters, 45, 1, 75-78 , 45, 1, 75-78 Tetrahedron Letters, 45, 1, 75-78 2004 英語 公開
H. Ohno; M. Okumura; S.-I. Maeda; H. Iwasaki; R. Wakayama; T. Tanaka H. Ohno; M. Okumura; S.-I. Maeda; H. Iwasaki; R. Wakayama; T. Tanaka Samarium(II)-promoted radical spirocyclization onto an aromatic ring Samarium(II)-promoted radical spirocyclization onto an aromatic ring Journal of Organic Chemistry, 68, 20, 7722-7732 , 68, 20, 7722-7732 Journal of Organic Chemistry, 68, 20, 7722-7732 2003/10/03 英語 公開
H. Ohno; R. Wakayama; S.-I. Maeda; H. Iwasaki; M. Okumura; C. Iwata; H. Mikamiyama; T. Tanaka H. Ohno; R. Wakayama; S.-I. Maeda; H. Iwasaki; M. Okumura; C. Iwata; H. Mikamiyama; T. Tanaka Radical cyclization by Ipso substitution of the methoxy group: Considerable effect of HMPA on samarium-mediated cyclization Radical cyclization by Ipso substitution of the methoxy group: Considerable effect of HMPA on samarium-mediated cyclization Journal of Organic Chemistry, 68, 15, 5909-5916 , 68, 15, 5909-5916 Journal of Organic Chemistry, 68, 15, 5909-5916 2003/07/25 英語 公開
H. Ohno; H. Hamaguchi; M. Ohata; T. Tanaka H. Ohno; H. Hamaguchi; M. Ohata; T. Tanaka Bromoallenes as synthetic equivalents of allyl dications: Synthesis of medium-sized nitrogen heterocycles through the cyclization of bromoallenes in the presence of a palladium(0) catalyst and an alcohol Bromoallenes as synthetic equivalents of allyl dications: Synthesis of medium-sized nitrogen heterocycles through the cyclization of bromoallenes in the presence of a palladium(0) catalyst and an alcohol Angewandte Chemie - International Edition, 42, 15, 1749-1753 , 42, 15, 1749-1753 Angewandte Chemie - International Edition, 42, 15, 1749-1753 2003 英語 公開
H. Ohno; K. Miyamura; Y. Takeoka; T. Tanaka H. Ohno; K. Miyamura; Y. Takeoka; T. Tanaka Palladium(0)-catalyzed tandem cyclization of allenenes Palladium(0)-catalyzed tandem cyclization of allenenes Angewandte Chemie - International Edition, 42, 23, 2647-2650 , 42, 23, 2647-2650 Angewandte Chemie - International Edition, 42, 23, 2647-2650 2003 英語 公開
H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka Novel synthesis of azocine, azepine, oxocine, and oxepine derivatives by palladium-catalyzed medium-ring formation from bromoallenes Novel synthesis of azocine, azepine, oxocine, and oxepine derivatives by palladium-catalyzed medium-ring formation from bromoallenes Heterocycles, 61, 65-68 , 61, 65-68 Heterocycles, 61, 65-68 2003 英語 公開
H. Ohno; K. Ando; H. Hamaguchi; Y. Takeoka; T. Tanaka H. Ohno; K. Ando; H. Hamaguchi; Y. Takeoka; T. Tanaka A highly cis-selective synthesis of 2-ethynylaziridines by intramolecular amination of chiral bromoallenes: Improvement of stereoselectivity based on the computational investigation A highly cis-selective synthesis of 2-ethynylaziridines by intramolecular amination of chiral bromoallenes: Improvement of stereoselectivity based on the computational investigation Journal of the American Chemical Society, 124, 51, 15255-15266 , 124, 51, 15255-15266 Journal of the American Chemical Society, 124, 51, 15255-15266 2002/12/25 英語 公開
M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka; Y. Takemoto M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka; Y. Takemoto Asymmetric synthesis of β<sup>2,3</sup>-amino acids by InI-Pd(0)-promoted metalation and addition of chiral 2-vinylaziridines Asymmetric synthesis of β<sup>2,3</sup>-amino acids by InI-Pd(0)-promoted metalation and addition of chiral 2-vinylaziridines Tetrahedron, 58, 26, 5231-5239 , 58, 26, 5231-5239 Tetrahedron, 58, 26, 5231-5239 2002/06/24 英語 公開
H. Ohno; S.-I. Maeda; M. Okumura; R. Wakayama; T. Tanaka H. Ohno; S.-I. Maeda; M. Okumura; R. Wakayama; T. Tanaka The first samarium(II)-mediated stereoselective spirocyclization onto an aromatic ring The first samarium(II)-mediated stereoselective spirocyclization onto an aromatic ring Chemical Communications, 4, 316-317 , 4, 316-317 Chemical Communications, 4, 316-317 2002 英語 公開
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka Stereoselective synthesis of chiral 2,3-cis-2-ethynylaziridines by base-mediated intramolecular amination of bromoallenes Stereoselective synthesis of chiral 2,3-cis-2-ethynylaziridines by base-mediated intramolecular amination of bromoallenes Organic Letters, 3, 15, 2269-2271 , 3, 15, 2269-2271 Organic Letters, 3, 15, 2269-2271 2001/07/26 英語 公開
H. Ohno; M. Anzai; A. Toda; S. Ohishi; N. Fujii; T. Tanaka; Y. Takemoto; T. Ibuka H. Ohno; M. Anzai; A. Toda; S. Ohishi; N. Fujii; T. Tanaka; Y. Takemoto; T. Ibuka Stereoselective synthesis of 2-alkenylaziridines and 2-alkenylazetidines by palladium-catalyzed intramolecular amination of α- and β-amino allenes Stereoselective synthesis of 2-alkenylaziridines and 2-alkenylazetidines by palladium-catalyzed intramolecular amination of α- and β-amino allenes Journal of Organic Chemistry, 66, 14, 4904-4914 , 66, 14, 4904-4914 Journal of Organic Chemistry, 66, 14, 4904-4914 2001/07/13 英語 公開
