大野 浩章

Last Update: 2018/06/13 12:57:01

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Name(Kanji/Kana/Abecedarium Latinum)
大野 浩章/オオノ ヒロアキ/Ohno, Hiroaki
Primary department(Org1/Job title)
Graduate Schools Pharmaceutical Sciences/Professor
Faculty
Org1 Job title
薬学部
Secondary departments to which you belong
Org1 Job title
Graduate Schools Pharmaceutical Sciences Professor
Contact address
Type Address(Japanese) Address(English)
Office 〒606-8501 京都市左京区吉田下阿達町46-29 46-29 Yoshidashimoadachi-cho, Sakyo-ku, Kyoto 606-8501, JAPAN
Phone
Type Number
Office 075-753-4571
Affiliated academic organization(s) (Japanese)
Organization name(Japanese) Organization name(English)
日本薬学会 The Pharmaceutical Society of Japan
有機合成化学協会 The Society of Synthetic Organic Chemistry, Japan
日本ペプチド学会 The Japanese Peptide Society
Academic degree
Field(Japanese) Field(English) University(Japanese) University(English) Method
修士(薬学) 京都大学
博士(薬学) 京都大学
Graduate school
University(Japanese) University(English) Faculty(Japanese) Faculty(English) Major(Japanese) Major(English) Degree
京都大学 大学院薬学研究科修士課程薬学専攻 修了
University
University(Japanese) University(English) Faculty(Japanese) Faculty(English) Major(s)(Japanese) Major(s)(English) Degree
京都大学 薬学部製薬化学科 卒業
Highschool
Highschool Kana
函館ラ・サール高等学校 はこだてら・さーるこうとうがっこう
Work Experience
Period Organization(Japanese) Organization(English) Job title(Japanese) Job title(English)
1999/01/01-1999/09/15 日本学術振興会 Japan Society for the Promotion of Science 特別研究員 JSPS Research Fellow
1999/09/16-2005/06/30 大阪大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Osaka University 助手 Assistant Professor
2005/07/01-2008/03/31 京都大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Kyoto University 助教授 Associate Professor
2008/04/01-2014/11/30 京都大学大学院薬学研究科 Graduate School of Pharmaceutical Sciences, Kyoto University 准教授 Associate Professor
2014/12/01- 京都大学国際高等教育院/薬学部・薬学研究科 Institute for Liberal Arts and Sciences/Graduate School of Pharmaceutical Sciences, Kyoto University 教授 Professor
Personal website address
URL
http://www.pharm.kyoto-u.ac.jp//seizo/
ORCID ID
orcid.org/0000-0002-3246-4809
Research Topics
(Japanese)
連続反応及び高原子効率反応による有機合成の効率化
(English)
Efficiency Improvement of Synthetic Organic Chemistry Based on Cascade and Atom-Economical Reactions
Overview of your research
(Japanese)
高い原子効率を有する素反応の開発やその連続化を通じて有機合成の効率化を図るとともに、有用な物質の効率的合成法の開発と創薬展開を行う。
(English)
Improvement of reaction efficiency by development of novel atom-economical cascade reactions, synthetic studies of bioactive compounds, and their medicinal application studies are conducted.
Fields of research (key words)
Key words(Japanese) Key words(English)
カスケード反応 cascade reactions
反応集積化 Reaction Integration
遷移金属 Transitiom Metals
含窒素複素環 Nitrogen Heterocycles
天然物合成 Natural Product Syntheses
Fields of research (kaken code)
Kaken code
Chemical pharmaceutical science
Organic chemistry
Published Papers
Author Author(Japanese) Author(English) Title Title(Japanese) Title(English) Bibliography Bibliography(Japanese) Bibliography(English) Publication date Refereed paper Language Publishing type Disclose
Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Ohara T, Kaneda M, Saito T, Fujii N, Ohno H, Oishi S Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Head-to-tail macrocyclization of cysteine-free peptides using an o-aminoanilide linker. Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 Bioorganic & medicinal chemistry letters, 28, 8, 1283-1286 2018/05 Refereed Disclose to all
Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Kobayashi Y, Hoshino M, Kameda T, Kobayashi K, Akaji K, Inuki S, Ohno H, Oishi S Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Use of a Compact Tripodal Tris(bipyridine) Ligand to Stabilize a Single-Metal-Centered Chirality: Stereoselective Coordination of Iron(II) and Ruthenium(II) on a Semirigid Hexapeptide Macrocycle. Inorganic chemistry Inorganic chemistry Inorganic chemistry 2018/04 Refereed Disclose to all
Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Sekiguchi H, Kuroyanagi T, Rhainds D, Kobayashi K, Kobayashi Y, Ohno H, Heveker N, Akaji K, Fujii N, Oishi S Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Structure-Activity Relationship Study of Cyclic Pentapeptide Ligands for Atypical Chemokine Receptor 3 (ACKR3). Journal of medicinal chemistry Journal of medicinal chemistry Journal of medicinal chemistry 2018/04 Refereed Disclose to all
Kaneda M, Inuki S, Ohno H, Oishi S Kaneda M, Inuki S, Ohno H, Oishi S Kaneda M, Inuki S, Ohno H, Oishi S Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. Total Synthesis and Stereochemical Revision of Stereocalpin A: Mirror-Image Approach for Stereochemical Assignments of the Peptide-Polyketide Macrocycle. The Journal of organic chemistry, 83, 6, 3047-3060 The Journal of organic chemistry, 83, 6, 3047-3060 The Journal of organic chemistry, 83, 6, 3047-3060 2018/03/16 Refereed Disclose to all
Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Kobayashi Y, Kameda T, Hoshino M, Fujii N, Ohno H, Oishi S Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Fe(ii)-Complexation of tripodal hexapeptide ligands with three bidentate triazolylpyridines: induction of metal-centred chirality by peptide macrocyclization. Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 Dalton transactions (Cambridge, England : 2003), 46, 40, 13673-13676 2017/10 Refereed Disclose to all
Hamada N, Yoshida Y, Oishi S, Ohno H Hamada N, Yoshida Y, Oishi S, Ohno H Hamada N, Yoshida Y, Oishi S, Ohno H Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Gold-Catalyzed Cascade Reaction of Skipped Diynes for the Construction of a Cyclohepta[b]pyrrole Scaffold. Organic letters, 19, 14, 3875-3878 Organic letters, 19, 14, 3875-3878 Organic letters, 19, 14, 3875-3878 2017/07 Refereed Disclose to all
Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Matsuoka J, Matsuda Y, Kawada Y, Oishi S, Ohno H Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Total Synthesis of Dictyodendrins by the Gold-Catalyzed Cascade Cyclization of Conjugated Diynes with Pyrroles. Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 Angewandte Chemie (International ed. in English), 56, 26, 7444-7448 2017/06 Refereed Disclose to all
Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Ohno H, Honda M, Hamada N, Miyagaki J, Iwata A, Otsuki K, Maruyama T, Nakamura S, Nakanishi I, Inuki S, Fujii N, Oishi S Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Identification of selective inhibitors of sphingosine kinases 1 and 2 through a structure-activity relationship study of 4-epi-jaspine B. Bioorganic & medicinal chemistry, 25, 12, 3046-3052 Bioorganic & medicinal chemistry, 25, 12, 3046-3052 Bioorganic & medicinal chemistry, 25, 12, 3046-3052 2017/06 Refereed Disclose to all
Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Ishiba H, Noguchi T, Shu K, Ohno H, Honda K, Kondoh Y, Osada H, Fujii N, Oishi S Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Investigation of the inhibitory mechanism of apomorphine against MDM2-p53 interaction. Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 Bioorganic & medicinal chemistry letters, 27, 11, 2571-2574 2017/06 Refereed Disclose to all
Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Noguchi T, Ishiba H, Honda K, Kondoh Y, Osada H, Ohno H, Fujii N, Oishi S Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Synthesis of Grb2 SH2 Domain Proteins for Mirror-Image Screening Systems. Bioconjugate chemistry, 28, 2, 609-619 Bioconjugate chemistry, 28, 2, 609-619 Bioconjugate chemistry, 28, 2, 609-619 2017/02 Refereed Disclose to all
Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Kaneda M, Sueyoshi K, Teruya T, Ohno H, Fujii N, Oishi S Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Total synthesis of odoamide, a novel cyclic depsipeptide, from an Okinawan marine cyanobacterium. Organic & biomolecular chemistry, 14, 38, 9104 Organic & biomolecular chemistry, 14, 38, 9104 Organic & biomolecular chemistry, 14, 38, 9104 2016/09 Refereed Disclose to all
Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Naoe S, Yoshida Y, Oishi S, Fujii N, Ohno H Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. Total Synthesis of (+)-Conolidine by the Gold(I)-Catalyzed Cascade Cyclization of a Conjugated Enyne. The Journal of organic chemistry, 81, 13, 5698 The Journal of organic chemistry, 81, 13, 5698 The Journal of organic chemistry, 81, 13, 5698 2016/07 Refereed Disclose to all
Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Hattori Y, Machida Y, Honda M, Takeuchi N, Yoshiike Y, Ohno H, Onishi H Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Small interfering RNA delivery into the liver by cationic cholesterol derivative-based liposomes. Journal of liposome research, 1-10 Journal of liposome research, 1-10 Journal of liposome research, 1-10 2016/06 Refereed Disclose to all
Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Ohno H, Osada H, Fujii N Screening of a virtual mirror-image library of natural products. Screening of a virtual mirror-image library of natural products. Screening of a virtual mirror-image library of natural products. Chemical communications (Cambridge, England), 52, 49, 7656 Chemical communications (Cambridge, England), 52, 49, 7656 Chemical communications (Cambridge, England), 52, 49, 7656 2016/06 Refereed Disclose to all
Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Yamamoto K, Okazaki S, Ohno H, Matsuda F, Ohkura S, Maeda KI, Fujii N, Oishi S Development of novel NK3 receptor antagonists with reduced environmental impact. Development of novel NK3 receptor antagonists with reduced environmental impact. Development of novel NK3 receptor antagonists with reduced environmental impact. Bioorganic & medicinal chemistry, 24, 16, 3500 Bioorganic & medicinal chemistry, 24, 16, 3500 Bioorganic & medicinal chemistry, 24, 16, 3500 2016/05 Refereed Disclose to all
Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Nishiyama D, Ohara A, Chiba H, Kumagai H, Oishi S, Fujii N, Ohno H Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Formal Total Synthesis of (±)-Strictamine Based on a Gold-Catalyzed Cyclization. Organic letters, 18, 7, 1673 Organic letters, 18, 7, 1673 Organic letters, 18, 7, 1673 2016/04 Refereed Disclose to all
Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Ohno H, Minamiguchi D, Nakamura S, Shu K, Okazaki S, Honda M, Misu R, Moriwaki H, Nakanishi S, Oishi S, Kinoshita T, Nakanishi I, Fujii N Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Structure-activity relationship study of 4-(thiazol-5-yl)benzoic acid derivatives as potent protein kinase CK2 inhibitors. Bioorganic & medicinal chemistry, 24, 5, 1141 Bioorganic & medicinal chemistry, 24, 5, 1141 Bioorganic & medicinal chemistry, 24, 5, 1141 2016/03 Refereed Disclose to all
Wagner B, Hiller W, Ohno H, Krause N Wagner B, Hiller W, Ohno H, Krause N Wagner B, Hiller W, Ohno H, Krause N Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Gold-catalyzed three-component spirocyclization: a one-pot approach to functionalized pyrazolidines. Organic & biomolecular chemistry, 14, 5, 1583 Organic & biomolecular chemistry, 14, 5, 1583 Organic & biomolecular chemistry, 14, 5, 1583 2016/02 Refereed Disclose to all
Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Nishiyama D, Sakai Y, Sekiguchi H, Chiba H, Misu R, Oishi S, Fujii N, Ohno H Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Novel 3,4,7-Substituted Benzofuran Derivatives Having Binding Affinity to κ-Opioid Receptor. Chemical & pharmaceutical bulletin, 64, 7, 1003 Chemical & pharmaceutical bulletin, 64, 7, 1003 Chemical & pharmaceutical bulletin, 64, 7, 1003 2016 Refereed Disclose to all
Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Taguchi M, Tokimizu Y, Oishi S, Fujii N, Ohno H Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Synthesis of Fused Carbazoles by Gold-Catalyzed Tricyclization of Conjugated Diynes via Rearrangement of an N-Propargyl Group. Organic letters, 17, 24, 6250-6253 Organic letters, 17, 24, 6250-6253 Organic letters, 17, 24, 6250-6253 2015/12 Refereed Disclose to all
Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Oishi S, Kuroyanagi T, Kubo T, Montpas N, Yoshikawa Y, Misu R, Kobayashi Y, Ohno H, Heveker N, Furuya T, Fujii N Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Development of Novel CXC Chemokine Receptor 7 (CXCR7) Ligands: Selectivity Switch from CXCR4 Antagonists with a Cyclic Pentapeptide Scaffold. Journal of medicinal chemistry, 58, 13, 5218-5225 Journal of medicinal chemistry, 58, 13, 5218-5225 Journal of medicinal chemistry, 58, 13, 5218-5225 2015/06 Refereed Disclose to all
Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group. Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 Angewandte Chemie (International ed. in English), 54, 27, 7862-7866 2015/05 Refereed Disclose to all
Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Okazaki S, Oishi S, Mizuhara T, Shimura K, Murayama H, Ohno H, Matsuoka M, Fujii N Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Investigations of possible prodrug structures for 2-(2-mercaptophenyl)tetrahydropyrimidines: reductive conversion from anti-HIV agents with pyrimidobenzothiazine and isothiazolopyrimidine scaffolds. Organic & biomolecular chemistry, 13, 16, 4706-4713 Organic & biomolecular chemistry, 13, 16, 4706-4713 Organic & biomolecular chemistry, 13, 16, 4706-4713 2015/04 Refereed Disclose to all
Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Naoe S, Saito T, Uchiyama M, Oishi S, Fujii N, Ohno H Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Direct construction of fused indoles by gold-catalyzed cascade cyclization of conjugated diynes. Organic letters, 17, 7, 1774-1777 Organic letters, 17, 7, 1774-1777 Organic letters, 17, 7, 1774-1777 2015/04 Refereed Disclose to all
Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Okazaki S, Mizuhara T, Shimura K, Murayama H, Ohno H, Oishi S, Matsuoka M, Fujii N Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold. Bioorganic & medicinal chemistry, 23, 7, 1447-1452 Bioorganic & medicinal chemistry, 23, 7, 1447-1452 Bioorganic & medicinal chemistry, 23, 7, 1447-1452 2015/04 Refereed Disclose to all
Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Tokimizu Y, Wieteck M, Rudolph M, Oishi S, Fujii N, Hashmi AS, Ohno H Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Dual gold catalysis: a novel synthesis of bicyclic and tricyclic pyrroles from N-propargyl ynamides. Organic letters, 17, 3, 604-607 Organic letters, 17, 3, 604-607 Organic letters, 17, 3, 604-607 2015/02 Refereed Disclose to all
Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Nabika R, Suyama TL, Hau AM, Misu R, Ohno H, Ishmael JE, McPhail KL, Oishi S, Fujii N Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Synthesis and biological evaluation of the [d-MeAla(11)]-epimer of coibamide A. Bioorganic & medicinal chemistry letters, 25, 2, 302-306 Bioorganic & medicinal chemistry letters, 25, 2, 302-306 Bioorganic & medicinal chemistry letters, 25, 2, 302-306 2015/01 Refereed Disclose to all
Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Matsuda Y, Naoe S, Oishi S, Fujii N, Ohno H Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Formal [4+2] reaction between 1,3-diynes and pyrroles: gold(I)-catalyzed indole synthesis by double hydroarylation. Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 Chemistry (Weinheim an der Bergstrasse, Germany), 21, 4, 1463-1467 2015/01 Refereed Disclose to all
Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E Hattori Y, Hara E, Shingu Y, Minamiguchi D, Nakamura A, Arai S, Ohno H, Kawano K, Fujii N, Yonemochi E siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. siRNA delivery into tumor cells by cationic cholesterol derivative-based nanoparticles and liposomes. Biological & pharmaceutical bulletin, 38, 1, 30-38 Biological & pharmaceutical bulletin, 38, 1, 30-38 Biological & pharmaceutical bulletin, 38, 1, 30-38 2015 Refereed Disclose to all
Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A Shi J, Liu N, Xiao Y, Takei Y, Yasue M, Suzuki Y, Hou Z, Ohno H, Yamada M, Fuchi N, Oshida K, Miyamoto Y, Tsujimoto G, Hirasawa A The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. The Effects of a Selective CK2 Inhibitor on Anti-glomerular Basement Membrane Glomerulonephritis in Rats. Biological & pharmaceutical bulletin, 38, 9, 1345-1351 Biological & pharmaceutical bulletin, 38, 9, 1345-1351 Biological & pharmaceutical bulletin, 38, 9, 1345-1351 2015 Refereed Disclose to all
Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Wieteck M, Tokimizu Y, Rudolph M, Rominger F, Ohno H, Fujii N, Hashmi AS Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Dual gold catalysis: synthesis of polycyclic compounds via C-H insertion of gold vinylidenes. Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 Chemistry (Weinheim an der Bergstrasse, Germany), 20, 49, 16331-16336 2014/12 Refereed Disclose to all
Nabika R, Oishi S, Misu R, Ohno H, Fujii N Nabika R, Oishi S, Misu R, Ohno H, Fujii N Nabika R, Oishi S, Misu R, Ohno H, Fujii N Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Synthesis of IB-01212 by multiple N-methylations of peptide bonds. Bioorganic & medicinal chemistry, 22, 21, 6156-6162 Bioorganic & medicinal chemistry, 22, 21, 6156-6162 Bioorganic & medicinal chemistry, 22, 21, 6156-6162 2014/11 Refereed Disclose to all
Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Misu R, Oishi S, Yamada A, Yamamura T, Matsuda F, Yamamoto K, Noguchi T, Ohno H, Okamura H, Ohkura S, Fujii N Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Development of novel neurokinin 3 receptor (NK3R) selective agonists with resistance to proteolytic degradation. Journal of medicinal chemistry, 57, 20, 8646-8651 Journal of medicinal chemistry, 57, 20, 8646-8651 Journal of medicinal chemistry, 57, 20, 8646-8651 2014/10 Refereed Disclose to all
Ohno H Ohno H Ohno H Synthesis and applications of vinylaziridines and ethynylaziridines. Synthesis and applications of vinylaziridines and ethynylaziridines. Synthesis and applications of vinylaziridines and ethynylaziridines. Chemical reviews, 114, 16, 7784-7814 Chemical reviews, 114, 16, 7784-7814 Chemical reviews, 114, 16, 7784-7814 2014/08 Refereed Disclose to all
Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Suzuki T, Sakano Y, Tokimizu Y, Miura Y, Katoono R, Fujiwara K, Yoshioka N, Fujii N, Ohno H Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Wurster's Blue-type cation radicals framed in a 5,10-dihydrobenzo[a]indolo[2,3-c]carbazole (BIC) skeleton: dual electrochromism with drastic changes in UV/Vis/NIR and fluorescence. Chemistry, an Asian journal, 9, 7, 1841-1846 Chemistry, an Asian journal, 9, 7, 1841-1846 Chemistry, an Asian journal, 9, 7, 1841-1846 2014/07 Refereed Disclose to all
Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Kaneda M, Misu R, Ohno H, Hirasawa A, Ieda N, Uenoyama Y, Tsukamura H, Maeda K, Oishi S, Fujii N Design and synthesis of fluorescent probes for GPR54. Design and synthesis of fluorescent probes for GPR54. Design and synthesis of fluorescent probes for GPR54. Bioorganic & medicinal chemistry, 22, 13, 3325-3330 Bioorganic & medicinal chemistry, 22, 13, 3325-3330 Bioorganic & medicinal chemistry, 22, 13, 3325-3330 2014/07 Refereed Disclose to all
Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Tokimizu Y, Oishi S, Fujii N, Ohno H Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Gold-catalyzed cascade cyclization of (azido)ynamides: an efficient strategy for the construction of indoloquinolines. Organic letters, 16, 11, 3138-3141 Organic letters, 16, 11, 3138-3141 Organic letters, 16, 11, 3138-3141 2014/06 Refereed Disclose to all
Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Takeuchi T, Oishi S, Kaneda M, Misu R, Ohno H, Sawada J, Asai A, Nakamura S, Nakanishi I, Fujii N Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Optimization of diaryl amine derivatives as kinesin spindle protein inhibitors. Bioorganic & medicinal chemistry, 22, 12, 3171-3179 Bioorganic & medicinal chemistry, 22, 12, 3171-3179 Bioorganic & medicinal chemistry, 22, 12, 3171-3179 2014/06 Refereed Disclose to all
Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Takeuchi T, Oishi S, Kaneda M, Ohno H, Nakamura S, Nakanishi I, Yamane M, Sawada J, Asai A, Fujii N Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. Kinesin spindle protein inhibitors with diaryl amine scaffolds: crystal packing analysis for improved aqueous solubility. ACS medicinal chemistry letters, 5, 5, 566-571 ACS medicinal chemistry letters, 5, 5, 566-571 ACS medicinal chemistry letters, 5, 5, 566-571 2014/05 Refereed Disclose to all
A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Iwata A, Inuki S, Oishi S, Fujii N, Ohno H A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation. Synthesis of fused tetracyclic spiroindoles via palladium-catalysed cascade cyclisation Chemical Communications, 50, 3, 298-300 Chemical communications (Cambridge, England), 50, 3, 298-300 Chemical Communications, 50, 3, 298-300 2014/01 Refereed English Disclose to all
T. Mizuhara; T. Kato; A. Hirai; H. Kurihara; Y. Shimada; M. Taniguchi; H. Maeta; H. Togami; K. Shimura; M. Matsuoka; S. Okazaki; T. Takeuchi; H. Ohno; S. Oishi; N. Fujii Mizuhara T, Kato T, Hirai A, Kurihara H, Shimada Y, Taniguchi M, Maeta H, Togami H, Shimura K, Matsuoka M, Okazaki S, Takeuchi T, Ohno H, Oishi S, Fujii N T. Mizuhara; T. Kato; A. Hirai; H. Kurihara; Y. Shimada; M. Taniguchi; H. Maeta; H. Togami; K. Shimura; M. Matsuoka; S. Okazaki; T. Takeuchi; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents. Structure-activity relationship study of phenylpyrazole derivatives as a novel class of anti-HIV agents Bioorganic and Medicinal Chemistry Letters, 23, 16, 4557-4561 Bioorganic & medicinal chemistry letters, 23, 16, 4557-4561 Bioorganic and Medicinal Chemistry Letters, 23, 16, 4557-4561 2013/08 Refereed English Disclose to all
T. Noguchi; S. Oishi; K. Honda; Y. Kondoh; T. Saito; T. Kubo; M. Kaneda; H. Ohno; H. Osada; N. Fujii Noguchi T, Oishi S, Honda K, Kondoh Y, Saito T, Kubo T, Kaneda M, Ohno H, Osada H, Fujii N T. Noguchi; S. Oishi; K. Honda; Y. Kondoh; T. Saito; T. Kubo; M. Kaneda; H. Ohno; H. Osada; N. Fujii Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: identification of novel peptidic inhibitors. Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors Bioorganic and Medicinal Chemistry Letters, 23, 13, 3802-3805 Bioorganic & medicinal chemistry letters, 23, 13, 3802-3805 Bioorganic and Medicinal Chemistry Letters, 23, 13, 3802-3805 2013/07 Refereed English Disclose to all
Y. Kobayashi; S. Oishi; K. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Kobayashi Y, Oishi S, Kobayashi K, Ohno H, Tsutsumi H, Hata Y, Fujii N Y. Kobayashi; S. Oishi; K. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Synthesis and functional analysis of deferriferrichrysin derivatives: Application to colorimetric pH indicators Synthesis and functional analysis of deferriferrichrysin derivatives: application to colorimetric pH indicators. Synthesis and functional analysis of deferriferrichrysin derivatives: Application to colorimetric pH indicators Bioorganic and Medicinal Chemistry, 21, 14, 4296-4300 Bioorganic & medicinal chemistry, 21, 14, 4296-4300 Bioorganic and Medicinal Chemistry, 21, 14, 4296-4300 2013/07 Refereed English Disclose to all
H. Chiba; Y. Sakai; A. Ohara; S. Oishi; N. Fujii; H. Ohno Chiba H, Sakai Y, Ohara A, Oishi S, Fujii N, Ohno H H. Chiba; Y. Sakai; A. Ohara; S. Oishi; N. Fujii; H. Ohno Convergent synthesis of (-)-quinocarcin based on the combination of sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination Convergent synthesis of (-)-quinocarcin based on the combination of Sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination. Convergent synthesis of (-)-quinocarcin based on the combination of sonogashira coupling and gold(I)-catalyzed 6-endo-dig hydroamination Chemistry - A European Journal, 19, 27, 8875-8883 Chemistry (Weinheim an der Bergstrasse, Germany), 19, 27, 8875-8883 Chemistry - A European Journal, 19, 27, 8875-8883 2013/07 Refereed English Disclose to all
Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: Synthetic study of laurendecumallene B Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: synthetic study of laurendecumallene B. Palladium-catalyzed medium-ring formation for construction of the core structure of laurencia oxacycles: Synthetic study of laurendecumallene B Organic Letters, 15, 12, 3046-3049 Organic letters, 15, 12, 3046-3049 Organic Letters, 15, 12, 3046-3049 2013/06 Refereed English Disclose to all
Z. Hou; S. Oishi; Y. Suzuki; T. Kure; I. Nakanishi; A. Hirasawa; G. Tsujimoto; H. Ohno; N. Fujii Hou Z, Oishi S, Suzuki Y, Kure T, Nakanishi I, Hirasawa A, Tsujimoto G, Ohno H, Fujii N Z. Hou; S. Oishi; Y. Suzuki; T. Kure; I. Nakanishi; A. Hirasawa; G. Tsujimoto; H. Ohno; N. Fujii Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: Application to the development of a new class of CK2 inhibitors Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: application to the development of a new class of CK2 inhibitors. Diversity-oriented synthesis of pyrazolo[4,3-b]indoles by gold-catalysed three-component annulation: Application to the development of a new class of CK2 inhibitors Organic and Biomolecular Chemistry, 11, 20, 3288-3296 Organic & biomolecular chemistry, 11, 20, 3288-3296 Organic and Biomolecular Chemistry, 11, 20, 3288-3296 2013/05 Refereed English Disclose to all
R. Misu; S. Oishi; S. Setsuda; T. Noguchi; M. Kaneda; H. Ohno; B. Evans; J.-M. Navenot; S.C. Peiper; N. Fujii Misu R, Oishi S, Setsuda S, Noguchi T, Kaneda M, Ohno H, Evans B, Navenot JM, Peiper SC, Fujii N R. Misu; S. Oishi; S. Setsuda; T. Noguchi; M. Kaneda; H. Ohno; B. Evans; J.-M. Navenot; S.C. Peiper; N. Fujii Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes. Characterization of the receptor binding residues of kisspeptins by positional scanning using peptide photoaffinity probes Bioorganic and Medicinal Chemistry Letters, 23, 9, 2628-2631 Bioorganic & medicinal chemistry letters, 23, 9, 2628-2631 Bioorganic and Medicinal Chemistry Letters, 23, 9, 2628-2631 2013/05 Refereed English Disclose to all
R. Misu; T. Noguchi; H. Ohno; S. Oishi; N. Fujii Misu R, Noguchi T, Ohno H, Oishi S, Fujii N R. Misu; T. Noguchi; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists. Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists Bioorganic and Medicinal Chemistry, 21, 8, 2413-2417 Bioorganic & medicinal chemistry, 21, 8, 2413-2417 Bioorganic and Medicinal Chemistry, 21, 8, 2413-2417 2013/04 Refereed English Disclose to all
T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182 Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182. Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182 Bioorganic and Medicinal Chemistry, 21, 7, 2079-2087 Bioorganic & medicinal chemistry, 21, 7, 2079-2087 Bioorganic and Medicinal Chemistry, 21, 7, 2079-2087 2013/04 Refereed English Disclose to all
Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani SiRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine siRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine. SiRNA delivery into tumor cells by lipid-based nanoparticles composed of hydroxyethylated cholesteryl triamine International Journal of Pharmaceutics, 443, 1-2, 221-229 International journal of pharmaceutics, 443, 1-2, 221-229 International Journal of Pharmaceutics, 443, 1-2, 221-229 2013/02 Refereed English Disclose to all
Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani Hattori Y, Nakamura T, Ohno H, Fujii N, Maitani Y Y. Hattori; T. Nakamura; H. Ohno; N. Fujii; Y. Maitani Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine. Enhanced plasmid DNA transfer into tumor cells by nanoparticle composed of cholesteryl triamine and diamine Biological and Pharmaceutical Bulletin, 36, 5, 856-860 Biological & pharmaceutical bulletin, 36, 5, 856-860 Biological and Pharmaceutical Bulletin, 36, 5, 856-860 2013 Refereed English Disclose to all
T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin- 6-imine derivatives for potent anti-HIV agents Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents. Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin- 6-imine derivatives for potent anti-HIV agents Bioorganic and Medicinal Chemistry, 20, 21, 6434-6441 Bioorganic & medicinal chemistry, 20, 21, 6434-6441 Bioorganic and Medicinal Chemistry, 20, 21, 6434-6441 2012/11 Refereed English Disclose to all
H. Chiba; S. Oishi; N. Fujii; H. Ohno Chiba H, Oishi S, Fujii N, Ohno H H. Chiba; S. Oishi; N. Fujii; H. Ohno Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination. Total synthesis of (-)-quinocarcin by gold(I)-catalyzed regioselective hydroamination Angewandte Chemie - International Edition, 51, 36, 9169-9172 Angewandte Chemie (International ed. in English), 51, 36, 9169-9172 Angewandte Chemie - International Edition, 51, 36, 9169-9172 2012/09 Refereed English Disclose to all
T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Mizuhara T, Oishi S, Ohno H, Shimura K, Matsuoka M, Fujii N T. Mizuhara; S. Oishi; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3] benzothiazin-6-imines and related tricyclic heterocycles Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles. Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3] benzothiazin-6-imines and related tricyclic heterocycles Organic and Biomolecular Chemistry, 10, 33, 6792-6802 Organic & biomolecular chemistry, 10, 33, 6792-6802 Organic and Biomolecular Chemistry, 10, 33, 6792-6802 2012/09 Refereed English Disclose to all
Y. Suzuki; S. Oishi; Y. Takei; M. Yasue; R. Misu; S. Naoe; Z. Hou; T. Kure; I. Nakanishi; H. Ohno; A. Hirasawa; G. Tsujimoto; N. Fujii Suzuki Y, Oishi S, Takei Y, Yasue M, Misu R, Naoe S, Hou Z, Kure T, Nakanishi I, Ohno H, Hirasawa A, Tsujimoto G, Fujii N Y. Suzuki; S. Oishi; Y. Takei; M. Yasue; R. Misu; S. Naoe; Z. Hou; T. Kure; I. Nakanishi; H. Ohno; A. Hirasawa; G. Tsujimoto; N. Fujii Design and synthesis of a novel class of CK2 inhibitors: Application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles. Design and synthesis of a novel class of CK2 inhibitors: Application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles Organic and Biomolecular Chemistry, 10, 25, 4907-4915 Organic & biomolecular chemistry, 10, 25, 4907-4915 Organic and Biomolecular Chemistry, 10, 25, 4907-4915 2012/07 Refereed English Disclose to all
S. Naoe; Y. Suzuki; K. Hirano; Y. Inaba; S. Oishi; N. Fujii; H. Ohno Naoe S, Suzuki Y, Hirano K, Inaba Y, Oishi S, Fujii N, Ohno H S. Naoe; Y. Suzuki; K. Hirano; Y. Inaba; S. Oishi; N. Fujii; H. Ohno Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes. Gold(I)-catalyzed regioselective inter-/intramolecular addition cascade of di- and triynes for direct construction of substituted naphthalenes Journal of Organic Chemistry, 77, 11, 4907-4916 The Journal of organic chemistry, 77, 11, 4907-4916 Journal of Organic Chemistry, 77, 11, 4907-4916 2012/06 Refereed English Disclose to all
R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; Y. Yano; K. Matsuzaki; J.-M. Navenot; S.C. Peiper; N. Fujii Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Yano Y, Matsuzaki K, Navenot JM, Peiper SC, Fujii N R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; Y. Yano; K. Matsuzaki; J.-M. Navenot; S.C. Peiper; N. Fujii Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists. Paradoxical downregulation of CXC chemokine receptor 4 induced by polyphemusin II-derived antagonists Bioconjugate Chemistry, 23, 6, 1259-1265 Bioconjugate chemistry, 23, 6, 1259-1265 Bioconjugate Chemistry, 23, 6, 1259-1265 2012/06 Refereed English Disclose to all
Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Masuda R, Oishi S, Tanahara N, Ohno H, Hirasawa A, Tsujimoto G, Kodama E, Matsuoka M, Fujii N Development and application of fluorescent SDF-1 derivatives. Development and application of fluorescent SDF-1 derivatives. Development and application of fluorescent SDF-1 derivatives. Future medicinal chemistry, 4, 7, 837-844 Future medicinal chemistry, 4, 7, 837-844 Future medicinal chemistry, 4, 7, 837-844 2012/05 Refereed Disclose to all
H. Ohno; M. Iuchi; N. Kojima; T. Yoshimitsu; N. Fujii; T. Tanaka Ohno H, Iuchi M, Kojima N, Yoshimitsu T, Fujii N, Tanaka T H. Ohno; M. Iuchi; N. Kojima; T. Yoshimitsu; N. Fujii; T. Tanaka Double C-H functionalization in sequential order: Direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade Double C-H functionalization in sequential order: direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade. Double C-H functionalization in sequential order: Direct synthesis of polycyclic compounds by a palladium-catalyzed C-H alkenylation-arylation cascade Chemistry - A European Journal, 18, 17, 5352-5360 Chemistry (Weinheim an der Bergstrasse, Germany), 18, 17, 5352-5360 Chemistry - A European Journal, 18, 17, 5352-5360 2012/04 Refereed English Disclose to all
K. Kobayashi; S. Oishi; Y. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Kobayashi K, Oishi S, Kobayashi Y, Ohno H, Tsutsumi H, Hata Y, Fujii N K. Kobayashi; S. Oishi; Y. Kobayashi; H. Ohno; H. Tsutsumi; Y. Hata; N. Fujii Synthesis and application of an N <sup>δ</sup>-acetyl-N <sup>δ</sup>-hydroxyornithine analog: Identification of novel metal complexes of deferriferrichrysin Synthesis and application of an Nδ-acetyl-Nδ-hydroxyornithine analog: identification of novel metal complexes of deferriferrichrysin. Synthesis and application of an N <sup>δ</sup>-acetyl-N <sup>δ</sup>-hydroxyornithine analog: Identification of novel metal complexes of deferriferrichrysin Bioorganic and Medicinal Chemistry, 20, 8, 2651-2655 Bioorganic & medicinal chemistry, 20, 8, 2651-2655 Bioorganic and Medicinal Chemistry, 20, 8, 2651-2655 2012/04 Refereed English Disclose to all
K. Kobayashi; S. Oishi; R. Hayashi; K. Tomita; T. Kubo; N. Tanahara; H. Ohno; Y. Yoshikawa; T. Furuya; M. Hoshino; N. Fujii Kobayashi K, Oishi S, Hayashi R, Tomita K, Kubo T, Tanahara N, Ohno H, Yoshikawa Y, Furuya T, Hoshino M, Fujii N K. Kobayashi; S. Oishi; R. Hayashi; K. Tomita; T. Kubo; N. Tanahara; H. Ohno; Y. Yoshikawa; T. Furuya; M. Hoshino; N. Fujii Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres. Structure-activity relationship study of a CXC chemokine receptor type 4 antagonist, FC131, using a series of alkene dipeptide isosteres Journal of Medicinal Chemistry, 55, 6, 2746-2757 Journal of medicinal chemistry, 55, 6, 2746-2757 Journal of Medicinal Chemistry, 55, 6, 2746-2757 2012/03 Refereed English Disclose to all
Z. Hou; I. Nakanishi; T. Kinoshita; Y. Takei; M. Yasue; R. Misu; Y. Suzuki; S. Nakamura; T. Kure; H. Ohno; K. Murata; K. Kitaura; A. Hirasawa; G. Tsujimoto; S. Oishi; N. Fujii Hou Z, Nakanishi I, Kinoshita T, Takei Y, Yasue M, Misu R, Suzuki Y, Nakamura S, Kure T, Ohno H, Murata K, Kitaura K, Hirasawa A, Tsujimoto G, Oishi S, Fujii N Z. Hou; I. Nakanishi; T. Kinoshita; Y. Takei; M. Yasue; R. Misu; Y. Suzuki; S. Nakamura; T. Kure; H. Ohno; K. Murata; K. Kitaura; A. Hirasawa; G. Tsujimoto; S. Oishi; N. Fujii Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds. Structure-based design of novel potent protein kinase CK2 (CK2) inhibitors with phenyl-azole scaffolds Journal of Medicinal Chemistry, 55, 6, 2899-2903 Journal of medicinal chemistry, 55, 6, 2899-2903 Journal of Medicinal Chemistry, 55, 6, 2899-2903 2012/03 Refereed English Disclose to all
Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Suzuki Y, Naoe S, Oishi S, Fujii N, Ohno H Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Gold-catalyzed three-component annulation: efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones. Organic letters, 14, 1, 326-329 Organic letters, 14, 1, 326-329 Organic letters, 14, 1, 326-329 2012/01 Refereed Disclose to all
K. Hirano; Y. Inaba; K. Takasu; S. Oishi; Y. Takemoto; N. Fujii; H. Ohno Hirano K, Inaba Y, Takasu K, Oishi S, Takemoto Y, Fujii N, Ohno H K. Hirano; Y. Inaba; K. Takasu; S. Oishi; Y. Takemoto; N. Fujii; H. Ohno Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade. Gold(I)-catalyzed polycyclizations of polyenyne-type anilines based on hydroamination and consecutive hydroarylation cascade Journal of Organic Chemistry, 76, 21, 9068-9080 The Journal of organic chemistry, 76, 21, 9068-9080 Journal of Organic Chemistry, 76, 21, 9068-9080 2011/11 Refereed English Disclose to all
