井貫 晋輔

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Name(Kanji/Kana/Abecedarium Latinum)
井貫 晋輔/イヌキ シンスケ/Inuki, Shinsuke
Primary Affiliation(Org1/Job title)
Graduate Schools Pharmaceutical Sciences/Assistant Professor
Faculty
Org1 Job title
薬学部
Academic Organizations You are Affiliated to in Japan
Organization name(Japanese) Organization name(English)
日本薬学会
日本化学会
有機合成化学協会
日本ケミカルバイオロジー学会
日本ペプチド学会
日本糖質学会
Academic Degree
Field(Japanese) Field(English) University(Japanese) University(English) Method
修士(薬学) 京都大学
博士(薬学) 京都大学
Graduate School
University(Japanese) University(English) Faculty(Japanese) Faculty(English) Major(Japanese) Major(English) Degree
京都大学 大学院薬学研究科修士課程創薬科学専攻 修了
京都大学 大学院薬学研究科博士後期課程創薬科学専攻 修了
Undergraduate School / Major(s)
University(Japanese) University(English) Faculty(Japanese) Faculty(English) Major(s)(Japanese) Major(s)(English) Degree
京都大学 薬学部総合薬学科 卒業
Work Experience
Period Organization(Japanese) Organization(English) Job title(Japanese) Job title(English)
2008/04/01-2011/03/31 日本学術振興会 Japan Society for the Promotion of Science 日本学術振興会特別研究員(DC1) JSPS Research Fellow (DC1)
2011/04/01-2014/03/31 富士フイルム株式会社 Fujifilm Co., Ltd. 研究員 Research Scientist
2014/04/01-2017/06/30 慶應義塾大学理工学部化学科 Department of Chemistry, Faculty of Science and Technology, Keio University 助教 Research Associate
2017/07/01- 京都大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Kyoto University 助教 Assistant Professor
ORCID ID
https://orcid.org/0000-0002-7525-1280
researchmap URL
https://researchmap.jp/7000020590
Research Topics
(Japanese)
生物活性化合物の合成と機能解析
Fields of research (key words)
Key words(Japanese) Key words(English)
有機化学
生物有機化学
医薬品化学
創薬化学
Published Papers
Author Author(Japanese) Author(English) Title Title(Japanese) Title(English) Bibliography Bibliography(Japanese) Bibliography(English) Publication date Refereed paper Language Publishing type Disclose
Shinsuke Inuki, Takashi Miyagawa, Shinya Oishi, Hiroaki Ohno Shinsuke Inuki, Takashi Miyagawa, Shinya Oishi, Hiroaki Ohno Shinsuke Inuki, Takashi Miyagawa, Shinya Oishi, Hiroaki Ohno Introduction of a Polar Functional Group to the Lipid Tail of 4-<i>epi</i>-Jaspine B Affects Sphingosine Kinase Isoform Selectivity Introduction of a Polar Functional Group to the Lipid Tail of 4-<i>epi</i>-Jaspine B Affects Sphingosine Kinase Isoform Selectivity Introduction of a Polar Functional Group to the Lipid Tail of 4-<i>epi</i>-Jaspine B Affects Sphingosine Kinase Isoform Selectivity Chemical and Pharmaceutical Bulletin, 66, 9, 866 Chemical and Pharmaceutical Bulletin, 66, 9, 866 Chemical and Pharmaceutical Bulletin, 66, 9, 866 2018/09 Refereed Disclose to all
Naoka Hamada, Ayuta Yamaguchi, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno Naoka Hamada, Ayuta Yamaguchi, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno Naoka Hamada, Ayuta Yamaguchi, Shinsuke Inuki, Shinya Oishi, Hiroaki Ohno Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds Gold(I)-Catalyzed Oxidative Cascade Cyclization of 1,4-Diyn-3-ones for the Construction of Tropone-Fused Furan Scaffolds Organic Letters, 20, 15, 4401 Organic Letters, 20, 15, 4401 Organic Letters, 20, 15, 4401 2018/07 Refereed Disclose to all
Shinsuke Inuki, Emi Kashiwabara, Natsumi Hirata, Junichiro Kishi, Etsuko Nabika, Yukari Fujimoto Shinsuke Inuki, Emi Kashiwabara, Natsumi Hirata, Junichiro Kishi, Etsuko Nabika, Yukari Fujimoto Shinsuke Inuki, Emi Kashiwabara, Natsumi Hirata, Junichiro Kishi, Etsuko Nabika, Yukari Fujimoto Potent Th2 Cytokine-Bias of Natural Killer T Cell by CD1d Glycolipid Ligands Based on "Anchoring Effect" of Polar Groups in Their Lipid Component Potent Th2 Cytokine-Bias of Natural Killer T Cell by CD1d Glycolipid Ligands Based on "Anchoring Effect" of Polar Groups in Their Lipid Component Potent Th2 Cytokine-Bias of Natural Killer T Cell by CD1d Glycolipid Ligands Based on "Anchoring Effect" of Polar Groups in Their Lipid Component Angewandte Chemie International Edition Angewandte Chemie International Edition Angewandte Chemie International Edition 2018/06 Refereed Disclose to all
Yohei Arai, Shinsuke Inuki, Yukari Fujimoto Yohei Arai, Shinsuke Inuki, Yukari Fujimoto Yohei Arai, Shinsuke Inuki, Yukari Fujimoto Site-specific effect of polar functional group-modification in lipids of TLR2 ligands for modulating the ligand immunostimulatory activity Site-specific effect of polar functional group-modification in lipids of TLR2 ligands for modulating the ligand immunostimulatory activity Site-specific effect of polar functional group-modification in lipids of TLR2 ligands for modulating the ligand immunostimulatory activity Bioorganic & Medicinal Chemistry Letters, 28, 9, 1638 Bioorganic & Medicinal Chemistry Letters, 28, 9, 1638 Bioorganic & Medicinal Chemistry Letters, 28, 9, 1638 2018/05 Refereed Disclose to all