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka 2-Ethynylaziridines as chiral carbon nucleophiles: Stereoselective synthesis of 1,3-amino alcohols with three stereocenters via allenylindium reagents bearing a protected amino group 2-Ethynylaziridines as chiral carbon nucleophiles: Stereoselective synthesis of 1,3-amino alcohols with three stereocenters via allenylindium reagents bearing a protected amino group Journal of Organic Chemistry, 66, 5, 1867-1875 , 66, 5, 1867-1875 Journal of Organic Chemistry, 66, 5, 1867-1875 2001/03/09 英語 公開
Y. Takemoto; M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka Y. Takemoto; M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka Stereoselective synthesis of nonracemic 1,3-amino alcohols from chiral 2-vinylaziridines by InI-Pd(0)-promoted metalation Stereoselective synthesis of nonracemic 1,3-amino alcohols from chiral 2-vinylaziridines by InI-Pd(0)-promoted metalation Tetrahedron Letters, 42, 9, 1725-1728 , 42, 9, 1725-1728 Tetrahedron Letters, 42, 9, 1725-1728 2001/02/26 英語 公開
S.M. Abdur Rahman; H. Ohno; H. Yoshino; N. Satoh; M. Tsukaguchi; K. Murakami; C. Iwata; N. Maezaki; T. Tanaka S.M. Abdur Rahman; H. Ohno; H. Yoshino; N. Satoh; M. Tsukaguchi; K. Murakami; C. Iwata; N. Maezaki; T. Tanaka A model study for the total synthesis of (±)-scopadulin: Stereoselective construction of the A/B ring system with desired functionalities A model study for the total synthesis of (±)-scopadulin: Stereoselective construction of the A/B ring system with desired functionalities Tetrahedron, 57, 1, 127-134 , 57, 1, 127-134 Tetrahedron, 57, 1, 127-134 2001 英語 公開
S.M.A. Rahman; H. Ohno; T. Tanaka S.M.A. Rahman; H. Ohno; T. Tanaka Improved method of an unusual conversion of aliphatic amines into alcohols Improved method of an unusual conversion of aliphatic amines into alcohols Tetrahedron Letters, 42, 45, 8007-8010 , 42, 45, 8007-8010 Tetrahedron Letters, 42, 45, 8007-8010 2001 英語 公開
S.M.A. Rahman; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki; T. Tanaka S.M.A. Rahman; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki; T. Tanaka Total synthesis of (±)-scopadulin Total synthesis of (±)-scopadulin Journal of Organic Chemistry, 66, 14, 4831-4840 , 66, 14, 4831-4840 Journal of Organic Chemistry, 66, 14, 4831-4840 2001 英語 公開
T. Tanaka; K. Murakami; A. Kanda; D. Patra; S. Yamamoto; N. Satoh; S.-W. Kim; S.M.A. Rahman; H. Ohno; C. Iwata T. Tanaka; K. Murakami; A. Kanda; D. Patra; S. Yamamoto; N. Satoh; S.-W. Kim; S.M.A. Rahman; H. Ohno; C. Iwata Total synthesis of (±)-stemodinone via an efficient ring-exchange strategy Total synthesis of (±)-stemodinone via an efficient ring-exchange strategy Journal of Organic Chemistry, 66, 21, 7107-7112 , 66, 21, 7107-7112 Journal of Organic Chemistry, 66, 21, 7107-7112 2001 英語 公開
S.M.A. Rahman; T. Tanaka; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki S.M.A. Rahman; T. Tanaka; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki The first total synthesis of (±)-scopadulin, an antiviral aphidicolane diterpene The first total synthesis of (±)-scopadulin, an antiviral aphidicolane diterpene Organic Letters, 3, 4, 619-621 , 3, 4, 619-621 Organic Letters, 3, 4, 619-621 2001 英語 公開
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka Umpolung of chiral 2-ethynylaziridines: Indium(I)-mediated stereoselective synthesis of nonracemic 1,3-amino alcohols bearing three chiral centers, catalyzed by palladium(0) Umpolung of chiral 2-ethynylaziridines: Indium(I)-mediated stereoselective synthesis of nonracemic 1,3-amino alcohols bearing three chiral centers, catalyzed by palladium(0) Organic Letters, 2, 14, 2161-2163 , 2, 14, 2161-2163 Organic Letters, 2, 14, 2161-2163 2000/07/13 英語 公開
H. Ohno; A. Toda; S. Oishi; T. Tanaka; Y. Takemoto; N. Fujii; T. Ibuka H. Ohno; A. Toda; S. Oishi; T. Tanaka; Y. Takemoto; N. Fujii; T. Ibuka Novel synthesis of chiral terminal allenes via palladium(o)catalyzed reduction of mesylates of 2-bromoalk-2-en-1-ols bearing a protected amino group, using diethylzinc Novel synthesis of chiral terminal allenes via palladium(o)catalyzed reduction of mesylates of 2-bromoalk-2-en-1-ols bearing a protected amino group, using diethylzinc Tetrahedron Letters, 41, 26, 5131-5134 , 41, 26, 5131-5134 Tetrahedron Letters, 41, 26, 5131-5134 2000/06/24 英語 公開
H. Ohno; A. Toda; N. Fujii; Y. Takemoto; T. Tanaka; T. Ibuka H. Ohno; A. Toda; N. Fujii; Y. Takemoto; T. Tanaka; T. Ibuka Stereoselective synthesis of chiral amino allenes by organocopper- mediated anti-S(N)2\\'-substitution reaction of chiral ethynylaziridines Stereoselective synthesis of chiral amino allenes by organocopper- mediated anti-S(N)2\\'-substitution reaction of chiral ethynylaziridines Tetrahedron, 56, 18, 2811-2820 , 56, 18, 2811-2820 Tetrahedron, 56, 18, 2811-2820 2000/04/28 英語 公開