T. Kinoshita; Y. Sekiguchi; H. Fukada; T. Nakaniwa; T. Tada; S. Nakamura; K. Kitaura; H. Ohno; Y. Suzuki; A. Hirasawa; I. Nakanishi; G. Tsujimoto Kinoshita T, Sekiguchi Y, Fukada H, Nakaniwa T, Tada T, Nakamura S, Kitaura K, Ohno H, Suzuki Y, Hirasawa A, Nakanishi I, Tsujimoto G T. Kinoshita; Y. Sekiguchi; H. Fukada; T. Nakaniwa; T. Tada; S. Nakamura; K. Kitaura; H. Ohno; Y. Suzuki; A. Hirasawa; I. Nakanishi; G. Tsujimoto A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase. A detailed thermodynamic profile of cyclopentyl and isopropyl derivatives binding to CK2 kinase Molecular and Cellular Biochemistry, 356, 1-2, 97-105 Molecular and cellular biochemistry, 356, 1-2, 97-105 Molecular and Cellular Biochemistry, 356, 1-2, 97-105 2011/10 Refereed English Disclose to all
Y. Yoshimitsu; S. Oishi; J. Miyagaki; S. Inuki; H. Ohno; N. Fujii Yoshimitsu Y, Oishi S, Miyagaki J, Inuki S, Ohno H, Fujii N Y. Yoshimitsu; S. Oishi; J. Miyagaki; S. Inuki; H. Ohno; N. Fujii Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C. Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase C Bioorganic and Medicinal Chemistry, 19, 18, 5402-5408 Bioorganic & medicinal chemistry, 19, 18, 5402-5408 Bioorganic and Medicinal Chemistry, 19, 18, 5402-5408 2011/09 Refereed English Disclose to all
T. Takeuchi; S. Oishi; T. Watanabe; H. Ohno; J.-I. Sawada; K. Matsuno; A. Asai; N. Asada; K. Kitaura; N. Fujii Takeuchi T, Oishi S, Watanabe T, Ohno H, Sawada J, Matsuno K, Asai A, Asada N, Kitaura K, Fujii N T. Takeuchi; S. Oishi; T. Watanabe; H. Ohno; J.-I. Sawada; K. Matsuno; A. Asai; N. Asada; K. Kitaura; N. Fujii Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors. Structure-activity relationships of carboline and carbazole derivatives as a novel class of ATP-competitive kinesin spindle protein inhibitors Journal of Medicinal Chemistry, 54, 13, 4839-4846 Journal of medicinal chemistry, 54, 13, 4839-4846 Journal of Medicinal Chemistry, 54, 13, 4839-4846 2011/07 Refereed English Disclose to all
A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Iwata A, Inuki S, Oishi S, Fujii N, Ohno H A. Iwata; S. Inuki; S. Oishi; N. Fujii; H. Ohno Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane. Formal total synthesis of (+)-lysergic acid via zinc(II)-mediated regioselective ring-opening reduction of 2-alkynyl-3-indolyloxirane Journal of Organic Chemistry, 76, 13, 5506-5512 The Journal of organic chemistry, 76, 13, 5506-5512 Journal of Organic Chemistry, 76, 13, 5506-5512 2011/07 Refereed English Disclose to all
E. Inokuchi; S. Oishi; T. Kubo; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Inokuchi E, Oishi S, Kubo T, Ohno H, Shimura K, Matsuoka M, Fujii N E. Inokuchi; S. Oishi; T. Kubo; H. Ohno; K. Shimura; M. Matsuoka; N. Fujii Potent CXCR4 antagonists containing amidine type peptide bond isosteres Potent CXCR4 antagonists containing amidine type Peptide bond isosteres. Potent CXCR4 antagonists containing amidine type peptide bond isosteres ACS Medicinal Chemistry Letters, 2, 6, 477-480 ACS medicinal chemistry letters, 2, 6, 477-480 ACS Medicinal Chemistry Letters, 2, 6, 477-480 2011/06 Refereed English Disclose to all
R. Masuda; S. Oishi; H. Ohno; H. Kimura; H. Saji; N. Fujii Masuda R, Oishi S, Ohno H, Kimura H, Saji H, Fujii N R. Masuda; S. Oishi; H. Ohno; H. Kimura; H. Saji; N. Fujii Concise site-specific synthesis of DTPA-peptide conjugates: Application to imaging probes for the chemokine receptor CXCR4 Concise site-specific synthesis of DTPA-peptide conjugates: application to imaging probes for the chemokine receptor CXCR4. Concise site-specific synthesis of DTPA-peptide conjugates: Application to imaging probes for the chemokine receptor CXCR4 Bioorganic and Medicinal Chemistry, 19, 10, 3216-3220 Bioorganic & medicinal chemistry, 19, 10, 3216-3220 Bioorganic and Medicinal Chemistry, 19, 10, 3216-3220 2011/05 Refereed English Disclose to all
E. Inokuchi; A. Yamada; K. Hozumi; K. Tomita; S. Oishi; H. Ohno; M. Nomizu; N. Fujii Inokuchi E, Yamada A, Hozumi K, Tomita K, Oishi S, Ohno H, Nomizu M, Fujii N E. Inokuchi; A. Yamada; K. Hozumi; K. Tomita; S. Oishi; H. Ohno; M. Nomizu; N. Fujii Design and synthesis of amidine-type peptide bond isosteres: Application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis Design and synthesis of amidine-type peptide bond isosteres: application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis. Design and synthesis of amidine-type peptide bond isosteres: Application of nitrile oxide derivatives as active ester equivalents in peptide and peptidomimetics synthesis Organic and Biomolecular Chemistry, 9, 9, 3421-3427 Organic & biomolecular chemistry, 9, 9, 3421-3427 Organic and Biomolecular Chemistry, 9, 9, 3421-3427 2011/05 Refereed English Disclose to all
S. Inuki; A. Iwata; S. Oishi; N. Fujii; H. Ohno Inuki S, Iwata A, Oishi S, Fujii N, Ohno H S. Inuki; A. Iwata; S. Oishi; N. Fujii; H. Ohno Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups. Enantioselective total synthesis of (+)-lysergic acid, (+)-lysergol, and (+)-isolysergol by palladium-catalyzed domino cyclization of allenes bearing amino and bromoindolyl groups Journal of Organic Chemistry, 76, 7, 2072-2083 The Journal of organic chemistry, 76, 7, 2072-2083 Journal of Organic Chemistry, 76, 7, 2072-2083 2011/04 Refereed English Disclose to all
K. Hirano; Y. Inaba; N. Takahashi; M. Shimano; S. Oishi; N. Fujii; H. Ohno Hirano K, Inaba Y, Takahashi N, Shimano M, Oishi S, Fujii N, Ohno H K. Hirano; Y. Inaba; N. Takahashi; M. Shimano; S. Oishi; N. Fujii; H. Ohno Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes. Direct synthesis of fused indoles by gold-catalyzed cascade cyclization of diynes Journal of Organic Chemistry, 76, 5, 1212-1227 The Journal of organic chemistry, 76, 5, 1212-1227 Journal of Organic Chemistry, 76, 5, 1212-1227 2011/03 Refereed English Disclose to all
S. Oishi; R. Misu; K. Tomita; S. Setsuda; R. Masuda; H. Ohno; Y. Naniwa; N. Ieda; N. Inoue; S. Ohkura; Y. Uenoyama; H. Tsukamura; K.-I. Maeda; A. Hirasawa; G. Tsujimoto; N. Fujii Oishi S, Misu R, Tomita K, Setsuda S, Masuda R, Ohno H, Naniwa Y, Ieda N, Inoue N, Ohkura S, Uenoyama Y, Tsukamura H, Maeda K, Hirasawa A, Tsujimoto G, Fujii N S. Oishi; R. Misu; K. Tomita; S. Setsuda; R. Masuda; H. Ohno; Y. Naniwa; N. Ieda; N. Inoue; S. Ohkura; Y. Uenoyama; H. Tsukamura; K.-I. Maeda; A. Hirasawa; G. Tsujimoto; N. Fujii Activation of neuropeptide FF receptors by kisspeptin receptor ligands Activation of Neuropeptide FF Receptors by Kisspeptin Receptor Ligands. Activation of neuropeptide FF receptors by kisspeptin receptor ligands ACS Medicinal Chemistry Letters, 2, 1, 53-57 ACS medicinal chemistry letters, 2, 1, 53-57 ACS Medicinal Chemistry Letters, 2, 1, 53-57 2011/01 Refereed English Disclose to all
Y. Ohta; Y. Tokimizu; S. Oishi; N. Fujii; H. Ohno Ohta Y, Tokimizu Y, Oishi S, Fujii N, Ohno H Y. Ohta; Y. Tokimizu; S. Oishi; N. Fujii; H. Ohno Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines. Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines Organic Letters, 12, 17, 3963-3965 Organic letters, 12, 17, 3963-3965 Organic Letters, 12, 17, 3963-3965 2010/09 Refereed English Disclose to all
A. Okano; K. Tsukamoto; S. Kosaka; H. Maeda; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Okano A, Tsukamoto K, Kosaka S, Maeda H, Oishi S, Tanaka T, Fujii N, Ohno H A. Okano; K. Tsukamoto; S. Kosaka; H. Maeda; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Synthesis of fused and linked bicyclic nitrogen heterocycles by palladiumcatalyzed domino cyclization of propargyl bromides Synthesis of fused and linked bicyclic nitrogen heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Synthesis of fused and linked bicyclic nitrogen heterocycles by palladiumcatalyzed domino cyclization of propargyl bromides Chemistry - A European Journal, 16, 28, 8410-8418 Chemistry (Weinheim an der Bergstrasse, Germany), 16, 28, 8410-8418 Chemistry - A European Journal, 16, 28, 8410-8418 2010/07 Refereed English Disclose to all
S. Oishi; T. Watanabe; J.-I. Sawada; A. Asai; H. Ohno; N. Fujii Oishi S, Watanabe T, Sawada J, Asai A, Ohno H, Fujii N S. Oishi; T. Watanabe; J.-I. Sawada; A. Asai; H. Ohno; N. Fujii Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds. Kinesin spindle protein (KSP) inhibitors with 2,3-fused indole scaffolds Journal of Medicinal Chemistry, 53, 13, 5054-5058 Journal of medicinal chemistry, 53, 13, 5054-5058 Journal of Medicinal Chemistry, 53, 13, 5054-5058 2010/07 Refereed English Disclose to all
S. Inuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H S. Inuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (Jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates. Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (Jaspine B) through palladium-catalyzed bis-cyclization of propargyl chlorides and carbonates Journal of Organic Chemistry, 75, 11, 3831-3842 The Journal of organic chemistry, 75, 11, 3831-3842 Journal of Organic Chemistry, 75, 11, 3831-3842 2010/06 Refereed English Disclose to all
Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Yoshimitsu Y, Inuki S, Oishi S, Fujii N, Ohno H Y. Yoshimitsu; S. Inuki; S. Oishi; N. Fujii; H. Ohno Stereoselective divergent synthesis of four diastereomers of pachastrissamine (Jaspine B) Stereoselective divergent synthesis of four diastereomers of pachastrissamine (jaspine B). Stereoselective divergent synthesis of four diastereomers of pachastrissamine (Jaspine B) Journal of Organic Chemistry, 75, 11, 3843-3846 The Journal of organic chemistry, 75, 11, 3843-3846 Journal of Organic Chemistry, 75, 11, 3843-3846 2010/06 Refereed English Disclose to all
A. Okano; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Okano A, Oishi S, Tanaka T, Fujii N, Ohno H A. Okano; S. Oishi; T. Tanaka; N. Fujii; H. Ohno Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with Isocyanate Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with isocyanate. Construction of linked nitrogen heterocycles by palladium(0)-catalyzed intramolecular domino cyclization of 2-alkynylaziridines bearing a 2-aminoethyl group via ring expansion with Isocyanate Journal of Organic Chemistry, 75, 10, 3396-3400 The Journal of organic chemistry, 75, 10, 3396-3400 Journal of Organic Chemistry, 75, 10, 3396-3400 2010/05 Refereed English Disclose to all
T. Narumi; R. Hayashi; K. Tomita; K. Kobayashi; N. Tanahara; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Narumi T, Hayashi R, Tomita K, Kobayashi K, Tanahara N, Ohno H, Naito T, Kodama E, Matsuoka M, Oishi S, Fujii N T. Narumi; R. Hayashi; K. Tomita; K. Kobayashi; N. Tanahara; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres. Synthesis and biological evaluation of selective CXCR4 antagonists containing alkene dipeptide isosteres Organic and Biomolecular Chemistry, 8, 3, 616-621 Organic & biomolecular chemistry, 8, 3, 616-621 Organic and Biomolecular Chemistry, 8, 3, 616-621 2010/02 Refereed English Disclose to all
T. Mizuhara; S. Oishi; N. Fujii; H. Ohno Mizuhara T, Oishi S, Fujii N, Ohno H T. Mizuhara; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S<sub>N</sub>Ar-type C-S, C-N, or C-O bond formation with heterocumulenes Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S(N)Ar-type C-S, C-N, or C-O bond formation with heterocumulenes. Efficient synthesis of pyrimido[1,2-c] [1,3]benzothiazin-6-imines and related tricyclic heterocycles by S<sub>N</sub>Ar-type C-S, C-N, or C-O bond formation with heterocumulenes Journal of Organic Chemistry, 75, 1, 265-268 The Journal of organic chemistry, 75, 1, 265-268 Journal of Organic Chemistry, 75, 1, 265-268 2010/01 Refereed English Disclose to all
K. Kajiwara; K. Watanabe; R. Tokiwa; T. Kurose; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Kajiwara K, Watanabe K, Tokiwa R, Kurose T, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N K. Kajiwara; K. Watanabe; R. Tokiwa; T. Kurose; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group. Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group Bioorganic and Medicinal Chemistry, 17, 23, 7964-7970 Bioorganic & medicinal chemistry, 17, 23, 7964-7970 Bioorganic and Medicinal Chemistry, 17, 23, 7964-7970 2009/12 Refereed English Disclose to all