Yuka Kobayashi, Masaru Hoshino, Tomoshi Kameda, Kazuya Kobayashi, Kenichi Akaji, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Yuka Kobayashi, Masaru Hoshino, Tomoshi Kameda, Kazuya Kobayashi, Kenichi Akaji, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Yuka Kobayashi, Masaru Hoshino, Tomoshi Kameda, Kazuya Kobayashi, Kenichi Akaji, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle Inorganic Chemistry, 57, 9, 5475 Inorganic Chemistry, 57, 9, 5475 Inorganic Chemistry, 57, 9, 5475 2018/04 Refereed Disclose to all
Takashi Miyagawa, Shinsuke Inuki, Maho Honda, Shinya Nakamura, Isao Nakanishi, Nobutaka Fujii, Shinya Oishi, Hiroaki Ohno Takashi Miyagawa, Shinsuke Inuki, Maho Honda, Shinya Nakamura, Isao Nakanishi, Nobutaka Fujii, Shinya Oishi, Hiroaki Ohno Takashi Miyagawa, Shinsuke Inuki, Maho Honda, Shinya Nakamura, Isao Nakanishi, Nobutaka Fujii, Shinya Oishi, Hiroaki Ohno Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases Synthesis of jaspine B regioisomers through palladium-catalyzed stereoselective tetrahydrofuran formation: Insight into the ligand recognition of sphingosine kinases Tetrahedron, 74, 15, 1802 Tetrahedron, 74, 15, 1802 Tetrahedron, 74, 15, 1802 2018/04 Refereed Disclose to all
Masato Kaneda, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Masato Kaneda, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Masato Kaneda, Shinsuke Inuki, Hiroaki Ohno, Shinya Oishi Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide–Polyketide Macrocycle Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide–Polyketide Macrocycle Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide–Polyketide Macrocycle The Journal of Organic Chemistry, 83, 6, 3047 The Journal of Organic Chemistry, 83, 6, 3047 The Journal of Organic Chemistry, 83, 6, 3047 2018/02 Refereed Disclose to all
Hiroaki Ohno, Shinsuke Inuki Hiroaki Ohno, Shinsuke Inuki Hiroaki Ohno, Shinsuke Inuki Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis Recent Progress in Palladium-Catalyzed Cascade Cyclizations for Natural Product Synthesis Synthesis, 50, 04, 700 Synthesis, 50, 04, 700 Synthesis, 50, 04, 700 2018/01 Refereed Disclose to all
Yuiki Kawada, Shunsuke Ohmura, Misaki Kobayashi, Wataru Nojo, Masaki Kondo, Yuka Matsuda, Junpei Matsuoka, Shinsuke Inuki, Shinya Oishi, Chao Wang, Tatsuo Saito, Masanobu Uchiyama, Takanori Suzuki, Hiroaki Ohno Yuiki Kawada, Shunsuke Ohmura, Misaki Kobayashi, Wataru Nojo, Masaki Kondo, Yuka Matsuda, Junpei Matsuoka, Shinsuke Inuki, Shinya Oishi, Chao Wang, Tatsuo Saito, Masanobu Uchiyama, Takanori Suzuki, Hiroaki Ohno Yuiki Kawada, Shunsuke Ohmura, Misaki Kobayashi, Wataru Nojo, Masaki Kondo, Yuka Matsuda, Junpei Matsuoka, Shinsuke Inuki, Shinya Oishi, Chao Wang, Tatsuo Saito, Masanobu Uchiyama, Takanori Suzuki, Hiroaki Ohno Direct synthesis of aryl-annulated [c]carbazoles by gold(i)-catalysed cascade reaction of azide-diynes and arenes Direct synthesis of aryl-annulated [c]carbazoles by gold(i)-catalysed cascade reaction of azide-diynes and arenes Direct synthesis of aryl-annulated [c]carbazoles by gold(i)-catalysed cascade reaction of azide-diynes and arenes Chemical Science Chemical Science Chemical Science 2018 Refereed Disclose to all
Yohei Arai, Kouhei Yokoyama, Yuki Kawahara, Qi Feng, Ippei Ohta, Atsushi Shimoyama, Shinsuke Inuki, Koichi Fukase, Kazuya Kabayama, Yukari Fujimoto Yohei Arai, Kouhei Yokoyama, Yuki Kawahara, Qi Feng, Ippei Ohta, Atsushi Shimoyama, Shinsuke Inuki, Koichi Fukase, Kazuya Kabayama, Yukari Fujimoto Yohei Arai, Kouhei Yokoyama, Yuki Kawahara, Qi Feng, Ippei Ohta, Atsushi Shimoyama, Shinsuke Inuki, Koichi Fukase, Kazuya Kabayama, Yukari Fujimoto Time-lapse monitoring of TLR2 ligand internalization with newly developed fluorescent probes Time-lapse monitoring of TLR2 ligand internalization with newly developed fluorescent probes Time-lapse monitoring of TLR2 ligand internalization with newly developed fluorescent probes Organic & Biomolecular Chemistry, 16, 20, 3824 Organic & Biomolecular Chemistry, 16, 20, 3824 Organic & Biomolecular Chemistry, 16, 20, 3824 2018 Refereed Disclose to all
Shinsuke Inuki, Junichiro Kishi, Emi Kashiwabara, Toshihiko Aiba, Yukari Fujimoto Shinsuke Inuki, Junichiro Kishi, Emi Kashiwabara, Toshihiko Aiba, Yukari Fujimoto Shinsuke Inuki, Junichiro Kishi, Emi Kashiwabara, Toshihiko Aiba, Yukari Fujimoto Convergent Synthesis of Digalactosyl Diacylglycerols Convergent Synthesis of Digalactosyl Diacylglycerols Convergent Synthesis of Digalactosyl Diacylglycerols Organic Letters, 19, 24, 6482 Organic Letters, 19, 24, 6482 Organic Letters, 19, 24, 6482 2017/11 Refereed Disclose to all