S.M.A. Rahman; H. Ohno; N. Maezaki; C. Iwata; T. Tanaka S.M.A. Rahman; H. Ohno; N. Maezaki; C. Iwata; T. Tanaka Efficient one-step conversion of primary aliphatic amines into primary alcohols: Application to a model study for the total synthesis of (±)-scopadulin Efficient one-step conversion of primary aliphatic amines into primary alcohols: Application to a model study for the total synthesis of (±)-scopadulin Organic Letters, 2, 18, 2893-2895 , 2, 18, 2893-2895 Organic Letters, 2, 18, 2893-2895 2000 英語 公開
K. Ando; T. Oishi; M. Hirama; H. Ohno; T. Ibuka K. Ando; T. Oishi; M. Hirama; H. Ohno; T. Ibuka Z-selective Horner-Wadsworth-Emmons reaction of ethyl (diarylphosphono)acetates using sodium iodide and DBU Z-selective Horner-Wadsworth-Emmons reaction of ethyl (diarylphosphono)acetates using sodium iodide and DBU Journal of Organic Chemistry, 65, 15, 4745-4749 , 65, 15, 4745-4749 Journal of Organic Chemistry, 65, 15, 4745-4749 2000 英語 公開
T. Tanaka; R. Wakayama; S.-I. Maeda; H. Mikamiyama; N. Maezaki; H. Ohno T. Tanaka; R. Wakayama; S.-I. Maeda; H. Mikamiyama; N. Maezaki; H. Ohno Unusual radical ipso-substitution reaction of an aromatic methoxy group induced by tris(trimethylsilyl)silane-AIBN or SmI<sub>2</sub> Unusual radical ipso-substitution reaction of an aromatic methoxy group induced by tris(trimethylsilyl)silane-AIBN or SmI<sub>2</sub> Chemical Communications, 14, 1287-1288 , 14, 1287-1288 Chemical Communications, 14, 1287-1288 2000 英語 公開
Ohno, H; Toda, A; Takemoto, Y; Fujii, N; Ibuka, T Ohno, H; Toda, A; Takemoto, Y; Fujii, N; Ibuka, T Convenient syntheses of chiral 3-substituted 2-ethynylaziridines Convenient syntheses of chiral 3-substituted 2-ethynylaziridines JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 20, 2949-2962 , 20, 2949-2962 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 20, 2949-2962 1999/10/21 英語 公開
M. Anzai; A. Toda; H. Ohno; Y. Takemoto; N. Fujii; T. Ibuka M. Anzai; A. Toda; H. Ohno; Y. Takemoto; N. Fujii; T. Ibuka Palladium-catalyzed regio- and stereoselective synthesis of N-protected 2,4-dialkylated azacyclobutanes from amino allenes Palladium-catalyzed regio- and stereoselective synthesis of N-protected 2,4-dialkylated azacyclobutanes from amino allenes Tetrahedron Letters, 40, 41, 7393-7397 , 40, 41, 7393-7397 Tetrahedron Letters, 40, 41, 7393-7397 1999/10/08 英語 公開
Ishii, K; Ohno, H; Takemoto, Y; Osawa, E; Yamaoka, Y; Fujii, N; Ibuka, T Ishii, K; Ohno, H; Takemoto, Y; Osawa, E; Yamaoka, Y; Fujii, N; Ibuka, T Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N arylsulfonylaminoalk-2-en-1-ols Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N arylsulfonylaminoalk-2-en-1-ols JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 15, 2155-2163 , 15, 2155-2163 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 15, 2155-2163 1999/08/07 英語 公開
H. Ohno; A. Toda; Y. Miwa; T. Taga; E. Osawa; Y. Yamaoka; N. Fujii; T. Ibuka H. Ohno; A. Toda; Y. Miwa; T. Taga; E. Osawa; Y. Yamaoka; N. Fujii; T. Ibuka First palladium-catalyzed aziridination reaction of amino allenes First palladium-catalyzed aziridination reaction of amino allenes Journal of Organic Chemistry, 64, 9, 2992-2993 , 64, 9, 2992-2993 Journal of Organic Chemistry, 64, 9, 2992-2993 1999/04/30 英語 公開
H. Ohno; A. Toda; N. Fujii; Y. Miwa; T. Taga; Y. Yamaoka; E. Osawa; T. Ibuka H. Ohno; A. Toda; N. Fujii; Y. Miwa; T. Taga; Y. Yamaoka; E. Osawa; T. Ibuka Sterically congested chiral activated aziridines: Synthesis of both 2,3- cis-and 2,3-Trans-2-alkenyl-3-alkylaziridines from common intermediates Sterically congested chiral activated aziridines: Synthesis of both 2,3- cis-and 2,3-Trans-2-alkenyl-3-alkylaziridines from common intermediates Tetrahedron Letters, 40, 7, 1331-1334 , 40, 7, 1331-1334 Tetrahedron Letters, 40, 7, 1331-1334 1999/02/12 英語 公開
Ishii, K; Ohno, H; Takemoto, Y; Ibuka, T Ishii, K; Ohno, H; Takemoto, Y; Ibuka, T Selective synthesis of nonracemic 3-pyrrolines and 2,3-cis-2-vinylaziridines from (Z)-amino allylic alcohols: A new synthetic route to chiral 3,4-dehydroproline Selective synthesis of nonracemic 3-pyrrolines and 2,3-cis-2-vinylaziridines from (Z)-amino allylic alcohols: A new synthetic route to chiral 3,4-dehydroproline SYNLETT, 2, 228-230 , 2, 228-230 SYNLETT, 2, 228-230 1999/02 英語 公開
H. Ohno; A. Toda; Y. Miwa; T. Taga; N. Fujii; T. Ibuka H. Ohno; A. Toda; Y. Miwa; T. Taga; N. Fujii; T. Ibuka Synthesis of chiral amino allenes via an organocyanocuprate-mediated ring-opening reaction of enantiopure ethynylaziridines Synthesis of chiral amino allenes via an organocyanocuprate-mediated ring-opening reaction of enantiopure ethynylaziridines Tetrahedron Letters, 40, 2, 349-352 , 40, 2, 349-352 Tetrahedron Letters, 40, 2, 349-352 1999/01/08 英語 公開