M. Tanaka; K. Kajiwara; R. Tokiwa; K. Watanabe; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Tanaka M, Kajiwara K, Tokiwa R, Watanabe K, Ohno H, Tsutsumi H, Hata Y, Izumi K, Kodama E, Matsuoka M, Oishi S, Fujii N M. Tanaka; K. Kajiwara; R. Tokiwa; K. Watanabe; H. Ohno; H. Tsutsumi; Y. Hata; K. Izumi; E. Kodama; M. Matsuoka; S. Oishi; N. Fujii Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins. Bioorganic synthesis of end-capped anti-HIV peptides by simultaneous cyanocysteine-mediated cleavages of recombinant proteins Bioorganic and Medicinal Chemistry, 17, 21, 7487-7492 Bioorganic & medicinal chemistry, 17, 21, 7487-7492 Bioorganic and Medicinal Chemistry, 17, 21, 7487-7492 2009/11 Refereed English Disclose to all
S. Lnuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Inuki S, Yoshimitsu Y, Oishi S, Fujii N, Ohno H S. Lnuki; Y. Yoshimitsu; S. Oishi; N. Fujii; H. Ohno Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes Ring-construction/stereoselective functionalization cascade: total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes. Ring-construction/stereoselective functionalization cascade: Total synthesis of pachastrissamine (jaspine B) through palladium-catalyzed bis-cyclization of bromoallenes Organic Letters, 11, 19, 4478-4481 Organic letters, 11, 19, 4478-4481 Organic Letters, 11, 19, 4478-4481 2009/10 Refereed English Disclose to all
Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization. Construction of nitrogen heterocycles bearing an aminomethyl group by copper-catalyzed domino three-component coupling-cyclization Journal of Organic Chemistry, 74, 18, 7052-7058 The Journal of organic chemistry, 74, 18, 7052-7058 Journal of Organic Chemistry, 74, 18, 7052-7058 2009/09 Refereed English Disclose to all
T. Watabe; Y. Terakawa; K. Watanabe; H. Ohno; H. Nakano; T. Nakatsu; H. Kato; K. Izumi; E. Kodama; M. Matsuoka; K. Kitaura; S. Oishi; N. Fujii Watabe T, Terakawa Y, Watanabe K, Ohno H, Nakano H, Nakatsu T, Kato H, Izumi K, Kodama E, Matsuoka M, Kitaura K, Oishi S, Fujii N T. Watabe; Y. Terakawa; K. Watanabe; H. Ohno; H. Nakano; T. Nakatsu; H. Kato; K. Izumi; E. Kodama; M. Matsuoka; K. Kitaura; S. Oishi; N. Fujii X-ray Crystallographic Study of an HIV-1 Fusion Inhibitor with the gp41 S138A Substitution X-ray crystallographic study of an HIV-1 fusion inhibitor with the gp41 S138A substitution. X-ray Crystallographic Study of an HIV-1 Fusion Inhibitor with the gp41 S138A Substitution Journal of Molecular Biology, 392, 3, 657-665 Journal of molecular biology, 392, 3, 657-665 Journal of Molecular Biology, 392, 3, 657-665 2009/09 Refereed English Disclose to all
Y. Ohta; Y. Kubota; T. Watabe; H. Chiba; S. Oishi; N. Fujii; H. Ohno Ohta Y, Kubota Y, Watabe T, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; Y. Kubota; T. Watabe; H. Chiba; S. Oishi; N. Fujii; H. Ohno Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation. Rapid access to 3-(aminomethyl)isoquinoline-fused polycyclic compounds by copper-catalyzed four-component coupling, cascade cyclization, and oxidation Journal of Organic Chemistry, 74, 16, 6299-6302 The Journal of organic chemistry, 74, 16, 6299-6302 Journal of Organic Chemistry, 74, 16, 6299-6302 2009/08 Refereed English Disclose to all
S. Oishi; H. Kamitani; Y. Kodera; K. Watanabe; K. Kobayashi; T. Narumi; K. Tomita; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Oishi S, Kamitani H, Kodera Y, Watanabe K, Kobayashi K, Narumi T, Tomita K, Ohno H, Naito T, Kodama E, Matsuoka M, Fujii N S. Oishi; H. Kamitani; Y. Kodera; K. Watanabe; K. Kobayashi; T. Narumi; K. Tomita; H. Ohno; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: Synthesis and bioevaluation of α-helical anti-HIV peptide analogues Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: synthesis and bioevaluation of alpha-helical anti-HIV peptide analogues. Peptide bond mimicry by (E)-alkene and (Z)-fluoroalkene peptide isosteres: Synthesis and bioevaluation of α-helical anti-HIV peptide analogues Organic and Biomolecular Chemistry, 7, 14, 2872-2877 Organic & biomolecular chemistry, 7, 14, 2872-2877 Organic and Biomolecular Chemistry, 7, 14, 2872-2877 2009/07 Refereed English Disclose to all
S. Oishi; Y. Kodera; H. Nishikawa; H. Kamitani; T. Watabe; H. Ohno; T. Tochikura; K. Shimane; E. Kodama; M. Matsuoka; F. Mizukoshi; H. Tsujimoto; N. Fujii Oishi S, Kodera Y, Nishikawa H, Kamitani H, Watabe T, Ohno H, Tochikura T, Shimane K, Kodama E, Matsuoka M, Mizukoshi F, Tsujimoto H, Fujii N S. Oishi; Y. Kodera; H. Nishikawa; H. Kamitani; T. Watabe; H. Ohno; T. Tochikura; K. Shimane; E. Kodama; M. Matsuoka; F. Mizukoshi; H. Tsujimoto; N. Fujii Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus. Design and synthesis of membrane fusion inhibitors against the feline immunodeficiency virus Bioorganic and Medicinal Chemistry, 17, 14, 4916-4920 Bioorganic & medicinal chemistry, 17, 14, 4916-4920 Bioorganic and Medicinal Chemistry, 17, 14, 4916-4920 2009/07 Refereed English Disclose to all
T. Watanabe; S. Oishi; N. Fujii; H. Ohno Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: Synthesis and mechanistic study Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: synthesis and mechanistic study. Palladium-catalyzed direct synthesis of carbazoles via one-pot N-arylation and oxidative biaryl coupling: Synthesis and mechanistic study Journal of Organic Chemistry, 74, 13, 4720-4726 The Journal of organic chemistry, 74, 13, 4720-4726 Journal of Organic Chemistry, 74, 13, 4720-4726 2009/07 Refereed English Disclose to all
T. Mizuhara; S. Inuki; S. Oishi; N. Fujii; H. Ohno Mizuhara T, Inuki S, Oishi S, Fujii N, Ohno H T. Mizuhara; S. Inuki; S. Oishi; N. Fujii; H. Ohno Cu(ii)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group Cu(II)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group. Cu(ii)-mediated oxidative intermolecular ortho C-H functionalisation using tetrahydropyrimidine as the directing group Chemical Communications, 23, 3413-3415 Chemical communications (Cambridge, England), 23, 3413-3415 Chemical Communications, 23, 3413-3415 2009/06 Refereed English Disclose to all
K. Kobayashi; T. Narumi; S. Oishi; H. Ohno; N. Fujii Kobayashi K, Narumi T, Oishi S, Ohno H, Fujii N K. Kobayashi; T. Narumi; S. Oishi; H. Ohno; N. Fujii Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper- mediated S<sub>N</sub>2′ alkylation Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper-mediated S(N)2' alkylation. Amino acid-based synthesis of trifluoromethylalkene dipeptide isosteres by alcohol-assisted nucleophilic trifluoromethylation and organozinc-copper- mediated S<sub>N</sub>2′ alkylation Journal of Organic Chemistry, 74, 12, 4626-4629 The Journal of organic chemistry, 74, 12, 4626-4629 Journal of Organic Chemistry, 74, 12, 4626-4629 2009/06 Refereed English Disclose to all
Y. Suzuki; Y. Ohta; S. Oishi; N. Fujii; H. Ohno Suzuki Y, Ohta Y, Oishi S, Fujii N, Ohno H Y. Suzuki; Y. Ohta; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization. Efficient synthesis of aminomethylated pyrroloindoles and dipyrrolopyridines via controlled copper-catalyzed domino multicomponent coupling and bis-cyclization Journal of Organic Chemistry, 74, 11, 4246-4251 The Journal of organic chemistry, 74, 11, 4246-4251 Journal of Organic Chemistry, 74, 11, 4246-4251 2009/06 Refereed English Disclose to all
Y. Ohta; S. Oishi; N. Fujii; H. Ohno Ohta Y, Oishi S, Fujii N, Ohno H Y. Ohta; S. Oishi; N. Fujii; H. Ohno Facile synthesis of 1,2,3,4-tetrahydro-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization Facile synthesis of 1,2,3,4-tetrahydro-beta-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization. Facile synthesis of 1,2,3,4-tetrahydro-carbolines by one-pot domino three-component indole formation and nucleophilic cyclization Organic Letters, 11, 9, 1979-1982 Organic letters, 11, 9, 1979-1982 Organic Letters, 11, 9, 1979-1982 2009/05 Refereed English Disclose to all
T. Nakaniwa; T. Kinoshita; Y. Sekiguchi; T. Tada; I. Nakanishi; K. Kitaura; Y. Suzuki; H. Ohno; A. Hirasawa; G. Tsujimoto Nakaniwa T, Kinoshita T, Sekiguchi Y, Tada T, Nakanishi I, Kitaura K, Suzuki Y, Ohno H, Hirasawa A, Tsujimoto G T. Nakaniwa; T. Kinoshita; Y. Sekiguchi; T. Tada; I. Nakanishi; K. Kitaura; Y. Suzuki; H. Ohno; A. Hirasawa; G. Tsujimoto Structure of human protein kinase CK2α2 with a potent indazole-derivative inhibitor Structure of human protein kinase CK2 alpha 2 with a potent indazole-derivative inhibitor. Structure of human protein kinase CK2α2 with a potent indazole-derivative inhibitor Acta Crystallographica Section F: Structural Biology and Crystallization Communications, 65, 75-79 Acta crystallographica. Section F, Structural biology and crystallization communications, 65, 75-79 Acta Crystallographica Section F: Structural Biology and Crystallization Communications, 65, 75-79 2009/02 Refereed English Disclose to all
K. Tomita; H.A. Popiel; Y. Nagai; T. Toda; Y. Yoshimitsu; H. Ohno; S. Oishi; N. Fujii Tomita K, Popiel HA, Nagai Y, Toda T, Yoshimitsu Y, Ohno H, Oishi S, Fujii N K. Tomita; H.A. Popiel; Y. Nagai; T. Toda; Y. Yoshimitsu; H. Ohno; S. Oishi; N. Fujii Structure-activity relationship study on polyglutamine binding peptide QBP1 Structure-activity relationship study on polyglutamine binding peptide QBP1. Structure-activity relationship study on polyglutamine binding peptide QBP1 Bioorganic and Medicinal Chemistry, 17, 3, 1259-1263 Bioorganic & medicinal chemistry, 17, 3, 1259-1263 Bioorganic and Medicinal Chemistry, 17, 3, 1259-1263 2009/02 Refereed English Disclose to all
S. Oishi; S. Ito; H. Nishikawa; M. Tanaka; H. Ohno; A. Otaka; K. Izumi; E. Kodama; M. Matsuoka; N. Fujii Oishi S, Ito S, Nishikawa H, Tanaka M, Ohno H, Otaka A, Izumi K, Kodama E, Matsuoka M, Fujii N S. Oishi; S. Ito; H. Nishikawa; M. Tanaka; H. Ohno; A. Otaka; K. Izumi; E. Kodama; M. Matsuoka; N. Fujii Development of a novel fusion inhibitor against T-20-resistant HIV-1. Development of a novel fusion inhibitor against T-20-resistant HIV-1. Development of a novel fusion inhibitor against T-20-resistant HIV-1. Advances in experimental medicine and biology, 611, 389-391 Advances in experimental medicine and biology, 611, 389-391 Advances in experimental medicine and biology, 611, 389-391 2009 Refereed English Disclose to all
K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Synthesis and application of (Z)-alkene- and (E)-fluoroalkene-dipeptide isosteres as cis-amide equivalents. Advances in experimental medicine and biology, 611, 365-366 Advances in experimental medicine and biology, 611, 365-366 Advances in experimental medicine and biology, 611, 365-366 2009 Refereed English Disclose to all
K. Tomita; S. Oishi; H. Ohno; S.C. Peiper; N. Fujii Tomita K, Oishi S, Ohno H, Peiper SC, Fujii N K. Tomita; S. Oishi; H. Ohno; S.C. Peiper; N. Fujii Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase. Development of novel G-protein-coupled receptor 54 agonists with resistance to degradation by matrix metalloproteinase Journal of Medicinal Chemistry, 51, 23, 7645-7649 Journal of medicinal chemistry, 51, 23, 7645-7649 Journal of Medicinal Chemistry, 51, 23, 7645-7649 2008/12 Refereed English Disclose to all
S. Inuki; S. Oishi; N. Fujii; H. Ohno Inuki S, Oishi S, Fujii N, Ohno H S. Inuki; S. Oishi; N. Fujii; H. Ohno Total synthesis of (±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group Total synthesis of (+/-)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group. Total synthesis of (±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group Organic Letters, 10, 22, 5239-5242 Organic letters, 10, 22, 5239-5242 Organic Letters, 10, 22, 5239-5242 2008/11 Refereed English Disclose to all