Qianqian Wang, Roberta Marchetti, Sladjana Prisic, Kentaro Ishii, Yohei Arai, Ippei Ohta, Shinsuke Inuki, Susumu Uchiyama, Alba Silipo, Antonio Molinaro, Robert N. Husson, Koichi Fukase, Yukari Fujimoto Qianqian Wang, Roberta Marchetti, Sladjana Prisic, Kentaro Ishii, Yohei Arai, Ippei Ohta, Shinsuke Inuki, Susumu Uchiyama, Alba Silipo, Antonio Molinaro, Robert N. Husson, Koichi Fukase, Yukari Fujimoto Qianqian Wang, Roberta Marchetti, Sladjana Prisic, Kentaro Ishii, Yohei Arai, Ippei Ohta, Shinsuke Inuki, Susumu Uchiyama, Alba Silipo, Antonio Molinaro, Robert N. Husson, Koichi Fukase, Yukari Fujimoto A Comprehensive Study of the Interaction between Peptidoglycan Fragments and the Extracellular Domain of Mycobacterium tuberculosis Ser/Thr Kinase PknB A Comprehensive Study of the Interaction between Peptidoglycan Fragments and the Extracellular Domain of Mycobacterium tuberculosis Ser/Thr Kinase PknB A Comprehensive Study of the Interaction between Peptidoglycan Fragments and the Extracellular Domain of Mycobacterium tuberculosis Ser/Thr Kinase PknB ChemBioChem, 18, 21, 2094 ChemBioChem, 18, 21, 2094 ChemBioChem, 18, 21, 2094 2017/09 Refereed Disclose to all
Shinsuke Inuki, Ippei Ohta, Shunichi Ishibashi, Masayuki Takamatsu, Koichi Fukase, Yukari Fujimoto Shinsuke Inuki, Ippei Ohta, Shunichi Ishibashi, Masayuki Takamatsu, Koichi Fukase, Yukari Fujimoto Shinsuke Inuki, Ippei Ohta, Shunichi Ishibashi, Masayuki Takamatsu, Koichi Fukase, Yukari Fujimoto Total Synthesis of Cardiolipins Containing Chiral Cyclopropane Fatty Acids Total Synthesis of Cardiolipins Containing Chiral Cyclopropane Fatty Acids Total Synthesis of Cardiolipins Containing Chiral Cyclopropane Fatty Acids The Journal of Organic Chemistry, 82, 15, 7832 The Journal of Organic Chemistry, 82, 15, 7832 The Journal of Organic Chemistry, 82, 15, 7832 2017/07 Refereed Disclose to all
Hiroaki Ohno, Maho Honda, Naoka Hamada, Jun Miyagaki, Akira Iwata, Kazuhiro Otsuki, Toru Maruyama, Shinya Nakamura, Isao Nakanishi, Shinsuke Inuki, Nobutaka Fujii, Shinya Oishi Hiroaki Ohno, Maho Honda, Naoka Hamada, Jun Miyagaki, Akira Iwata, Kazuhiro Otsuki, Toru Maruyama, Shinya Nakamura, Isao Nakanishi, Shinsuke Inuki, Nobutaka Fujii, Shinya Oishi Hiroaki Ohno, Maho Honda, Naoka Hamada, Jun Miyagaki, Akira Iwata, Kazuhiro Otsuki, Toru Maruyama, Shinya Nakamura, Isao Nakanishi, Shinsuke Inuki, Nobutaka Fujii, Shinya Oishi Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure–activity relationship study of 4- epi -jaspine B Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure–activity relationship study of 4- epi -jaspine B Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure–activity relationship study of 4- epi -jaspine B Bioorganic & Medicinal Chemistry, 25, 12, 3046 Bioorganic & Medicinal Chemistry, 25, 12, 3046 Bioorganic & Medicinal Chemistry, 25, 12, 3046 2017/06 Refereed Disclose to all
Shinsuke Inuki, Toshihiko Aiba, Shota Kawakami, Taishin Akiyama, Jun-ichiro Inoue, Yukari Fujimoto Shinsuke Inuki, Toshihiko Aiba, Shota Kawakami, Taishin Akiyama, Jun-ichiro Inoue, Yukari Fujimoto Shinsuke Inuki, Toshihiko Aiba, Shota Kawakami, Taishin Akiyama, Jun-ichiro Inoue, Yukari Fujimoto Chemical Synthesis of d-glycero-d-manno-Heptose 1,7-Bisphosphate and Evaluation of Its Ability to Modulate NF-κB Activation Chemical Synthesis of d-glycero-d-manno-Heptose 1,7-Bisphosphate and Evaluation of Its Ability to Modulate NF-κB Activation Chemical Synthesis of d-glycero-d-manno-Heptose 1,7-Bisphosphate and Evaluation of Its Ability to Modulate NF-κB Activation Organic Letters, 19, 12, 3079 Organic Letters, 19, 12, 3079 Organic Letters, 19, 12, 3079 2017/05 Refereed Disclose to all
Toshihiko Aiba, Sae Suehara, Siew-Ling Choy, Yuuki Maekawa, Hannelore Lotter, Toshiaki Murai, Shinsuke Inuki, Koichi Fukase, Yukari Fujimoto Toshihiko Aiba, Sae Suehara, Siew-Ling Choy, Yuuki Maekawa, Hannelore Lotter, Toshiaki Murai, Shinsuke Inuki, Koichi Fukase, Yukari Fujimoto Toshihiko Aiba, Sae Suehara, Siew-Ling Choy, Yuuki Maekawa, Hannelore Lotter, Toshiaki Murai, Shinsuke Inuki, Koichi Fukase, Yukari Fujimoto Employing BINOL-Phosphoroselenoyl Chloride for Selective Inositol Phosphorylation and Synthesis of Glycosyl Inositol Phospholipid from Entamoeba histolytica Employing BINOL-Phosphoroselenoyl Chloride for Selective Inositol Phosphorylation and Synthesis of Glycosyl Inositol Phospholipid from Entamoeba histolytica Employing BINOL-Phosphoroselenoyl Chloride for Selective Inositol Phosphorylation and Synthesis of Glycosyl Inositol Phospholipid from Entamoeba histolytica Chemistry - A European Journal, 23, 34, 8304 Chemistry - A European Journal, 23, 34, 8304 Chemistry - A European Journal, 23, 34, 8304 2017/05 Refereed Disclose to all
Shinsuke Inuki, Keisuke Sato, Takahide Fukuyama, Ilhyong Ryu, Yukari Fujimoto Shinsuke Inuki, Keisuke Sato, Takahide Fukuyama, Ilhyong Ryu, Yukari Fujimoto Shinsuke Inuki, Keisuke Sato, Takahide Fukuyama, Ilhyong Ryu, Yukari Fujimoto Formal Total Synthesis of l-Ossamine via Decarboxylative Functionalization Using Visible-Light-Mediated Photoredox Catalysis in a Flow System Formal Total Synthesis of l-Ossamine via Decarboxylative Functionalization Using Visible-Light-Mediated Photoredox Catalysis in a Flow System Formal Total Synthesis of l-Ossamine via Decarboxylative Functionalization Using Visible-Light-Mediated Photoredox Catalysis in a Flow System The Journal of Organic Chemistry, 82, 2, 1248 The Journal of Organic Chemistry, 82, 2, 1248 The Journal of Organic Chemistry, 82, 2, 1248 2017/01 Refereed Disclose to all