H. Tamamura; M. Yamashita; Y. Nakajima; K. Sakano; A. Otaka; H. Ohno; T. Ibuka; N. Fujii H. Tamamura; M. Yamashita; Y. Nakajima; K. Sakano; A. Otaka; H. Ohno; T. Ibuka; N. Fujii Regiospecific ring-opening reactions of β-aziridinyl ct, β-enoates with acids: Application to the stereoselective synthesis of a couple of diastereoisomeric (Zi)-alkene dipeptide isosteres from a single β-aziridinyl a, β-enoate and to the convenient prepa Regiospecific ring-opening reactions of β-aziridinyl ct, β-enoates with acids: Application to the stereoselective synthesis of a couple of diastereoisomeric (Zi)-alkene dipeptide isosteres from a single β-aziridinyl a, β-enoate and to the convenient prepa Journal of the Chemical Society - Perkin Transactions 1, 20, 2983-2996 , 20, 2983-2996 Journal of the Chemical Society - Perkin Transactions 1, 20, 2983-2996 1999 英語 公開
H. Ohno; A. Toda; N. Fujii; T. Ibuka H. Ohno; A. Toda; N. Fujii; T. Ibuka A convenient synthesis of activated enantiomerically pure 2- ethynylaziridines A convenient synthesis of activated enantiomerically pure 2- ethynylaziridines Tetrahedron Asymmetry, 9, 22, 3929-3933 , 9, 22, 3929-3933 Tetrahedron Asymmetry, 9, 22, 3929-3933 1998/11/27 英語 公開
Ohno, H; Ishii, K; Honda, A; Tamamura, H; Fujii, N; Takemoto, Y; Ibuka, T Ohno, H; Ishii, K; Honda, A; Tamamura, H; Fujii, N; Takemoto, Y; Ibuka, T A 2,3-cis-selective synthesis of aziridines bearing a vinyl group from allyl methyl carbonates and allyl mesylates A 2,3-cis-selective synthesis of aziridines bearing a vinyl group from allyl methyl carbonates and allyl mesylates JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 22, 3703-3716 , 22, 3703-3716 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 22, 3703-3716 1998/11/21 英語 公開
A. Honda; H. Ohno; N. Mimura; T. Ibuka A. Honda; H. Ohno; N. Mimura; T. Ibuka Rhodium(I)- or iridium(I)-mediated equilibrated reactions of activated 2,3-cis- and trans-3-alkyl-2-vinylaziridines Rhodium(I)- or iridium(I)-mediated equilibrated reactions of activated 2,3-cis- and trans-3-alkyl-2-vinylaziridines Synlett, 9, 969-+ , 9, 969-+ Synlett, 9, 969-+ 1998/09 英語 公開
A. Toda; H. Aoyama; N. Mimura; H. Ohno; N. Fujii; T. Ibuka A. Toda; H. Aoyama; N. Mimura; H. Ohno; N. Fujii; T. Ibuka Reactions of n-arylsulfonyl-2,3-cis- and n-arylsulfonyl-2,3-frans-3-alkyl-2-vinylaziridines with organocopper reagents: importance of 2,3-cis-stereochemistry in controlling regio- and stereoselectivity Reactions of n-arylsulfonyl-2,3-cis- and n-arylsulfonyl-2,3-frans-3-alkyl-2-vinylaziridines with organocopper reagents: importance of 2,3-cis-stereochemistry in controlling regio- and stereoselectivity Journal of Organic Chemistry, 63, 20, 7053-7061 , 63, 20, 7053-7061 Journal of Organic Chemistry, 63, 20, 7053-7061 1998 英語 公開
T. Ibuka; N. Mimura; H. Ohno; K. Nakai; M. Akaji; H. Habashita; H. Tamamura; Y. Miwa; T. Taga; N. Fujii; Y. Yamamoto T. Ibuka; N. Mimura; H. Ohno; K. Nakai; M. Akaji; H. Habashita; H. Tamamura; Y. Miwa; T. Taga; N. Fujii; Y. Yamamoto Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an α,β-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsvdfonyl) 2-Enoates over the Other Three Stereoisomers Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an α,β-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsvdfonyl) 2-Enoates over the Other Three Stereoisomers Journal of Organic Chemistry, 62, 9, 2982-2991 , 62, 9, 2982-2991 Journal of Organic Chemistry, 62, 9, 2982-2991 1997/05/02 英語 公開
H. Ohno; N. Mimura; A. Otaka; H. Tamamura; N. Fujii; T. Ibuka; I. Shimizu; A. Satake; Y. Yamamoto H. Ohno; N. Mimura; A. Otaka; H. Tamamura; N. Fujii; T. Ibuka; I. Shimizu; A. Satake; Y. Yamamoto Palladium-catalyzed reductive ring opening with formic acid of aziridines bearing an α,β-unsaturated ester group Palladium-catalyzed reductive ring opening with formic acid of aziridines bearing an α,β-unsaturated ester group Tetrahedron, 53, 38, 12933-12946 , 53, 38, 12933-12946 Tetrahedron, 53, 38, 12933-12946 1997 英語 公開
T. Ibuka; N. Mimura; H. Aoyama; M. Akaji; H. Ohno; Y. Miwa; T. Taga; K. Nakai; H. Tamamura; N. Fujii; Y. Yamamoto T. Ibuka; N. Mimura; H. Aoyama; M. Akaji; H. Ohno; Y. Miwa; T. Taga; K. Nakai; H. Tamamura; N. Fujii; Y. Yamamoto A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres Journal of Organic Chemistry, 62, 4, 999-1015 , 62, 4, 999-1015 Journal of Organic Chemistry, 62, 4, 999-1015 1997 英語 公開
H. Aoyama; N. Mimura; H. Ohno; K. Ishii; A. Toda; H. Tamamura; A. Otaka; N. Fujii; T. Ibuka H. Aoyama; N. Mimura; H. Ohno; K. Ishii; A. Toda; H. Tamamura; A. Otaka; N. Fujii; T. Ibuka Regio- and stereoselectivity in reactions of 2,3-cis- and trans-3-alkyl-2-vinylaziridines with organocopper reagents: Importance of 2,3-cis-stereochemistry in controlling selectivity Regio- and stereoselectivity in reactions of 2,3-cis- and trans-3-alkyl-2-vinylaziridines with organocopper reagents: Importance of 2,3-cis-stereochemistry in controlling selectivity Tetrahedron Letters, 38, 42, 7383-7386 , 38, 42, 7383-7386 Tetrahedron Letters, 38, 42, 7383-7386 1997 英語 公開