H. Nishikawa; S. Oishi; M. Fujita; K. Watanabe; R. Tokiwa; H. Ohno; E. Kodama; K. Izumi; K. Kajiwara; T. Naitoh; M. Matsuoka; A. Otaka; N. Fujii Nishikawa H, Oishi S, Fujita M, Watanabe K, Tokiwa R, Ohno H, Kodama E, Izumi K, Kajiwara K, Naitoh T, Matsuoka M, Otaka A, Fujii N H. Nishikawa; S. Oishi; M. Fujita; K. Watanabe; R. Tokiwa; H. Ohno; E. Kodama; K. Izumi; K. Kajiwara; T. Naitoh; M. Matsuoka; A. Otaka; N. Fujii Identification of minimal sequence for HIV-1 fusion inhibitors Identification of minimal sequence for HIV-1 fusion inhibitors. Identification of minimal sequence for HIV-1 fusion inhibitors Bioorganic and Medicinal Chemistry, 16, 20, 9184-9187 Bioorganic & medicinal chemistry, 16, 20, 9184-9187 Bioorganic and Medicinal Chemistry, 16, 20, 9184-9187 2008/10 Refereed English Disclose to all
Y. Suzuki; J. Cluzeau; T. Hara; A. Hirasawa; G. Tsujimoto; S. Oishi; H. Ohno; N. Fujii Suzuki Y, Cluzeau J, Hara T, Hirasawa A, Tsujimoto G, Oishi S, Ohno H, Fujii N Y. Suzuki; J. Cluzeau; T. Hara; A. Hirasawa; G. Tsujimoto; S. Oishi; H. Ohno; N. Fujii Structure-activity relationships of pyrazine-based CK2 inhibitors: Synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines Structure-activity relationships of pyrazine-based CK2 inhibitors: synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines. Structure-activity relationships of pyrazine-based CK2 inhibitors: Synthesis and evaluation of 2,6-disubstituted pyrazines and 4,6-disubstituted pyrimidines Archiv der Pharmazie, 341, 9, 554-561 Archiv der Pharmazie, 341, 9, 554-561 Archiv der Pharmazie, 341, 9, 554-561 2008/09 Refereed English Disclose to all
H. Iwasaki; T. Eguchi; N. Tsutsui; H. Ohno; T. Tanaka Iwasaki H, Eguchi T, Tsutsui N, Ohno H, Tanaka T H. Iwasaki; T. Eguchi; N. Tsutsui; H. Ohno; T. Tanaka Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring. Samarium(II)-mediated spirocyclization by intramolecular aryl radical addition onto an aromatic ring Journal of Organic Chemistry, 73, 18, 7145-7152 The Journal of organic chemistry, 73, 18, 7145-7152 Journal of Organic Chemistry, 73, 18, 7145-7152 2008/09 Refereed English Disclose to all
A. Okano; T. Mizutani; S. Oishi; T. Tanaka; H. Ohno; N. Fujii Okano A, Mizutani T, Oishi S, Tanaka T, Ohno H, Fujii N A. Okano; T. Mizutani; S. Oishi; T. Tanaka; H. Ohno; N. Fujii Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade. Palladium-catalysed biscyclisation of allenic bromoalkenes through a zipper-mode cascade Chemical Communications, 30, 3534-3536 Chemical communications (Cambridge, England), 30, 3534-3536 Chemical Communications, 30, 3534-3536 2008/08 Refereed English Disclose to all
Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Ohta Y, Chiba H, Oishi S, Fujii N, Ohno H Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Concise synthesis of indole-fused 1,4-diazepines through copper(l)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation Concise synthesis of indole-fused 1,4-diazepines through copper(I)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation. Concise synthesis of indole-fused 1,4-diazepines through copper(l)-catalyzed domino three-component coupling-cyclization-N-arylation under microwave irradiation Organic Letters, 10, 16, 3535-3538 Organic letters, 10, 16, 3535-3538 Organic Letters, 10, 16, 3535-3538 2008/08 Refereed English Disclose to all
S. Ueda; M. Kato; S. Inuki; H. Ohno; B. Evans; Z.-x. Wang; S.C. Peiper; K. Izumi; E. Kodama; M. Matsuoka; H. Nagasawa; S. Oishi; N. Fujii Ueda S, Kato M, Inuki S, Ohno H, Evans B, Wang ZX, Peiper SC, Izumi K, Kodama E, Matsuoka M, Nagasawa H, Oishi S, Fujii N S. Ueda; M. Kato; S. Inuki; H. Ohno; B. Evans; Z.-x. Wang; S.C. Peiper; K. Izumi; E. Kodama; M. Matsuoka; H. Nagasawa; S. Oishi; N. Fujii Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach. Identification of novel non-peptide CXCR4 antagonists by ligand-based design approach Bioorganic and Medicinal Chemistry Letters, 18, 14, 4124-4129 Bioorganic & medicinal chemistry letters, 18, 14, 4124-4129 Bioorganic and Medicinal Chemistry Letters, 18, 14, 4124-4129 2008/07 Refereed English Disclose to all
E. Inokuchi; T. Narumi; A. Niida; K. Kobayashi; K. Tomita; S. Oishi; H. Ohno; N. Fujii Inokuchi E, Narumi T, Niida A, Kobayashi K, Tomita K, Oishi S, Ohno H, Fujii N E. Inokuchi; T. Narumi; A. Niida; K. Kobayashi; K. Tomita; S. Oishi; H. Ohno; N. Fujii Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates. Efficient synthesis of trifluoromethyl and related trisubstituted alkene dipeptide isosteres by palladium-catalyzed carbonylation of amino acid derived allylic carbonates Journal of Organic Chemistry, 73, 10, 3942-3945 The Journal of organic chemistry, 73, 10, 3942-3945 Journal of Organic Chemistry, 73, 10, 3942-3945 2008/05 Refereed English Disclose to all
S. Oishi; R. Masuda; B. Evans; S. Ueda; Y. Goto; H. Ohno; A. Hirasawa; G. Tsujimoto; Z. Wang; S.C. Peiper; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Oishi S, Masuda R, Evans B, Ueda S, Goto Y, Ohno H, Hirasawa A, Tsujimoto G, Wang Z, Peiper SC, Naito T, Kodama E, Matsuoka M, Fujii N S. Oishi; R. Masuda; B. Evans; S. Ueda; Y. Goto; H. Ohno; A. Hirasawa; G. Tsujimoto; Z. Wang; S.C. Peiper; T. Naito; E. Kodama; M. Matsuoka; N. Fujii Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4 Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4. Synthesis and application of fluorescein- and biotin-labeled molecular probes for the chemokine receptor CXCR4 ChemBioChem, 9, 7, 1154-1158 Chembiochem : a European journal of chemical biology, 9, 7, 1154-1158 ChemBioChem, 9, 7, 1154-1158 2008/05 Refereed English Disclose to all
T. Watanabe; S. Oishi; N. Fujii; H. Ohno Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Palladium-catalyzed sp<sup>3</sup> C-H activation of simple alkyl groups: Direct preparation of indoline derivatives from N-alkyl-2-bromoanilines Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines. Palladium-catalyzed sp<sup>3</sup> C-H activation of simple alkyl groups: Direct preparation of indoline derivatives from N-alkyl-2-bromoanilines Organic Letters, 10, 9, 1759-1762 Organic letters, 10, 9, 1759-1762 Organic Letters, 10, 9, 1759-1762 2008/05 Refereed English Disclose to all
H. Ohno; A. Okano; S. Kosaka; K. Tsukamoto; M. Ohata; K. Ishihara; H. Maeda; T. Tanaka; N. Fujii Ohno H, Okano A, Kosaka S, Tsukamoto K, Ohata M, Ishihara K, Maeda H, Tanaka T, Fujii N H. Ohno; A. Okano; S. Kosaka; K. Tsukamoto; M. Ohata; K. Ishihara; H. Maeda; T. Tanaka; N. Fujii Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides. Direct construction of bicyclic heterocycles by palladium-catalyzed domino cyclization of propargyl bromides Organic Letters, 10, 6, 1171-1174 Organic letters, 10, 6, 1171-1174 Organic Letters, 10, 6, 1171-1174 2008/03 Refereed English Disclose to all
Y. Ohta; S. Oishi; N. Fujii; H. Ohno Ohta Y, Oishi S, Fujii N, Ohno H Y. Ohta; S. Oishi; N. Fujii; H. Ohno Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation. Facile synthesis of 3-(aminomethyl)isoquinolines by copper-catalysed domino four-component coupling and cyclisation Chemical Communications, 7, 835-837 Chemical communications (Cambridge, England), 7, 835-837 Chemical Communications, 7, 835-837 2008/02 Refereed English Disclose to all
S. Oishi; S. Ito; H. Nishikawa; K. Watanabe; M. Tanaka; H. Ohno; K. Izumi; Y. Sakagami; E. Kodama; M. Matsuoka; N. Fujii Oishi S, Ito S, Nishikawa H, Watanabe K, Tanaka M, Ohno H, Izumi K, Sakagami Y, Kodama E, Matsuoka M, Fujii N S. Oishi; S. Ito; H. Nishikawa; K. Watanabe; M. Tanaka; H. Ohno; K. Izumi; Y. Sakagami; E. Kodama; M. Matsuoka; N. Fujii Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity. Design of a novel HIV-1 fusion inhibitor that displays a minimal interface for binding affinity Journal of Medicinal Chemistry, 51, 3, 388-391 Journal of medicinal chemistry, 51, 3, 388-391 Journal of Medicinal Chemistry, 51, 3, 388-391 2008/02 Refereed English Disclose to all
S. Oishi; T. Narumi; H. Ohno; A. Otaka; N. Fujii S. Oishi; T. Narumi; H. Ohno; A. Otaka; N. Fujii Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides Synthesis of highly functionalized alkene dipeptide isosteres and its application to the structure-activity relationship study on bioactive peptides Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry, 66, 9, 846-857 Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry, 66, 9, 846-857 , 66, 9, 846-857 2008 Refereed Japanese Disclose to all
K. Tomita; S. Oishi; H. Ohno; N. Fujii Tomita K, Oishi S, Ohno H, Fujii N K. Tomita; S. Oishi; H. Ohno; N. Fujii Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists. Structure-activity relationship study and NMR analysis of fluorobenzoyl pentapeptide GPR54 agonists Biopolymers - Peptide Science Section, 90, 4, 503-511 Biopolymers, 90, 4, 503-511 Biopolymers - Peptide Science Section, 90, 4, 503-511 2008 Refereed English Disclose to all
T. Watanabe; S. Ueda; S. Inuki; S. Oishi; N. Fujii; H. Ohno Watanabe T, Ueda S, Inuki S, Oishi S, Fujii N, Ohno H T. Watanabe; S. Ueda; S. Inuki; S. Oishi; N. Fujii; H. Ohno One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling. One-pot synthesis of carbazoles by palladium-catalyzed N-arylation and oxidative coupling Chemical Communications, 43, 4516-4518 Chemical communications (Cambridge, England), 43, 4516-4518 Chemical Communications, 43, 4516-4518 2007/11 Refereed English Disclose to all
T. Watanabe; S. Oishi; N. Fujii; H. Ohno Watanabe T, Oishi S, Fujii N, Ohno H T. Watanabe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed hydroarylation of allenes: A highly regioselective carbon-carbon bond formation producing six-membered rings Gold-catalyzed hydroarylation of allenes: a highly regioselective carbon-carbon bond formation producing six-membered rings. Gold-catalyzed hydroarylation of allenes: A highly regioselective carbon-carbon bond formation producing six-membered rings Organic Letters, 9, 23, 4821-4824 Organic letters, 9, 23, 4821-4824 Organic Letters, 9, 23, 4821-4824 2007/11 Refereed English Disclose to all
H. Ohno; M. Iuchi; N. Fujii; T. Tanaka Ohno H, Iuchi M, Fujii N, Tanaka T H. Ohno; M. Iuchi; N. Fujii; T. Tanaka Zipper-mode double C-H activation: Palladium-catalyzed direct construction of highly-fused heterocyclic systems Zipper-mode double C-H activation: palladium-catalyzed direct construction of highly-fused heterocyclic systems. Zipper-mode double C-H activation: Palladium-catalyzed direct construction of highly-fused heterocyclic systems Organic Letters, 9, 23, 4813-4815 Organic letters, 9, 23, 4813-4815 Organic Letters, 9, 23, 4813-4815 2007/11 Refereed English Disclose to all
T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii Narumi T, Tomita K, Inokuchi E, Kobayashi K, Oishi S, Ohno H, Fujii N T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides. Facile synthesis of fluoroalkenes by palladium-catalyzed reductive defluorination of allylic gem-difluorides Organic Letters, 9, 17, 3465-3468 Organic letters, 9, 17, 3465-3468 Organic Letters, 9, 17, 3465-3468 2007/08 Refereed English Disclose to all
K. Tomita; S. Oishi; J. Cluzeau; H. Ohno; J.-M. Navenot; Z.-X. Wang; S.C. Peiper; M. Akamatsu; N. Fujii Tomita K, Oishi S, Cluzeau J, Ohno H, Navenot JM, Wang ZX, Peiper SC, Akamatsu M, Fujii N K. Tomita; S. Oishi; J. Cluzeau; H. Ohno; J.-M. Navenot; Z.-X. Wang; S.C. Peiper; M. Akamatsu; N. Fujii SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54 SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54. SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54 Journal of Medicinal Chemistry, 50, 14, 3222-3228 Journal of medicinal chemistry, 50, 14, 3222-3228 Journal of Medicinal Chemistry, 50, 14, 3222-3228 2007/07 Refereed English Disclose to all
J. Cluzeau; S. Oishi; H. Ohno; Z. Wang; B. Evans; S.C. Peiper; N. Fujii Cluzeau J, Oishi S, Ohno H, Wang Z, Evans B, Peiper SC, Fujii N J. Cluzeau; S. Oishi; H. Ohno; Z. Wang; B. Evans; S.C. Peiper; N. Fujii Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists. Design and synthesis of all diastereomers of cyclic pseudo-dipeptides as mimics of cyclic CXCR4 pentapeptide antagonists Organic and Biomolecular Chemistry, 5, 12, 1915-1923 Organic & biomolecular chemistry, 5, 12, 1915-1923 Organic and Biomolecular Chemistry, 5, 12, 1915-1923 2007/06 Refereed English Disclose to all