井貫晋輔, 相羽俊彦, 平田菜摘, 柏原瑛美, 喜多俊介, 前仲勝実, 深瀬浩一, 藤本ゆかり 井貫晋輔, 相羽俊彦, 平田菜摘, 柏原瑛美, 喜多俊介, 前仲勝実, 深瀬浩一, 藤本ゆかり 糖脂質 α-GalCer を基盤とした脂質改変型 CD1d リガンドの創製研究 糖脂質 α-GalCer を基盤とした脂質改変型 CD1d リガンドの創製研究 エンドトキシン・自然免疫研究20 –自然免疫における化学生物学の貢献–, 20, 64-67 エンドトキシン・自然免疫研究20 –自然免疫における化学生物学の貢献–, 20, 64-67 , 20, 64-67 2017 Disclose to all
Shinsuke Inuki, Toshihiko Aiba, Natsumi Hirata, Osamu Ichihara, Daisuke Yoshidome, Shunsuke Kita, Katsumi Maenaka, Koichi Fukase, Yukari Fujimoto Shinsuke Inuki, Toshihiko Aiba, Natsumi Hirata, Osamu Ichihara, Daisuke Yoshidome, Shunsuke Kita, Katsumi Maenaka, Koichi Fukase, Yukari Fujimoto Shinsuke Inuki, Toshihiko Aiba, Natsumi Hirata, Osamu Ichihara, Daisuke Yoshidome, Shunsuke Kita, Katsumi Maenaka, Koichi Fukase, Yukari Fujimoto Isolated Polar Amino Acid Residues Modulate Lipid Binding in the Large Hydrophobic Cavity of CD1d Isolated Polar Amino Acid Residues Modulate Lipid Binding in the Large Hydrophobic Cavity of CD1d Isolated Polar Amino Acid Residues Modulate Lipid Binding in the Large Hydrophobic Cavity of CD1d ACS Chemical Biology, 11, 11, 3132 ACS Chemical Biology, 11, 11, 3132 ACS Chemical Biology, 11, 11, 3132 2016/10 Refereed Disclose to all
Shinsuke Inuki Shinsuke Inuki Shinsuke Inuki Gold-Catalyzed Activation of Glycosyl Donors with Alkyne Moieties for Glycosylation Reaction Gold-Catalyzed Activation of Glycosyl Donors with Alkyne Moieties for Glycosylation Reaction Gold-Catalyzed Activation of Glycosyl Donors with Alkyne Moieties for Glycosylation Reaction Journal of Synthetic Organic Chemistry, Japan, 74, 1, 69 Journal of Synthetic Organic Chemistry, Japan, 74, 1, 69 Journal of Synthetic Organic Chemistry, Japan, 74, 1, 69 2016 Refereed Disclose to all
Zenyu Shiokawa, Emi Kashiwabara, Daisuke Yoshidome, Koichi Fukase, Shinsuke Inuki, Yukari Fujimoto Zenyu Shiokawa, Emi Kashiwabara, Daisuke Yoshidome, Koichi Fukase, Shinsuke Inuki, Yukari Fujimoto Zenyu Shiokawa, Emi Kashiwabara, Daisuke Yoshidome, Koichi Fukase, Shinsuke Inuki, Yukari Fujimoto Discovery of a Novel Scaffold as an Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on the Pyrrolopiperazinone Alkaloid, Longamide B Discovery of a Novel Scaffold as an Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on the Pyrrolopiperazinone Alkaloid, Longamide B Discovery of a Novel Scaffold as an Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on the Pyrrolopiperazinone Alkaloid, Longamide B ChemMedChem, 11, 24, 2682 ChemMedChem, 11, 24, 2682 ChemMedChem, 11, 24, 2682 2016 Refereed Disclose to all
Shinsuke Inuki, Keisuke Sato, Yukari Fujimoto Shinsuke Inuki, Keisuke Sato, Yukari Fujimoto Shinsuke Inuki, Keisuke Sato, Yukari Fujimoto Visible-light-mediated decarboxylative benzoyloxylation of β-hydroxy amino acids and its application to synthesis of functional 1,2-amino alcohol derivatives Visible-light-mediated decarboxylative benzoyloxylation of β-hydroxy amino acids and its application to synthesis of functional 1,2-amino alcohol derivatives Visible-light-mediated decarboxylative benzoyloxylation of β-hydroxy amino acids and its application to synthesis of functional 1,2-amino alcohol derivatives Tetrahedron Letters, 56, 42, 5787 Tetrahedron Letters, 56, 42, 5787 Tetrahedron Letters, 56, 42, 5787 2015/10 Refereed Disclose to all
Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Convenient synthesis of spiroindole derivatives via palladium-catalyzed cyclization of propargyl chlorides Convenient synthesis of spiroindole derivatives via palladium-catalyzed cyclization of propargyl chlorides Convenient synthesis of spiroindole derivatives via palladium-catalyzed cyclization of propargyl chlorides Tetrahedron, 71, 37, 6580 Tetrahedron, 71, 37, 6580 Tetrahedron, 71, 37, 6580 2015/09 Refereed Disclose to all
Koichi Fukase, Yukari Fujimoto, Zenyu Shiokawa, Shinsuke Inuki Koichi Fukase, Yukari Fujimoto, Zenyu Shiokawa, Shinsuke Inuki Koichi Fukase, Yukari Fujimoto, Zenyu Shiokawa, Shinsuke Inuki Efficient Synthesis of (–)-Hanishin, (–)-Longamide B, and (–)-Longamide B Methyl Ester through Piperazinone Formation from 1,2-Cyclic Sulfamidates Efficient Synthesis of (–)-Hanishin, (–)-Longamide B, and (–)-Longamide B Methyl Ester through Piperazinone Formation from 1,2-Cyclic Sulfamidates Efficient Synthesis of (–)-Hanishin, (–)-Longamide B, and (–)-Longamide B Methyl Ester through Piperazinone Formation from 1,2-Cyclic Sulfamidates Synlett, 27, 04, 616 Synlett, 27, 04, 616 Synlett, 27, 04, 616 2015 Refereed Disclose to all
Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Chem. Commun., 50, 3, 298 Chem. Commun., 50, 3, 298 Chem. Commun., 50, 3, 298 2014 Refereed Disclose to all
Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Palladium-Catalyzed Medium-Ring Formation for Construction of the Core Structure of Laurencia Oxacycles: Synthetic Study of Laurendecumallene B Palladium-Catalyzed Medium-Ring Formation for Construction of the Core Structure of Laurencia Oxacycles: Synthetic Study of Laurendecumallene B Palladium-Catalyzed Medium-Ring Formation for Construction of the Core Structure of Laurencia Oxacycles: Synthetic Study of Laurendecumallene B Organic Letters, 15, 12, 3046 Organic Letters, 15, 12, 3046 Organic Letters, 15, 12, 3046 2013/05 Refereed Disclose to all
Hiroaki Ohno, Nobutaka Fujii, Hiroaki Chiba, Shinsuke Inuki, Shinya Oishi Hiroaki Ohno, Nobutaka Fujii, Hiroaki Chiba, Shinsuke Inuki, Shinya Oishi Hiroaki Ohno, Nobutaka Fujii, Hiroaki Chiba, Shinsuke Inuki, Shinya Oishi The Synthesis of Alkaloids Using Transition-Metal-Catalyzed Intramolecular Amination Reactions The Synthesis of Alkaloids Using Transition-Metal-Catalyzed Intramolecular Amination Reactions The Synthesis of Alkaloids Using Transition-Metal-Catalyzed Intramolecular Amination Reactions Synlett, 25, 02, 179 Synlett, 25, 02, 179 Synlett, 25, 02, 179 2013 Refereed Disclose to all
Yuji Yoshimitsu, Shinya Oishi, Jun Miyagaki, Shinsuke Inuki, Hiroaki Ohno, Nobutaka Fujii Yuji Yoshimitsu, Shinya Oishi, Jun Miyagaki, Shinsuke Inuki, Hiroaki Ohno, Nobutaka Fujii Yuji Yoshimitsu, Shinya Oishi, Jun Miyagaki, Shinsuke Inuki, Hiroaki Ohno, Nobutaka Fujii Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Bioorganic & Medicinal Chemistry, 19, 18, 5402 Bioorganic & Medicinal Chemistry, 19, 18, 5402 Bioorganic & Medicinal Chemistry, 19, 18, 5402 2011/09 Refereed Disclose to all
Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Akira Iwata, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Formal Total Synthesis of (+)-Lysergic Acid via Zinc(II)-Mediated Regioselective Ring-Opening Reduction of 2-Alkynyl-3-indolyloxirane Formal Total Synthesis of (+)-Lysergic Acid via Zinc(II)-Mediated Regioselective Ring-Opening Reduction of 2-Alkynyl-3-indolyloxirane Formal Total Synthesis of (+)-Lysergic Acid via Zinc(II)-Mediated Regioselective Ring-Opening Reduction of 2-Alkynyl-3-indolyloxirane The Journal of Organic Chemistry, 76, 13, 5506 The Journal of Organic Chemistry, 76, 13, 5506 The Journal of Organic Chemistry, 76, 13, 5506 2011/07 Refereed Disclose to all
Shinsuke Inuki, Akira Iwata, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Akira Iwata, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Akira Iwata, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups Enantioselective Total Synthesis of (+)-Lysergic Acid, (+)-Lysergol, and (+)-Isolysergol by Palladium-Catalyzed Domino Cyclization of Allenes Bearing Amino and Bromoindolyl Groups The Journal of Organic Chemistry, 76, 7, 2072 The Journal of Organic Chemistry, 76, 7, 2072 The Journal of Organic Chemistry, 76, 7, 2072 2011/04 Refereed Disclose to all
Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Organic Letters, 13, 8, 2145 Organic Letters, 13, 8, 2145 Organic Letters, 13, 8, 2145 2011/04 Refereed Disclose to all
Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Propargyl Chlorides and Carbonates The Journal of Organic Chemistry, 75, 11, 3831 The Journal of Organic Chemistry, 75, 11, 3831 The Journal of Organic Chemistry, 75, 11, 3831 2010/06 Refereed Disclose to all
Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Yuji Yoshimitsu, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B) Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B) Stereoselective Divergent Synthesis of Four Diastereomers of Pachastrissamine (Jaspine B) The Journal of Organic Chemistry, 75, 11, 3843 The Journal of Organic Chemistry, 75, 11, 3843 The Journal of Organic Chemistry, 75, 11, 3843 2010/06 Refereed Disclose to all
Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Yuji Yoshimitsu, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes Organic Letters, 11, 19, 4478 Organic Letters, 11, 19, 4478 Organic Letters, 11, 19, 4478 2009/10 Refereed Disclose to all
Tsukasa Mizuhara, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Tsukasa Mizuhara, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Tsukasa Mizuhara, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Cu(ii)-mediated oxidative intermolecular ortho C–H functionalisation using tetrahydropyrimidine as the directing group Cu(ii)-mediated oxidative intermolecular ortho C–H functionalisation using tetrahydropyrimidine as the directing group Cu(ii)-mediated oxidative intermolecular ortho C–H functionalisation using tetrahydropyrimidine as the directing group Chemical Communications, 23, 3413 Chemical Communications, 23, 3413 Chemical Communications, 23, 3413 2009 Refereed Disclose to all
Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Total Synthesis of (±)-Lysergic Acid, Lysergol, and Isolysergol by Palladium-Catalyzed Domino Cyclization of Amino Allenes Bearing a Bromoindolyl Group Organic Letters, 10, 22, 5239 Organic Letters, 10, 22, 5239 Organic Letters, 10, 22, 5239 2008/11 Refereed Disclose to all