H. Tamamura; M. Yamashita; H. Muramatsu; H. Ohno; T. Ibuka; A. Otaka; N. Fujii H. Tamamura; M. Yamashita; H. Muramatsu; H. Ohno; T. Ibuka; A. Otaka; N. Fujii Regiospecific ring-opening reactions of aziridines bearing an α,β-unsaturated ester group with trifluoroacetic acid or methanesulfonic acid: Application to the stereoselective synthesis of (E)-alkene dipeptide isosteres Regiospecific ring-opening reactions of aziridines bearing an α,β-unsaturated ester group with trifluoroacetic acid or methanesulfonic acid: Application to the stereoselective synthesis of (E)-alkene dipeptide isosteres Chemical Communications, 23, 2327-2328 , 23, 2327-2328 Chemical Communications, 23, 2327-2328 1997 英語 公開

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タイトル言語:
講演・口頭発表等
タイトル タイトル(日本語) タイトル(英語) 会議名 会議名(日本語) 会議名(英語) 主催者 主催者(日本語) 主催者(英語) 開催年月日 記述言語 会議種別 公開
⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤[招待あり] ⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤ [招待あり] 千葉大学大学院 薬学研究院 特別講義 千葉大学大学院 薬学研究院 特別講義 2018/06/08 日本語 口頭発表(招待・特別) 公開
⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤[招待あり] ⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤ [招待あり] 岡山大学医歯薬学総合研究科 特別講演会 岡山大学医歯薬学総合研究科 特別講演会 2017/09/29 日本語 口頭発表(招待・特別) 公開
⾦触媒を⽤いた複素環⾻格構築法の開発と応⽤[招待あり] ⾦触媒を⽤いた複素環⾻格構築法の開発と応⽤ [招待あり] 中外製薬 講演会 中外製薬 講演会 2017/09/13 日本語 口頭発表(招待・特別) 公開
金触媒によるアルカロイド型骨格の構築と全合成研究[招待あり] 金触媒によるアルカロイド型骨格の構築と全合成研究 [招待あり] 第37回有機合成若手セミナー 第37回有機合成若手セミナー 2017/08/09 日本語 口頭発表(招待・特別) 公開
Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations[招待あり] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations [招待あり] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations [招待あり] Nordic/Kyoto OMCOS 2017 Nordic/Kyoto OMCOS 2017 Nordic/Kyoto OMCOS 2017 2017/06/24 英語 口頭発表(招待・特別) 公開
金触媒によるアルキンの活性化を基盤とした骨格構築反応の開発と応用[招待あり] 金触媒によるアルキンの活性化を基盤とした骨格構築反応の開発と応用 [招待あり] 明治薬科大学 特別講義 明治薬科大学 特別講義 2016/12/19 日本語 口頭発表(招待・特別) 公開
金触媒を用いた反応の開発と応用[招待あり] 金触媒を用いた反応の開発と応用 [招待あり] 塩野義製薬(株) 創薬化学研究所セミナー 塩野義製薬(株) 創薬化学研究所セミナー 2016/10/03 日本語 口頭発表(招待・特別) 公開
多重結合の連続活性化を用いた骨格構築反応の開発と応用[招待あり] 多重結合の連続活性化を用いた骨格構築反応の開発と応用 [招待あり] 近畿大学薬学研究科 大学院特別講義 近畿大学薬学研究科 大学院特別講義 2016/04/23 日本語 口頭発表(招待・特別) 公開
Efficient Construction of Heterocyclic Scaffolds and Its Application[招待あり] Efficient Construction of Heterocyclic Scaffolds and Its Application [招待あり] Efficient Construction of Heterocyclic Scaffolds and Its Application [招待あり] AGORA Bayer Meeting 2016 AGORA Bayer Meeting 2016 AGORA Bayer Meeting 2016 2016/04/15 英語 口頭発表(招待・特別) 公開
Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles[招待あり] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles [招待あり] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles [招待あり] Pacifichem Pacifichem Pacifichem 2015/12/15 英語 口頭発表(招待・特別) 公開
金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用[招待あり] 金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用 [招待あり] 名城大学特別講演会 名城大学特別講演会 2015/12/04 日本語 口頭発表(招待・特別) 公開
アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用[招待あり] アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用 [招待あり] 京大有機金属化学若手勉強会 京大有機金属化学若手勉強会 2015/10/31 日本語 口頭発表(招待・特別) 公開
アルキンの活性化を基盤とする連続反応の開発と応用[招待あり] アルキンの活性化を基盤とする連続反応の開発と応用 [招待あり] 日本薬学会東海支部特別講演会 日本薬学会東海支部特別講演会 2015/05/29 日本語 口頭発表(招待・特別) 公開
π結合の活性化を基盤とする連続反応の開発と応用[招待あり] π結合の活性化を基盤とする連続反応の開発と応用 [招待あり] 東京医科歯科大学 生材研セミナー 東京医科歯科大学 生材研セミナー 2015/01/26 日本語 口頭発表(招待・特別) 公開
Gold-Catalyzed Annulations and Their Medicinal Applications[招待あり] Gold-Catalyzed Annulations and Their Medicinal Applications [招待あり] Gold-Catalyzed Annulations and Their Medicinal Applications [招待あり] DPhG Annual Meeting 2014 DPhG Annual Meeting 2014 DPhG Annual Meeting 2014 2014/09/25 英語 口頭発表(招待・特別) 公開
アレンやアルキンを合成素子とする連続反応の開発と応用[招待あり] アレンやアルキンを合成素子とする連続反応の開発と応用 [招待あり] 金沢大学 医歯薬保健研究域薬学系 講演会 金沢大学 医歯薬保健研究域薬学系 講演会 2014/06/13 日本語 口頭発表(招待・特別) 公開
金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用[招待あり] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用 [招待あり] 京都府立大学 鴨叡会・生命分子化学科セミナー 京都府立大学 鴨叡会・生命分子化学科セミナー 2013/12/17 日本語 口頭発表(招待・特別) 公開
金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用[招待あり] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用 [招待あり] 立命館大学 創薬基盤科学若手セミナー 立命館大学 創薬基盤科学若手セミナー 2013/12/09 日本語 口頭発表(招待・特別) 公開
付加反応を用いて中心骨格を構築する天然物合成[招待あり] 付加反応を用いて中心骨格を構築する天然物合成 [招待あり] 第12回化学系薬学若手研究者セミナー 第12回化学系薬学若手研究者セミナー 2013/08/24 日本語 口頭発表(招待・特別) 公開
高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究[招待あり] 高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究 [招待あり] 天然物ケミカルバイオロジー:分子標的と活性制御地区シンポジウム 天然物ケミカルバイオロジー:分子標的と活性制御地区シンポジウム 新学術領域「天然物ケミカルバイオロジー:分子標的と活性制御」 新学術領域「天然物ケミカルバイオロジー:分子標的と活性制御」 2013/03/16 日本語 口頭発表(招待・特別) 公開
Gold-Catalyzed Reactions for Construction of Heterocycles[招待あり] Gold-Catalyzed Reactions for Construction of Heterocycles [招待あり] Gold-Catalyzed Reactions for Construction of Heterocycles [招待あり] Dortmund University Special Lecture Dortmund University Special Lecture Dortmund University Special Lecture 2013/03/06 英語 口頭発表(招待・特別) 公開