H. Ohno; T. Mizutani; Y. Kadoh; A. Aso; K. Miyamura; N. Fujii; T. Tanaka Ohno H, Mizutani T, Kadoh Y, Aso A, Miyamura K, Fujii N, Tanaka T H. Ohno; T. Mizutani; Y. Kadoh; A. Aso; K. Miyamura; N. Fujii; T. Tanaka A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes. A highly regio- and stereoselective formation of bicyclo[4.2.0]oct-5-ene derivatives through thermal intramolecular [2 + 2] cycloaddition of allenes Journal of Organic Chemistry, 72, 12, 4378-4389 The Journal of organic chemistry, 72, 12, 4378-4389 Journal of Organic Chemistry, 72, 12, 4378-4389 2007/06 Refereed English Disclose to all
S. Ueda; S. Oishi; Z.-X. Wang; T. Araki; H. Tamamura; J. Cluzeau; H. Ohno; S. Kusano; H. Nakashima; J.O. Trent; S.C. Peiper; N. Fujii Ueda S, Oishi S, Wang ZX, Araki T, Tamamura H, Cluzeau J, Ohno H, Kusano S, Nakashima H, Trent JO, Peiper SC, Fujii N S. Ueda; S. Oishi; Z.-X. Wang; T. Araki; H. Tamamura; J. Cluzeau; H. Ohno; S. Kusano; H. Nakashima; J.O. Trent; S.C. Peiper; N. Fujii Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: Disclosing the importance of side-chain and backbone functionalities Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: disclosing the importance of side-chain and backbone functionalities. Structure-activity relationships of cyclic peptide-based chemokine receptor CXCR4 antagonists: Disclosing the importance of side-chain and backbone functionalities Journal of Medicinal Chemistry, 50, 2, 192-198 Journal of medicinal chemistry, 50, 2, 192-198 Journal of Medicinal Chemistry, 50, 2, 192-198 2007/01 Refereed English Disclose to all
H. Ohno; A. Aso; Y. Kadoh; N. Fujii; T. Tanaka Ohno H, Aso A, Kadoh Y, Fujii N, Tanaka T H. Ohno; A. Aso; Y. Kadoh; N. Fujii; T. Tanaka Heck-type cyclization of oxime ethers: Stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes Heck-type cyclization of oxime ethers: stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes. Heck-type cyclization of oxime ethers: Stereoselective carbon-carbon bond formation with aryl halides to produce heterocyclic oximes Angewandte Chemie - International Edition, 46, 33, 6325-6328 Angewandte Chemie (International ed. in English), 46, 33, 6325-6328 Angewandte Chemie - International Edition, 46, 33, 6325-6328 2007 Refereed English Disclose to all
H. Ohno; Y. Ohta; S. Oishi; N. Fujii Ohno H, Ohta Y, Oishi S, Fujii N H. Ohno; Y. Ohta; S. Oishi; N. Fujii Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions. Direct synthesis of 2-(aminomethyl)indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions Angewandte Chemie - International Edition, 46, 13, 2295-2298 Angewandte Chemie (International ed. in English), 46, 13, 2295-2298 Angewandte Chemie - International Edition, 46, 13, 2295-2298 2007 Refereed English Disclose to all
K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Tomita K, Narumi T, Niida A, Oishi S, Ohno H, Fujii N K. Tomita; T. Narumi; A. Niida; S. Oishi; H. Ohno; N. Fujii Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres. Fmoc-based solid-phase synthesis of GPR54-agonistic pentapeptide derivatives containing alkene- and fluoroalkene-dipeptide isosteres Biopolymers - Peptide Science Section, 88, 2, 272-278 Biopolymers, 88, 2, 272-278 Biopolymers - Peptide Science Section, 88, 2, 272-278 2007 Refereed English Disclose to all
H. Hamaguchi; S. Kosaka; H. Ohno; N. Fujii; T. Tanaka Hamaguchi H, Kosaka S, Ohno H, Fujii N, Tanaka T H. Hamaguchi; S. Kosaka; H. Ohno; N. Fujii; T. Tanaka Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): Direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the presence or absence of palladium(0): Direct construction of bicyclic sulfamides containing five- to eight-membered rings by tandem cyclization of bromoallenes Chemistry - A European Journal, 13, 6, 1692-1708 Chemistry (Weinheim an der Bergstrasse, Germany), 13, 6, 1692-1708 Chemistry - A European Journal, 13, 6, 1692-1708 2007 Refereed English Disclose to all
T. Narumi; A. Niida; K. Tomita; S. Oishi; A. Otaka; H. Ohno; N. Fujii Narumi T, Niida A, Tomita K, Oishi S, Otaka A, Ohno H, Fujii N T. Narumi; A. Niida; K. Tomita; S. Oishi; A. Otaka; H. Ohno; N. Fujii A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres. A novel one-pot reaction involving organocopper-mediated reduction/transmetalation/asymmetric alkylation, leading to the diastereoselective synthesis of functionalized (Z)-fluoroalkene dipeptide isosteres Chemical Communications, 45, 4720-4722 Chemical communications (Cambridge, England), 45, 4720-4722 Chemical Communications, 45, 4720-4722 2006/12 Refereed English Disclose to all
K. Tomita; A. Niida; S. Oishi; H. Ohno; J. Cluzeau; J.-M. Navenot; Z.-x. Wang; S.C. Peiper; N. Fujii Tomita K, Niida A, Oishi S, Ohno H, Cluzeau J, Navenot JM, Wang ZX, Peiper SC, Fujii N K. Tomita; A. Niida; S. Oishi; H. Ohno; J. Cluzeau; J.-M. Navenot; Z.-x. Wang; S.C. Peiper; N. Fujii Structure-activity relationship study on small peptidic GPR54 agonists Structure-activity relationship study on small peptidic GPR54 agonists. Structure-activity relationship study on small peptidic GPR54 agonists Bioorganic and Medicinal Chemistry, 14, 22, 7595-7603 Bioorganic & medicinal chemistry, 14, 22, 7595-7603 Bioorganic and Medicinal Chemistry, 14, 22, 7595-7603 2006/11 Refereed English Disclose to all
T. Tanaka; S. Yamamoto; K. Hiramatsu; K. Murakami; H. Yoshino; D. Patra; C. Iwata; H. Ohno Tanaka T, Yamamoto S, Hiramatsu K, Murakami K, Yoshino H, Patra D, Iwata C, Ohno H T. Tanaka; S. Yamamoto; K. Hiramatsu; K. Murakami; H. Yoshino; D. Patra; C. Iwata; H. Ohno Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system. Construction of tricyclic enone, a common precursor for aphidicolane and stemodane B/C/D-ring system Chemical and Pharmaceutical Bulletin, 54, 8, 1138-1143 Chemical & pharmaceutical bulletin, 54, 8, 1138-1143 Chemical and Pharmaceutical Bulletin, 54, 8, 1138-1143 2006/08 Refereed English Disclose to all
A. Niida; M. Mizumoto; T. Narumi; E. Inokuchi; S. Oishi; H. Ohno; A. Otaka; K. Kitaura; N. Fujii Niida A, Mizumoto M, Narumi T, Inokuchi E, Oishi S, Ohno H, Otaka A, Kitaura K, Fujii N A. Niida; M. Mizumoto; T. Narumi; E. Inokuchi; S. Oishi; H. Ohno; A. Otaka; K. Kitaura; N. Fujii Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations. Synthesis of (Z)-alkene and (E)-fluoroalkene-containing diketopiperazine mimetics utilizing organocopper-mediated reduction-alkylation and diastereoselectivity examination using DFT calculations Journal of Organic Chemistry, 71, 11, 4118-4129 The Journal of organic chemistry, 71, 11, 4118-4129 Journal of Organic Chemistry, 71, 11, 4118-4129 2006/05 Refereed English Disclose to all
A. Niida; H. Tanigaki; E. Inokuchi; Y. Sasaki; S. Oishi; H. Ohno; H. Tamamura; Z. Wang; S.C. Peiper; K. Kitaura; A. Otaka; N. Fujii Niida A, Tanigaki H, Inokuchi E, Sasaki Y, Oishi S, Ohno H, Tamamura H, Wang Z, Peiper SC, Kitaura K, Otaka A, Fujii N A. Niida; H. Tanigaki; E. Inokuchi; Y. Sasaki; S. Oishi; H. Ohno; H. Tamamura; Z. Wang; S.C. Peiper; K. Kitaura; A. Otaka; N. Fujii Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-S <sub>N</sub>2′ reactions and their use in the preparation of low-molecule CXCR4 antagonists Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-SN2' reactions and their use in the preparation of low-molecule CXCR4 antagonists. Stereoselective synthesis of 3,6-disubstituted-3,6-dihydropyridin-2-ones as potential diketopiperazine mimetics using organocopper-mediated anti-S <sub>N</sub>2′ reactions and their use in the preparation of low-molecule CXCR4 antagonists Journal of Organic Chemistry, 71, 10, 3942-3951 The Journal of organic chemistry, 71, 10, 3942-3951 Journal of Organic Chemistry, 71, 10, 3942-3951 2006/05 Refereed English Disclose to all
H. Ohno; Y. Kadoh; N. Fujii; T. Tanaka Ohno H, Kadoh Y, Fujii N, Tanaka T H. Ohno; Y. Kadoh; N. Fujii; T. Tanaka Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals. Potassium carbonate-promoted stereospecific 5-endo-trig cyclization of unactivated allenes in the absence of any transition metals Organic Letters, 8, 5, 947-950 Organic letters, 8, 5, 947-950 Organic Letters, 8, 5, 947-950 2006/03 Refereed English Disclose to all
Ohno H H. Ohno Ohno H Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations. Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations Development of useful reactions based on the novel reactivities of allenic compounds and their application to tandem cyclizations. Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 125, 12, 899-925 Yakugaku Zasshi, 125, 12, 899-925 Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 125, 12, 899-925 2005/12 Refereed Japanese Disclose to all
H. Ohno Ohno H H. Ohno Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds. Development of useful reactions involving tandem cyclizations based on the novel reactivities of allenic compounds Chemical and Pharmaceutical Bulletin, 53, 10, 1211-1226 Chemical & pharmaceutical bulletin, 53, 10, 1211-1226 Chemical and Pharmaceutical Bulletin, 53, 10, 1211-1226 2005/10 Refereed English Disclose to all
H. Ohno; T. Mizutani; Y. Kadoh; K. Miyamura; T. Tanaka Ohno H, Mizutani T, Kadoh Y, Miyamura K, Tanaka T H. Ohno; T. Mizutani; Y. Kadoh; K. Miyamura; T. Tanaka Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: Diastereoselective access to bicyclic nitrogen heterocycles Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: diastereoselective access to bicyclic nitrogen heterocycles. Thermal intramolecular [2+2] cycloaddition of allenenes and allenynes: Diastereoselective access to bicyclic nitrogen heterocycles Angewandte Chemie - International Edition, 44, 32, 5113-5115 Angewandte Chemie (International ed. in English), 44, 32, 5113-5115 Angewandte Chemie - International Edition, 44, 32, 5113-5115 2005/08 Refereed English Disclose to all
H. Ohno; M. Yamamoto; M. Iuchi; T. Tanaka Ohno H, Yamamoto M, Iuchi M, Tanaka T H. Ohno; M. Yamamoto; M. Iuchi; T. Tanaka Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization. Palladium-catalyzed tandem cyclization of bromoenynes through aromatic C-H bond functionalization Angewandte Chemie - International Edition, 44, 32, 5103-5106 Angewandte Chemie (International ed. in English), 44, 32, 5103-5106 Angewandte Chemie - International Edition, 44, 32, 5103-5106 2005/08 Refereed English Disclose to all
H. Ohno; K. Miyamura; T. Mizutani; Y. Kadoh; Y. Takeoka; H. Hamaguchi; T. Tanaka Ohno H, Miyamura K, Mizutani T, Kadoh Y, Takeoka Y, Hamaguchi H, Tanaka T H. Ohno; K. Miyamura; T. Mizutani; Y. Kadoh; Y. Takeoka; H. Hamaguchi; T. Tanaka Palladium(0)-catalyzed tandem cyclization of alleneues: Direct construction of tricyclic heterocycles through aromatic C-H activation Palladium(0)-catalyzed tandem cyclization of allenenes: direct construction of tricyclic heterocycles through aromatic C--H activation. Palladium(0)-catalyzed tandem cyclization of alleneues: Direct construction of tricyclic heterocycles through aromatic C-H activation Chemistry - A European Journal, 11, 12, 3728-3741 Chemistry (Weinheim an der Bergstrasse, Germany), 11, 12, 3728-3741 Chemistry - A European Journal, 11, 12, 3728-3741 2005/06 Refereed English Disclose to all
H. Hamaguchi; S. Kosaka; H. Ohno; T. Tanaka Hamaguchi H, Kosaka S, Ohno H, Tanaka T H. Hamaguchi; S. Kosaka; H. Ohno; T. Tanaka Bromoallenes as allyl dication equivalents in the absence of palladium(0): Synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes Bromoallenes as allyl dication equivalents in the absence of palladium(0): synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes. Bromoallenes as allyl dication equivalents in the absence of palladium(0): Synthesis of bicyclic sulfamides by tandem cyclization of bromoallenes Angewandte Chemie - International Edition, 44, 10, 1513-1517 Angewandte Chemie (International ed. in English), 44, 10, 1513-1517 Angewandte Chemie - International Edition, 44, 10, 1513-1517 2005/02 Refereed English Disclose to all
H. Ohno; H. Iwasaki; T. Eguchi; T. Tanaka Ohno H, Iwasaki H, Eguchi T, Tanaka T H. Ohno; H. Iwasaki; T. Eguchi; T. Tanaka The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring. The first samarium(II)-mediated aryl radical cyclisation onto an aromatic ring Chemical Communications, 19, 2228-2229 Chemical communications (Cambridge, England), 19, 2228-2229 Chemical Communications, 19, 2228-2229 2004/10 Refereed English Disclose to all