Satoshi Ueda, Manabu Kato, Shinsuke Inuki, Hiroaki Ohno, Barry Evans, Zi-xuan Wang, Stephen C. Peiper, Kazuki Izumi, Eiichi Kodama, Masao Matsuoka, Hideko Nagasawa, Shinya Oishi, Nobutaka Fujii Satoshi Ueda, Manabu Kato, Shinsuke Inuki, Hiroaki Ohno, Barry Evans, Zi-xuan Wang, Stephen C. Peiper, Kazuki Izumi, Eiichi Kodama, Masao Matsuoka, Hideko Nagasawa, Shinya Oishi, Nobutaka Fujii Satoshi Ueda, Manabu Kato, Shinsuke Inuki, Hiroaki Ohno, Barry Evans, Zi-xuan Wang, Stephen C. Peiper, Kazuki Izumi, Eiichi Kodama, Masao Matsuoka, Hideko Nagasawa, Shinya Oishi, Nobutaka Fujii Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Bioorganic & Medicinal Chemistry Letters, 18, 14, 4124 Bioorganic & Medicinal Chemistry Letters, 18, 14, 4124 Bioorganic & Medicinal Chemistry Letters, 18, 14, 4124 2008/07 Refereed Disclose to all
Toshiaki Watanabe, Satoshi Ueda, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Toshiaki Watanabe, Satoshi Ueda, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno Toshiaki Watanabe, Satoshi Ueda, Shinsuke Inuki, Shinya Oishi, Nobutaka Fujii, Hiroaki Ohno One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling Chemical Communications, 43, 4516 Chemical Communications, 43, 4516 Chemical Communications, 43, 4516 2007 Refereed Disclose to all

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Title language:
Conference Activities & Talks
Title Title(Japanese) Title(English) Conference Conference(Japanese) Conference(English) Promotor Promotor(Japanese) Promotor(English) Date Language Assortment Disclose
免疫機構の調節に関わる複合脂質・糖質の合成と構造展開による生物有機化学研究 免疫機構の調節に関わる複合脂質・糖質の合成と構造展開による生物有機化学研究 平成30年度 天然物化学談話会 平成30年度 天然物化学談話会 2018/07/05 Disclose to all
免疫調節作用を有する化合物の合成と機能解析[Invited] 免疫調節作用を有する化合物の合成と機能解析 [Invited] ナノ・マイクロ横断型人材育成講演会 ナノ・マイクロ横断型人材育成講演会 2018/03/16 Japanese Oral presentation(invited, special) Disclose to all
脂質部位の構造展開を基盤とする新規CD1dリガンドの創製研究[Invited] 脂質部位の構造展開を基盤とする新規CD1dリガンドの創製研究 [Invited] 第11回 次世代アジュバント研究会 第11回 次世代アジュバント研究会 2018/01/23 Japanese Oral presentation(invited, special) Disclose to all
脂質改変型CD1dリガンドの創製研究[Invited] 脂質改変型CD1dリガンドの創製研究 [Invited] 生理化学研究ユニット第7 回シンポジウム 生理化学研究ユニット第7 回シンポジウム 2017/12/22 Japanese Oral presentation(invited, special) Disclose to all
Development of novel CD1d ligands containing modified lipid moieties[Invited] Development of novel CD1d ligands containing modified lipid moieties [Invited] Development of novel CD1d ligands containing modified lipid moieties [Invited] The Second A3 Roundtable Meeting on Chemical Probe Research Hub The Second A3 Roundtable Meeting on Chemical Probe Research Hub The Second A3 Roundtable Meeting on Chemical Probe Research Hub 2017/11/25 English Oral presentation(invited, special) Disclose to all
脂質部位の構造展開を基盤とするTh2サイトカイン選択的CD1dリガンドの創製研究 脂質部位の構造展開を基盤とするTh2サイトカイン選択的CD1dリガンドの創製研究 第35回 メディシナルケミストリーシンポジウム 第35回 メディシナルケミストリーシンポジウム 2017/10/26 Japanese Poster presentation Disclose to all
脂質改変型CD1dリガンドの創製研究 脂質改変型CD1dリガンドの創製研究 第四回 新学術領域研究「反応集積化が導く中分子戦略:高次生物機能分子の創製」若手シンポ 第四回 新学術領域研究「反応集積化が導く中分子戦略:高次生物機能分子の創製」若手シンポ 2017/08/18 Japanese Oral presentation(general) Disclose to all
Development of novel CD1d ligands modulating lipid-protein binding[Invited] Development of novel CD1d ligands modulating lipid-protein binding [Invited] A3アジア化学プローブ研究拠点事業若手研究者ミーティング A3アジア化学プローブ研究拠点事業若手研究者ミーティング 2017/07/12 English Oral presentation(invited, special) Disclose to all
Th2サイトカイン選択的誘導活性を有する新規CD1dリガンドの創製 Th2サイトカイン選択的誘導活性を有する新規CD1dリガンドの創製 日本ケミカルバイオロジー学会 第12回年会 日本ケミカルバイオロジー学会 第12回年会 2017/06/08 Japanese Poster presentation Disclose to all
脂質抗原受容体CD1dの脂質認識部位に存在する親水性アミノ酸残基の機能解析とその制御[Invited] 脂質抗原受容体CD1dの脂質認識部位に存在する親水性アミノ酸残基の機能解析とその制御 [Invited] 日本薬学会 第137年会 脂質結合タンパク質の構造生物学~最近の展開~ 日本薬学会 第137年会 脂質結合タンパク質の構造生物学~最近の展開~ 2017/03/25 Japanese Oral presentation(invited, special) Disclose to all
糖脂質α-GalCerを基盤とした脂質改変型CD1dリガンドの創製研究 糖脂質α-GalCerを基盤とした脂質改変型CD1dリガンドの創製研究 第22回 日本エンドトキシン・自然免疫研究会 第22回 日本エンドトキシン・自然免疫研究会 2016/12/03 Japanese Oral presentation(general) Disclose to all
糖脂質リガンドにおける脂質部位の構造展開を基盤とした新規CD1dリガンドの創製研究 糖脂質リガンドにおける脂質部位の構造展開を基盤とした新規CD1dリガンドの創製研究 第34回 メディシナルケミストリーシンポジウム 第34回 メディシナルケミストリーシンポジウム 2016/12/01 Japanese Oral presentation(general) Disclose to all
糖脂質リガンドにおける脂質部位の構造展開を基盤とした新規CD1dリガンドの創製研究[Invited] 糖脂質リガンドにおける脂質部位の構造展開を基盤とした新規CD1dリガンドの創製研究 [Invited] Schrödinger Japanese User Group Meeting 2016, Tokyo Schrödinger Japanese User Group Meeting 2016, Tokyo 2016/10/20 Japanese Oral presentation(invited, special) Disclose to all
CD1dの脂質認識部位への高親和性を指向した新規リガンドの創製研究 CD1dの脂質認識部位への高親和性を指向した新規リガンドの創製研究 第58回 天然物有機化合物討論会 第58回 天然物有機化合物討論会 2016/09/16 Japanese Oral presentation(general) Disclose to all
グラム陰性菌由来へプトース1β,7-ビスリン酸の合成研究 グラム陰性菌由来へプトース1β,7-ビスリン酸の合成研究 第35回 日本糖質学会 第35回 日本糖質学会 2016/09/02 Japanese Poster presentation Disclose to all
CD1dの脂質認識部位への高親和性を指向した新規リガンドの創製研究 CD1dの脂質認識部位への高親和性を指向した新規リガンドの創製研究 日本ケミカルバイオロジー学会 第11回年会 日本ケミカルバイオロジー学会 第11回年会 2016/06/15 Japanese Oral presentation(general) Disclose to all
Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives 2015 International Chemical Congress of Pacific Basin Societies 2015 International Chemical Congress of Pacific Basin Societies 2015 International Chemical Congress of Pacific Basin Societies 2015/12/18 English Poster presentation Disclose to all
Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives Decarboxylative Functionalization of β-Hydroxy Amino Acids via Photoredox Catalysis and Its Application to Synthesis of Functional 1,2-Amino Alcohol Derivatives The 13th International Kyoto Conference on New Aspects of Organic Chemistry The 13th International Kyoto Conference on New Aspects of Organic Chemistry The 13th International Kyoto Conference on New Aspects of Organic Chemistry 2015/11/11 English Poster presentation Disclose to all
Photoredox触媒を用いた光学活性1,2-アミノアルコール類の合成法開発 Photoredox触媒を用いた光学活性1,2-アミノアルコール類の合成法開発 第14回 新規素材探索研究会 第14回 新規素材探索研究会 2015/06/05 Japanese Poster presentation Disclose to all
パラジウム触媒によるブロモアレンとプロパルギル化合物の連続環化反応を利用したJaspine Bの全合成とその応用 パラジウム触媒によるブロモアレンとプロパルギル化合物の連続環化反応を利用したJaspine Bの全合成とその応用 第36回 反応と合成の進歩シンポジウム 第36回 反応と合成の進歩シンポジウム 2010/11 Japanese Oral presentation(general) Disclose to all
Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates Ring-Construction/Stereoselective Functionalization Cascade: Total Synthesis of Pachastrissamine (Jaspine B) through Palladium-Catalyzed Bis-cyclization of Bromoallenes and Propargyl Carbonates The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists The 5th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for Young Scientists 2010/05 English Oral presentation(general) Disclose to all
Direct Construction of the Ergot Alkaloid Scaffold by Palladium Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic acid, (±)-Lysergol and (±)-Isolysergol Direct Construction of the Ergot Alkaloid Scaffold by Palladium Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic acid, (±)-Lysergol and (±)-Isolysergol Direct Construction of the Ergot Alkaloid Scaffold by Palladium Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic acid, (±)-Lysergol and (±)-Isolysergol The 11th International KYOTO conference on New Aspects of Organic Chemistry The 11th International KYOTO conference on New Aspects of Organic Chemistry The 11th International KYOTO conference on New Aspects of Organic Chemistry 2009/11 English Poster presentation Disclose to all
A Direct Construction of Ergot Alkaloids Scaffold by Palladium-Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic Acid, Lysergol and Isolysergol A Direct Construction of Ergot Alkaloids Scaffold by Palladium-Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic Acid, Lysergol and Isolysergol A Direct Construction of Ergot Alkaloids Scaffold by Palladium-Catalyzed Domino Cyclization of Amino Allenes: Total Synthesis of (±)-Lysergic Acid, Lysergol and Isolysergol 41st National Organic Chemistry Symposium 41st National Organic Chemistry Symposium 41st National Organic Chemistry Symposium 2009/06 English Poster presentation Disclose to all
Pd触媒によるアレン連続環化反応を利用した Ergot Alkaloid 骨格の一挙構築法開発と応用 Pd触媒によるアレン連続環化反応を利用した Ergot Alkaloid 骨格の一挙構築法開発と応用 ケミカルバイオロジーシンポジウム ケミカルバイオロジーシンポジウム 2008/12 Japanese Poster presentation Disclose to all
Pd触媒によるアレン連続環化反応を利用したErgot alkaloid骨格の一挙構築法開発と応用 Pd触媒によるアレン連続環化反応を利用したErgot alkaloid骨格の一挙構築法開発と応用 第34回 反応と合成の進歩シンポジウム 第34回 反応と合成の進歩シンポジウム 2008/11 Japanese Poster presentation Disclose to all
Pd触媒によるアレン連続環化反応を利用したErgot alkaloid骨格の一挙構築法開発と応用 Pd触媒によるアレン連続環化反応を利用したErgot alkaloid骨格の一挙構築法開発と応用 第6回 次世代を担う有機化学シンポジウム 第6回 次世代を担う有機化学シンポジウム 2008/05 Japanese Oral presentation(general) Disclose to all
パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 日本薬学会 第128回年会 日本薬学会 第128回年会 2008/03 Japanese Oral presentation(general) Disclose to all
パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 第27回 有機合成若手セミナー 第27回 有機合成若手セミナー 2007/11 Japanese Poster presentation Disclose to all
パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 パラジウム触媒を用いたアレンの連続環化反応によるErgot alkaloid骨格の一挙構築 第57回 日本薬学会近畿支部総会・大会 第57回 日本薬学会近畿支部総会・大会 2007/10 Japanese Oral presentation(general) Disclose to all
One-pot Synthesis of Carbazoles by Palladium-catalyzed N-Arylation and Oxidative Coupling One-pot Synthesis of Carbazoles by Palladium-catalyzed N-Arylation and Oxidative Coupling One-pot Synthesis of Carbazoles by Palladium-catalyzed N-Arylation and Oxidative Coupling 6th AFMC Medicinal Chemistry Symposium (AIMECS 07) 6th AFMC Medicinal Chemistry Symposium (AIMECS 07) 6th AFMC Medicinal Chemistry Symposium (AIMECS 07) 2007/07 English Poster presentation Disclose to all

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Title language:
Books etc
Author Author(Japanese) Author(English) Title Title(Japanese) Title(English) Publisher Publisher(Japanese) Publisher(English) Publication date Language Type Disclose