Gold-Catalyzed Reactions for Construction of Heterocycles[招待あり] Gold-Catalyzed Reactions for Construction of Heterocycles [招待あり] Gold-Catalyzed Reactions for Construction of Heterocycles [招待あり] Heidelberg University Special Lecture Heidelberg University Special Lecture Heidelberg University Special Lecture 2013/03/04 英語 口頭発表(招待・特別) 公開
触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用[招待あり] 触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用 [招待あり] 6th Organic Syntheses Lectureship 6th Organic Syntheses Lectureship 東京大学薬学研究科 東京大学薬学研究科 2011/02/22 日本語 口頭発表(招待・特別) 公開
触媒的連続結合形成反応による複素環骨格構築法の開発研究[招待あり] 触媒的連続結合形成反応による複素環骨格構築法の開発研究 [招待あり] 京都大学グローバルCOE プログラム有機若手ワークショップ 京都大学グローバルCOE プログラム有機若手ワークショップ 京都大学グローバルCOE プログラム 京都大学グローバルCOE プログラム 2010/09/14 日本語 口頭発表(招待・特別) 公開
触媒的連続結合形成反応の開発とErgotアルカロイド全合成への応用[招待あり] 触媒的連続結合形成反応の開発とErgotアルカロイド全合成への応用 [招待あり] 第43回天然物化学談話会 第43回天然物化学談話会 天然物化学談話会 天然物化学談話会 2008/07/10 日本語 口頭発表(招待・特別) 公開
アレンを合成素子とする触媒的連続結合形成反応の開発[招待あり] アレンを合成素子とする触媒的連続結合形成反応の開発 [招待あり] 有機合成協会関西支部賞受賞講演 有機合成協会関西支部賞受賞講演 有機合成協会関西支部 有機合成協会関西支部 2006/11/08 日本語 口頭発表(招待・特別) 公開
アレン系化合物の新しい反応性に基づく有用反応の開発と連続環化反応への展開[招待あり] アレン系化合物の新しい反応性に基づく有用反応の開発と連続環化反応への展開 [招待あり] 日本薬学会第124年会(奨励賞受賞講演) 日本薬学会第124年会(奨励賞受賞講演) 日本薬学会 日本薬学会 2005/03/30 日本語 口頭発表(招待・特別) 公開
アレンとパラジウム触媒の新しい反応性を利用した複素環合成[招待あり] アレンとパラジウム触媒の新しい反応性を利用した複素環合成 [招待あり] 日本薬学会第124年会ミニシンポジウム「有機合成化学の若い力」 日本薬学会第124年会ミニシンポジウム「有機合成化学の若い力」 日本薬学会 日本薬学会 2004/03/29 日本語 口頭発表(招待・特別) 公開
パラジウム(0)を触媒としたアミノアレンの環化反応[招待あり] パラジウム(0)を触媒としたアミノアレンの環化反応 [招待あり] 第51回日本薬学会近畿支部総会・大会(受賞講演) 第51回日本薬学会近畿支部総会・大会(受賞講演) 日本薬学会近畿支部 日本薬学会近畿支部 2001/10/27 日本語 口頭発表(招待・特別) 公開
From amino acids to peptide isosteres and heterocycles: implications to vinylaziridines and amino allene chemistry From amino acids to peptide isosteres and heterocycles: implications to vinylaziridines and amino allene chemistry 11th Akabori conference 11th Akabori conference Akabori Society Akabori Society 2006/09/11 英語 口頭発表(招待・特別) 公開

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タイトル言語:
書籍等出版物
著者 著者(日本語) 著者(英語) タイトル タイトル(日本語) タイトル(英語) 出版社 出版社(日本語) 出版社(英語) 出版年月 記述言語 担当区分 公開
Hiroaki Ohno Hiroaki Ohno Intramolecular C−X Bond Formation between C=X or X−H and Alkynes (in Transition-Metal-Mediated Aromatic Ring Construction) Intramolecular C−X Bond Formation between C=X or X−H and Alkynes (in Transition-Metal-Mediated Aromatic Ring Construction) Wiley Wiley 2013 英語 公開
Hiroaki Ohno and Kiyoshi Tomioka Hiroaki Ohno and Kiyoshi Tomioka Synthesis by Substitution (in Science of Synthesis) Synthesis by Substitution (in Science of Synthesis) Thieme Thieme 2007 英語 公開
Hiroaki Ohno Hiroaki Ohno Vinylaziridines in Organic Synthesis (in Aziridines and Epoxides in Organic Synthesis) Vinylaziridines in Organic Synthesis (in Aziridines and Epoxides in Organic Synthesis) Wiley-VCH Wiley-VCH 2005 英語 公開
Hiroaki Ohno, Yasuo Nagaoka, and Kiyoshi Tomioka Hiroaki Ohno, Yasuo Nagaoka, and Kiyoshi Tomioka Enantioselective Synthesis of Allenes (in Modern Allene Chemistry) Enantioselective Synthesis of Allenes (in Modern Allene Chemistry) Wiley-VCH Wiley-VCH 2004 英語 公開
タイトル言語:
特許
発明者 発明者(日本語) 発明者(英語) 発明の名称 発明の名称(日本語) 発明の名称(英語) 審査の段階 番号 年月 公開
前田 英樹, 加藤 貴之, 松岡 雅雄, 志村 和也, 藤井 信孝, 大野 浩章, 大石 真也, 水原 司 前田 英樹, 加藤 貴之, 松岡 雅雄, 志村 和也, 藤井 信孝, 大野 浩章, 大石 真也, 水原 司 ピリミドベンゾチアジン−6−イミン誘導体またはその塩を含有するウイルス感染症の治療および/または予防のための薬剤 ピリミドベンゾチアジン−6−イミン誘導体またはその塩を含有するウイルス感染症の治療および/または予防のための薬剤 特許公開 特開2012-250973 2012/12/20 公開
辻本 豪三, 平澤 明, 村田 克美, 藤井 信孝, 大野 浩章, 大石 真也, 鈴木 大和, ゾンイェ ホウ, 仲西 功, 木下 誉富, 高倉 喜信, 西川 元也 辻本 豪三, 平澤 明, 村田 克美, 藤井 信孝, 大野 浩章, 大石 真也, 鈴木 大和, ゾンイェ ホウ, 仲西 功, 木下 誉富, 高倉 喜信, 西川 元也 キナーゼ阻害剤 キナーゼ阻害剤 特許公開 WO2012-121168 2012/09/13 公開
藤井 信孝, 大野 浩章, 大石 真也, 井ノ口 恵利子, 久保 達彦, 松岡 雅雄, 志村 和也 藤井 信孝, 大野 浩章, 大石 真也, 井ノ口 恵利子, 久保 達彦, 松岡 雅雄, 志村 和也 新規ケモカイン受容体拮抗剤 新規ケモカイン受容体拮抗剤 特許公開 WO2012-118124 2012/09/07 公開
藤井 信孝, 大野 浩章, 大石 真也, 渡部 敏明, 浅井 章良, 澤田 潤一 藤井 信孝, 大野 浩章, 大石 真也, 渡部 敏明, 浅井 章良, 澤田 潤一 Eg5阻害剤 Eg5阻害剤 特許公開 特開2012-051804 2012/03/15 公開
タイトル言語:
学術賞等
賞の名称(日本語) 賞の名称(英語) 授与組織名(日本語) 授与組織名(英語) 年月
近畿支部奨励賞 Kinki Branch Award for Encouragement of Research 日本薬学会 The Pharmaceutical Society of Japan 2001/01/
奨励賞 Award for Young Scientists 日本薬学会 The Pharmaceutical Society of Japan 2005/03/
研究企画賞 Meiji Seika Award in Synthetic Organic Chemistry, Japan 有機合成化学協会 The Society of Synthetic Organic Chemistry, Japan 2005/12/
関西支部賞 Kansai Branch Award 有機合成化学協会関西支部 Kansai Branch, The Society of Synthetic Organic Chemistry, Japan 2006/11/
Banyu Chemist Award Banyu Chemist Award 万有生命科学振興国際交流財団 Banyu Life Science Foundation 2013/11/
Thieme Chemistry Journals Award Thieme Chemistry Journals Award Thieme Thieme 2014/02/
最優秀教員賞 Best Teacher Award 京都大学薬学部 Faculty of Pharmaceutical Sciences, Kyoto University 2014/10/24
外部資金:競争的資金・科学研究費補助金
種別 代表/分担 テーマ(日本語) テーマ(英語) 期間
奨励研究(A) 代表 高活性な降圧剤及びプロテアーゼ阻害剤の開発を指向したアミノアレンの合成研究 2000〜2001
若手研究(B) 代表 生物活性を有する含窒素複素環の自在な合成を指向した新規環形成反応の開発研究 2003〜2004
若手研究(B) 代表 複雑な構造を有する生物活性複素環の一挙合成法の開発と環境調和型連続反応への展開 2005〜2006
若手研究(A) 代表 触媒的連続多点制御反応を基盤とする高原子効率分子構築法の開発と機能性分子への応用 2007〜2009
基盤研究(C) 代表 触媒的連続環化反応を基盤とした生物活性天然物の多様性指向型全合成研究 2010〜2012
新学術領域研究 代表 触媒的多成分反応・高原子効率反応の高度集積化と創薬展開 2010〜2011
若手研究(A) 代表 π結合の連続活性化を基軸とする革新的分子変換法の開発と創薬リードの創出 Development of Inovative Molecular Transformations Based on Consecutive pai-Activation and Its Application to Drug Discovery 2012〜2015
新学術領域研究 代表 原子移動型反応の高度集積化による多環式芳香族化合物の合成と創薬展開 Integration of Atom-Transfer Reactions for the Synthesis of Polycyclic Arenes and Its Application to Drug Discovery 2012〜2013
基盤研究(B) 代表 近接効果を利用した遷移状態制御による選択的活性化法の開発と創薬展開 Selective Activation Based on Control of Transition States by the Neighboring Effect and Its Medicinal Applications 2015〜2018
基盤研究(B) 代表 多環式骨格構築反応を基軸とする生物活性インドールアルカロイドの全合成と創薬展開 Synthetic and Medicinal Studies on Bioactive Indole Alkaloids Based on Direct Construction of Polycyclic Ring Systems 2017〜2020
基盤研究(B) 代表 近接効果を利用した遷移状態制御による選択的活性化法の開発と創薬展開 (平成29年度分) 2017/04/01〜2018/03/31
基盤研究(B) 代表 多環式骨格構築反応を基軸とする生物活性インドールアルカロイドの全合成と創薬展開 (平成29年度分) 2017/04/01〜2018/03/31
新学術領域研究 代表 反応集積化によるアルカロイドの全合成と中分子化戦略 Syntheses and Middle Molecular Strategy of Alkaloids Based on Reaction Integration 2018/04/01〜2019/03/31

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担当科目
講義名(日本語) 講義名(英語) 開講期 学部/研究科 年度
有機化学I(化学結合論) 前期 薬学部 2011/04〜2012/03
特別実習(ケモゲノミクス・薬品有機製造学) 通年 薬学部 2011/04〜2012/03
基礎有機化学A Basic Organic Chemistry A 前期 全学共通科目 2011/04〜2012/03
特別実習[ケモゲノミクス・薬品有機製造学 通年 薬学部 2011/04〜2012/03
創薬リード探索技術 Drug Discovery & Development II: 後期不定 薬学研究科 2011/04〜2012/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2011/04〜2012/03
リード化合物探索スキル(秋入学用) Skill Development for Lead Discovery 後期前期 薬学研究科 2011/04〜2012/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2011/04〜2012/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 前期不定 薬学研究科 2011/04〜2012/03
基盤有機化学実験技術(秋入学用) Basic Laboratory Techniques in Organic Chemistry 後期不定 薬学研究科 2011/04〜2012/03
基盤有機化学概論 Introduction to Basic Organic Chemistry 前期不定 薬学研究科 2011/04〜2012/03
基盤有機化学特論Ⅰ Advanced Basic Organic Chemistry I 後期不定 薬学研究科 2011/04〜2012/03
基盤薬品創製化学実習 Laboratory Practice in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04〜2012/03
基盤薬品創製化学実験 Research in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04〜2012/03
基盤薬品創製化学演習 Seminar in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems 通年不定 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系コンテンツ制作(秋入学) Advanced Methods in Systems 後期前期 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系研究 Research in Systems 通年不定 薬学研究科 2011/04〜2012/03
システム生物学・医薬創成系研究(秋入学用) Research in Systems 後期前期 薬学研究科 2011/04〜2012/03
薬学専門実習II 前期 薬学部 2011/04〜2012/03
薬学専門実習2 前期 薬学部 2011/04〜2012/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2012/04〜2013/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2012/04〜2013/03
博士後期課程特論 doctoral program 前期集中 薬学研究科 2012/04〜2013/03
博士後期課程特論 doctoral program 後期集中 薬学研究科 2012/04〜2013/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 前期不定 薬学研究科 2012/04〜2013/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 後期不定 薬学研究科 2012/04〜2013/03
基盤有機化学概論 Introduction to Basic Organic Chemistry 前期不定 薬学研究科 2012/04〜2013/03
基盤有機化学特論II Advanced Basic Organic Chemistry II 後期不定 薬学研究科 2012/04〜2013/03
基盤薬品創製化学実習 Laboratory Practice in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04〜2013/03
基盤薬品創製化学実験 Research in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04〜2013/03
基盤薬品創製化学演習 Seminar in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04〜2013/03
基礎有機化学A Basic Organic Chemistry A 前期 全学共通科目 2012/04〜2013/03
有機化学I(化学結合論) Organic Chemistry I(Bonding in Organic Chemistry) 前期 薬学部 2012/04〜2013/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2012/04〜2013/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2012/04〜2013/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2012/04〜2013/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2012/04〜2013/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2012/04〜2013/03
薬学専門実習II Pharmaceutical Laboratory II:Organic Chemistry 前期 薬学部 2012/04〜2013/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2012/04〜2013/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2013/04〜2014/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2013/04〜2014/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2013/04〜2014/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2013/04〜2014/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2013/04〜2014/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2013/04〜2014/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2013/04〜2014/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2013/04〜2014/03
博士後期課程特論 doctoral program 前期集中 薬学研究科 2013/04〜2014/03
博士後期課程特論 doctoral program 後期集中 薬学研究科 2013/04〜2014/03