Shinsuke Inuki 井貫 晋輔 Shinsuke Inuki Total Synthesis of Bioactive Natural Products by Palladium-Catalyzed Domino Cyclization of Allenes and Related Compounds. Total Synthesis of Bioactive Natural Products by Palladium-Catalyzed Domino Cyclization of Allenes and Related Compounds. Total Synthesis of Bioactive Natural Products by Palladium-Catalyzed Domino Cyclization of Allenes and Related Compounds. Springer Springer Springer 2011 Single Work Disclose to all
Title language:
Patents
Inventor(s) Inventor(s) (Japanese) Inventor(s) (English) Title Title(Japanese) Title(English) Stage Patent number Date Disclose
Inuki, S.; Hirata, N.; Kashiwabara, E.; Kishi, J.; Aiba, T.; Fujimoto, Y. Inuki, S.; Hirata, N.; Kashiwabara, E.; Kishi, J.; Aiba, T.; Fujimoto, Y. Inuki, S.; Hirata, N.; Kashiwabara, E.; Kishi, J.; Aiba, T.; Fujimoto, Y. Compound or Salt Thereof, Natural Killer T Cell Activator, and Pharmaceutical Composition. Compound or Salt Thereof, Natural Killer T Cell Activator, and Pharmaceutical Composition. Compound or Salt Thereof, Natural Killer T Cell Activator, and Pharmaceutical Composition. 特許出願 特願WO/2017/163808 Disclose to all
井貫 晋輔、藤本ゆかり、他 井貫 晋輔、藤本ゆかり、他 化合物又はその塩、ナチュラルキラーT細胞活性化剤、及び医薬組成物 化合物又はその塩、ナチュラルキラーT細胞活性化剤、及び医薬組成物 特許出願 特願2016-57416 Disclose to all
Furuyama, H.; Terao, T.; Nakagawa, D.; Tanabe, S.; Kato, T.; Yamamoto, M.; Sekine, S.; Mashiko, T.; Inuki, S.; Ueda, S. Furuyama, H.; Terao, T.; Nakagawa, D.; Tanabe, S.; Kato, T.; Yamamoto, M.; Sekine, S.; Mashiko, T.; Inuki, S.; Ueda, S. Furuyama, H.; Terao, T.; Nakagawa, D.; Tanabe, S.; Kato, T.; Yamamoto, M.; Sekine, S.; Mashiko, T.; Inuki, S.; Ueda, S. Nitorogen-containing Heterocyclic Compound of Salt Thereof. Nitorogen-containing Heterocyclic Compound of Salt Thereof. Nitorogen-containing Heterocyclic Compound of Salt Thereof. 特許出願 特願WO/2014/109414 Disclose to all
Takasaki, M.; Tsujino, T.; Tanabe, S.; Ookubo, M.; Sato, K.; Hirai, A.; Terada, D.; Inuki, S.; Mizumoto, S. Takasaki, M.; Tsujino, T.; Tanabe, S.; Ookubo, M.; Sato, K.; Hirai, A.; Terada, D.; Inuki, S.; Mizumoto, S. Takasaki, M.; Tsujino, T.; Tanabe, S.; Ookubo, M.; Sato, K.; Hirai, A.; Terada, D.; Inuki, S.; Mizumoto, S. Nitorogen-containing Heterocyclic Compound of Salt Thereof. Nitorogen-containing Heterocyclic Compound of Salt Thereof. Nitorogen-containing Heterocyclic Compound of Salt Thereof. 特許出願 特願WO/2013/157540 Disclose to all
Title language:
Awards
Title(Japanese) Title(English) Organization name(Japanese) Organization name(English) Date
Springer Theses Award ドイツSpringer社 2011/06/20
天然物化学談話会奨励賞 天然物化学談話会 2018/07/04
日本薬学会奨励賞 日本薬学会 2019/03/20
External funds: competitive funds and Grants-in-Aid for Scientific Research (Kakenhi)
Type Position Title(Japanese) Title(English) Period
若手研究(B) Representative 免疫におけるサイトカインバランスの制御を指向した脂質抗原受容体リガンドの創製研究 (平成29年度分) 2016/04/01-2019/03/31
新学術領域研究(研究領域提案型) Representative 腸管免疫に関わる化学シグナルの理解と制御を目指したケミカルツールの創製と機能解析 2018/04/01-2020/03/31
研究活動スタート支援 Representative 脂質抗原受容体CD1dの機能解明を目指した共有結合形成型リガンドの開発とその展開 2014/04/01-2016/03/31
基盤研究(B) Assignment 多環式骨格構築反応を基軸とする生物活性アルカロイドの全合成研究と創薬展開 2017/04/01-2018/03/31
基盤研究(B) Assignment 自然免疫-獲得免疫を制御する外因性・内因性分子の合成と機能解析、新規制御分子創製 2014/04/01-2017/03/31
日本医療研究開発機構 (AMED)・創薬基盤推進研究事業 Representative 脂質抗原受容体の機能を利用した新規糖脂質アジュバントの創製研究 2017/04/01-2020/03/31
特別研究員奨励費 Representative インドール系複素環化合物の高効率的合成法の開発と応用 2008/04/01-2011/03/31
若手研究(B) Representative 免疫におけるサイトカインバランスの制御を指向した脂質抗原受容体リガンドの創製研究 (平成30年度分) 2018/04/01-2019/03/31
新学術領域研究(研究領域提案型) Representative 腸管免疫に関わる化学シグナルの理解と制御を目指したケミカルツールの創製と機能解析 (平成30年度分) 2018/04/01-2019/03/31
External funds: other than those above
System Main person Title(Japanese) Title(English) Period
三島海雲記念財団学術研究奨励金 藤本ゆかり 食品および腸管内細菌・寄生虫の細胞表層脂質成分の合成と免疫調節機能解析 2017/04/01-2018/06/30
慶応工学会研究費援助 井貫晋輔 フォトレドックス触媒を用いた光学活性アミノアルコール類の効率的な合成法開発 2015/04/01-2016/03/31
金子・成田研究奨励金 井貫晋輔 NKT細胞活性化を担う脂質抗原受容体タンパク質の制御と機能解析 2014/04/01-2015/03/31
日本医療研究開発機構 (AMED)・年度医療研究開発推進事業費補助金 橋渡し研究加速ネットワークプログラム【シーズA】 藤本ゆかり 機能付加型セラミド含有糖脂質類およびそれらの免疫療法剤としての開発 2016/04/01-2017/03/31
上原記念生命科学財団 研究奨励金 井貫晋輔 自然リンパ球を制御するリガンドの探索と合成研究 2019/04/01-2020/03/31
上尾竹圓会 教育研究助成金 井貫晋輔 免疫調節活性を有する天然脂質化合物の合成と構造展開 2019/04/01-2020/03/31
Teaching subject(s)
Name(Japanese) Name(English) Term Department Period
ILASセミナー ILAS Seminar 前期 全学共通科目 2018/04-2019/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2018/04-2019/03
創薬有機化学エクササイズ1 Organic Chemistry Exercise 1 後期 薬学部 2018/04-2019/03
創薬有機化学エクササイズ2 Organic Chemistry Exercise 2 後期 薬学部 2018/04-2019/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2018/04-2019/03
基盤有機化学特論II Advanced Basic Organic Chemistry II 後期不定 薬学研究科 2018/04-2019/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2018/04-2019/03
創薬有機化学エクササイズ2 Organic Chemistry Exercise 2 後期 薬学部 2019/04-2020/03
創薬有機化学演習 Organic Chemistry Seminar 後期 薬学部 2019/04-2020/03
リード化合物探索スキル Skill Development for Lead Discovery 前期不定 薬学研究科 2019/04-2020/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2019/04-2020/03
基礎化学実験 Fundamental Chemical Experiments 後期 全学共通科目 2019/04-2020/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2019/04-2020/03

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Faculty management (title, position)
Title Period
NMR運営管理委員会 委員 2019/04/01-