基礎有機化学B Basic Organic Chemistry B 後期 全学共通科目 2013/04〜2014/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2013/04〜2014/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2014/04〜2015/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2014/04〜2015/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2014/04〜2015/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2014/04〜2015/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2014/04〜2015/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2014/04〜2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2014/04〜2015/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2014/04〜2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2014/04〜2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2014/04〜2015/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2014/04〜2015/03
基礎有機化学B Basic Organic Chemistry B 後期 全学共通科目 2014/04〜2015/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2014/04〜2015/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2015/04〜2016/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2015/04〜2016/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2015/04〜2016/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2015/04〜2016/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2015/04〜2016/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2015/04〜2016/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2015/04〜2016/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2015/04〜2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2015/04〜2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2015/04〜2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2015/04〜2016/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2015/04〜2016/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2016/04〜2017/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2016/04〜2017/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2016/04〜2017/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2016/04〜2017/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2016/04〜2017/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2016/04〜2017/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2016/04〜2017/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2016/04〜2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2016/04〜2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2016/04〜2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2016/04〜2017/03
創薬有機化学概論 Introduction to Organic Chemistry for Drug Discovery 前期不定 薬学研究科 2017/04〜2018/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2017/04〜2018/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2017/04〜2018/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2017/04〜2018/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2017/04〜2018/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2017/04〜2018/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2017/04〜2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2017/04〜2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2017/04〜2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2017/04〜2018/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2018/04〜2019/03
創薬有機化学概論 Introduction to Organic Chemistry for Drug Discovery 前期不定 薬学研究科 2018/04〜2019/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2018/04〜2019/03
基盤有機化学特論II Advanced Basic Organic Chemistry II 後期不定 薬学研究科 2018/04〜2019/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2018/04〜2019/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2018/04〜2019/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2018/04〜2019/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2018/04〜2019/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2018/04〜2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 後期前期 薬学研究科 2018/04〜2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2018/04〜2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2018/04〜2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2018/04〜2019/03
生理化学概論 Outline of Physiological Chemistry 後期集中 全学共通科目 2018/04〜2019/03
臨床薬学概論 Introduction to Clinical Pharmacy 前期不定 薬学研究科 2018/04〜2019/03

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全学運営(役職等)
役職名 期間
外国語教育専門委員会 委員 2008/04/01〜2011/03/31
国際高等教育院 企画評価専門委員会 委員 2015/04/01〜2017/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2013/07/05〜2014/06/30
国際高等教育院 企画評価専門委員会 化学部会 委員 2015/05/01〜2016/04/30
国際高等教育院 企画評価専門委員会 化学部会 委員 2016/05/01〜2017/04/30
学生生活委員会 委員 2016/04/01〜2018/03/31
学生生活委員会第一小委員会 委員 2016/04/01〜2018/03/31
京都大学奨学金返還免除候補者選考委員会 4号委員 2016/04/01〜2018/03/31
オープンキャンパス委員会 委員 2016/01/01〜2016/12/31
図書館協議会 協議員 2017/04/01〜2019/03/31
学生生活委員会第一小委員会 委員長 2016/04/01〜2018/03/31
京都大学奨学金返還免除候補者選考委員会 委員長 2016/04/01〜2018/03/31
学生表彰選考委員会 委員
国際高等教育院 企画評価専門委員会 委員 2017/04/01〜2019/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2017/05/01〜2018/03/31
学生表彰選考委員会 2018/01/01〜2018/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2018/04/01〜2019/03/31
国際高等教育院 基盤企画評価専門委員会 委員 2017/04/01〜2019/03/31

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部局運営(役職等)
役職名 期間
薬学研究科 就職委員 2017/04/01〜2019/03/31
薬学研究科 学生委員(先任教員) 2017/04/01〜2018/03/31
薬学研究科 環境・安全衛生委員会委員長 2016/04/01〜2018/03/31
薬学研究科 図書委員会委員長 2017/04/01〜2019/03/31