K. Hayashi; S.M.A. Rahman; H. Ohno; T. Tanaka; N. Toyooka; H. Nemoto; T. Hayashi Hayashi K, Rahman SM, Ohno H, Tanaka T, Toyooka N, Nemoto H, Hayashi T K. Hayashi; S.M.A. Rahman; H. Ohno; T. Tanaka; N. Toyooka; H. Nemoto; T. Hayashi Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against Herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells. Evaluation of scopadulciol-related molecules for their stimulatory effect on the cytotoxicity of acyclovir and ganciclovir against herpes simplex virus type 1 thymidine kinase gene-transfected HeLa cells Chemical and Pharmaceutical Bulletin, 52, 8, 1015-1017 Chemical & pharmaceutical bulletin, 52, 8, 1015-1017 Chemical and Pharmaceutical Bulletin, 52, 8, 1015-1017 2004/08 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka Ohno H, Hamaguchi H, Ohata M, Kosaka S, Tanaka T H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent. Palladium(0)-catalyzed synthesis of medium-sized heterocycles by using bromoallenes as an allyl dication equivalent Journal of the American Chemical Society, 126, 28, 8744-8754 Journal of the American Chemical Society, 126, 28, 8744-8754 Journal of the American Chemical Society, 126, 28, 8744-8754 2004/07 Refereed English Disclose to all
H. Ohno; Y. Takeoka; Y. Kadoh; K. Miyamura; T. Tanaka Ohno H, Takeoka Y, Kadoh Y, Miyamura K, Tanaka T H. Ohno; Y. Takeoka; Y. Kadoh; K. Miyamura; T. Tanaka Palladium(0)-catalyzed stereoselective cyclization of allenenes: Divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes Palladium(0)-catalyzed stereoselective cyclization of allenenes: divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes. Palladium(0)-catalyzed stereoselective cyclization of allenenes: Divergent synthesis of pyrrolidines and 3-azabicyclo[3.1.0]hexanes from single allenenes Journal of Organic Chemistry, 69, 13, 4541-4544 The Journal of organic chemistry, 69, 13, 4541-4544 Journal of Organic Chemistry, 69, 13, 4541-4544 2004/06 Refereed English Disclose to all
H. Ohno; Y. Takemoto; N. Fujii; T. Tanaka; T. Ibukab Ohno H, Takemoto Y, Fujii N, Tanaka T, Ibuka T H. Ohno; Y. Takemoto; N. Fujii; T. Tanaka; T. Ibukab Stereodivergent synthesis of chiral 2-alkenylaziridines: Palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination Stereodivergent synthesis of chiral 2-alkenylaziridines: palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination. Stereodivergent synthesis of chiral 2-alkenylaziridines: Palladium(0)-catalyzed 2,3-cis-selective aziridination and base-mediated 2,3-trans-selective aziridination Chemical and Pharmaceutical Bulletin, 52, 1, 111-119 Chemical & pharmaceutical bulletin, 52, 1, 111-119 Chemical and Pharmaceutical Bulletin, 52, 1, 111-119 2004/01 Refereed English Disclose to all
H. Ohno; Y. Takeoka; K. Miyamura; Y. Kadoh; T. Tanaka Ohno H, Takeoka Y, Miyamura K, Kadoh Y, Tanaka T H. Ohno; Y. Takeoka; K. Miyamura; Y. Kadoh; T. Tanaka Novel Synthesis of 3-Azabicyclo[3.1.0]hexanes by Unusual Palladium(0)-Catalyzed Cyclopropanation of Allenenes Novel synthesis of 3-azabicyclo[3.1.0]hexanes by unusual palladium(0)-catalyzed cyclopropanation of allenenes. Novel Synthesis of 3-Azabicyclo[3.1.0]hexanes by Unusual Palladium(0)-Catalyzed Cyclopropanation of Allenenes Organic Letters, 5, 25, 4763-4766 Organic letters, 5, 25, 4763-4766 Organic Letters, 5, 25, 4763-4766 2003/12 Refereed English Disclose to all
H. Ohno; K. Miyamura; T. Tanaka; S. Oishi; A. Toda; Y. Takemoto; N. Fujii; T. Ibuka Ohno H, Miyamura K, Tanaka T, Oishi S, Toda A, Takemoto Y, Fujii N, Ibuka T H. Ohno; K. Miyamura; T. Tanaka; S. Oishi; A. Toda; Y. Takemoto; N. Fujii; T. Ibuka Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system. Synthesis of allenes from allylic alcohol derivatives bearing a bromine atom using a palladium(0)/diethylzinc system Journal of Organic Chemistry, 67, 4, 1359-1367 The Journal of organic chemistry, 67, 4, 1359-1367 Journal of Organic Chemistry, 67, 4, 1359-1367 2002/02 Refereed English Disclose to all
H. Ohno H. Ohno Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst Development of aziridination and azetizination reactions of amino allenes using a palladium catalyst Yakugaku Zasshi, 121, 10, 733-741 Yakugaku Zasshi, 121, 10, 733-741 , 121, 10, 733-741 2001 Refereed Japanese Disclose to all
K. Graf; P.D. Hindenberg; Y. Tokimizu; S. Naoe; M. Rudolph; F. Rominger; H. Ohno; A.S.K. Hashmi K. Graf; P.D. Hindenberg; Y. Tokimizu; S. Naoe; M. Rudolph; F. Rominger; H. Ohno; A.S.K. Hashmi The role of acetylides in dual gold catalysis: A mechanistic investigation of the selectivity difference in the naphthalene synthesis from diynes The role of acetylides in dual gold catalysis: A mechanistic investigation of the selectivity difference in the naphthalene synthesis from diynes ChemCatChem, 6, 1, 199-204 , 6, 1, 199-204 ChemCatChem, 6, 1, 199-204 2014 Refereed English Disclose to all
H. Ohno; H. Chiba; S. Inuki; S. Oishi; N. Fujii H. Ohno; H. Chiba; S. Inuki; S. Oishi; N. Fujii The synthesis of alkaloids using transition-metal-catalyzed intramolecular amination reactions The synthesis of alkaloids using transition-metal-catalyzed intramolecular amination reactions Synlett, 25, 2, 179-192 , 25, 2, 179-192 Synlett, 25, 2, 179-192 2014 Refereed English Disclose to all
Y. Yoshimitsu; J. Miyagaki; S. Oishi; N. Fujii; H. Ohno Y. Yoshimitsu; J. Miyagaki; S. Oishi; N. Fujii; H. Ohno Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis Synthesis of pachastrissamine (jaspine B) and its derivatives by the late-stage introduction of the C-2 alkyl side-chains using olefin cross metathesis Tetrahedron, 69, 21, 4211-4220 , 69, 21, 4211-4220 Tetrahedron, 69, 21, 4211-4220 2013/05/27 Refereed English Disclose to all
T. Suzuki; Y. Tokimizu; Y. Sakano; R. Katoono; K. Fujiwara; S. Naoe; N. Fujii; H. Ohno T. Suzuki; Y. Tokimizu; Y. Sakano; R. Katoono; K. Fujiwara; S. Naoe; N. Fujii; H. Ohno 5,10-Dihydrobenzo[a]indolo[2,3-c]carbazole: A highly fluorescent disk-shaped electron donor exhibiting dual UVvisNIR and fluorescence spectral changes upon electrolysis 5,10-Dihydrobenzo[a]indolo[2,3-c]carbazole: A highly fluorescent disk-shaped electron donor exhibiting dual UVvisNIR and fluorescence spectral changes upon electrolysis Chemistry Letters, 42, 9, 1001-1003 , 42, 9, 1001-1003 Chemistry Letters, 42, 9, 1001-1003 2013 Refereed English Disclose to all
H. Ohno H. Ohno Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds Gold-Catalyzed Cascade Reactions of Alkynes for Construction of Polycyclic Compounds Israel Journal of Chemistry, 53, 11-12, 869-882 , 53, 11-12, 869-882 Israel Journal of Chemistry, 53, 11-12, 869-882 2013 Refereed English Disclose to all
H. Chiba; Y. Sakai; S. Oishi; N. Fujii; H. Ohno H. Chiba; Y. Sakai; S. Oishi; N. Fujii; H. Ohno Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (-)-quinocarcinamide Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (-)-quinocarcinamide Tetrahedron Letters, 53, 46, 6273-6276 , 53, 46, 6273-6276 Tetrahedron Letters, 53, 46, 6273-6276 2012/11/14 Refereed English Disclose to all
R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; E. Kodama; M. Matsuoka; N. Fujii R. Masuda; S. Oishi; N. Tanahara; H. Ohno; A. Hirasawa; G. Tsujimoto; E. Kodama; M. Matsuoka; N. Fujii Development and application of fluorescent SDF-1 derivatives Development and application of fluorescent SDF-1 derivatives Future Medicinal Chemistry, 4, 7, 837-844 , 4, 7, 837-844 Future Medicinal Chemistry, 4, 7, 837-844 2012/05 Refereed English Disclose to all
Z. Hou; Y. Suzuki; S. Oishi; N. Fujii; H. Ohno Z. Hou; Y. Suzuki; S. Oishi; N. Fujii; H. Ohno Efficient synthesis of aminomethylated azaindoles and corresponding pyrrole-fused derivatives by copper-catalyzed domino multicomponent coupling and cyclization Efficient synthesis of aminomethylated azaindoles and corresponding pyrrole-fused derivatives by copper-catalyzed domino multicomponent coupling and cyclization Tetrahedron, 68, 6, 1695-1703 , 68, 6, 1695-1703 Tetrahedron, 68, 6, 1695-1703 2012/02/11 Refereed English Disclose to all
Y. Suzuki; S. Naoe; S. Oishi; N. Fujii; H. Ohno Y. Suzuki; S. Naoe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed three-component annulation: Efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones Gold-catalyzed three-component annulation: Efficient synthesis of highly functionalized dihydropyrazoles from alkynes, hydrazines, and aldehydes or ketones Organic Letters, 14, 1, 326-329 , 14, 1, 326-329 Organic Letters, 14, 1, 326-329 2012/01/06 Refereed English Disclose to all
H. Ohno; M. Yamamoto; M. Iuchi; N. Fujii; T. Tanaka H. Ohno; M. Yamamoto; M. Iuchi; N. Fujii; T. Tanaka Palladium-catalyzed construction of polycyclic heterocycles by an alkyne insertion and direct arylation cascade Palladium-catalyzed construction of polycyclic heterocycles by an alkyne insertion and direct arylation cascade Synthesis, 16, 2567-2578 , 16, 2567-2578 Synthesis, 16, 2567-2578 2011/08 Refereed English Disclose to all
Y. Tokimizu; Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Y. Tokimizu; Y. Ohta; H. Chiba; S. Oishi; N. Fujii; H. Ohno Direct synthesis of highly fused perimidines by copper(I)-catalyzed hydroamination of 2-ethynylbenzaldehydes Direct synthesis of highly fused perimidines by copper(I)-catalyzed hydroamination of 2-ethynylbenzaldehydes Tetrahedron, 67, 29, 5168-5175 , 67, 29, 5168-5175 Tetrahedron, 67, 29, 5168-5175 2011/07/22 Refereed English Disclose to all
H. Iwasaki; N. Tsutsui; T. Eguchi; H. Ohno; M. Yamashita; T. Tanaka H. Iwasaki; N. Tsutsui; T. Eguchi; H. Ohno; M. Yamashita; T. Tanaka A novel samarium(II)-mediated tandem spirocyclization onto an aromatic ring A novel samarium(II)-mediated tandem spirocyclization onto an aromatic ring Tetrahedron Letters, 52, 15, 1770-1772 , 52, 15, 1770-1772 Tetrahedron Letters, 52, 15, 1770-1772 2011 Refereed English Disclose to all
S. Inuki; S. Oishi; N. Fujii; H. Ohno S. Inuki; S. Oishi; N. Fujii; H. Ohno Total synthesis of ((±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group (Oroganic Letters (2008) 10 (5239)) Total synthesis of ((±)-lysergic acid, lysergol, and isolysergol by palladium-catalyzed domino cyclization of amino allenes bearing a bromoindolyl group (Oroganic Letters (2008) 10 (5239)) Organic Letters, 13, 8, 2145- , 13, 8, 2145- Organic Letters, 13, 8, 2145- 2011 Refereed English Disclose to all
S. Oishi; K. Watanabe; S. Ito; M. Tanaka; H. Nishikawa; H. Ohno; K. Shimane; K. Izumi; Y. Sakagami; E.N. Kodama; M. Matsuoka; A. Asai; N. Fujii S. Oishi; K. Watanabe; S. Ito; M. Tanaka; H. Nishikawa; H. Ohno; K. Shimane; K. Izumi; Y. Sakagami; E.N. Kodama; M. Matsuoka; A. Asai; N. Fujii Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants MedChemComm, 1, 4, 276-281 , 1, 4, 276-281 MedChemComm, 1, 4, 276-281 2010/10 Refereed English Disclose to all
K. Hirano; Y. Inaba; T. Watanabe; S. Oishi; N. Fujii; H. Ohno K. Hirano; Y. Inaba; T. Watanabe; S. Oishi; N. Fujii; H. Ohno Gold-catalyzed intramolecular alkyne cycloisomerization cascade: Direct synthesis of aryl-annulated[a]carbazoles from aniline-substituted diethynylarenes Gold-catalyzed intramolecular alkyne cycloisomerization cascade: Direct synthesis of aryl-annulated[a]carbazoles from aniline-substituted diethynylarenes Advanced Synthesis and Catalysis, 352, 2/3, 368-372 , 352, 2/3, 368-372 Advanced Synthesis and Catalysis, 352, 2/3, 368-372 2010/02 Refereed English Disclose to all
T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii T. Narumi; K. Tomita; E. Inokuchi; K. Kobayashi; S. Oishi; H. Ohno; N. Fujii Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic Diastereoselective synthesis of highly functionalized fluoroalkene dipeptide isosteres and its application to Fmoc-based solid-phase synthesis of a cyclic pentapeptide mimetic Tetrahedron, 64, 19, 4332-4346 , 64, 19, 4332-4346 Tetrahedron, 64, 19, 4332-4346 2008/05/05 Refereed English Disclose to all
M. Tanaka; S. Oishi; H. Ohno; N. Fujii M. Tanaka; S. Oishi; H. Ohno; N. Fujii A novel oxazolidine linker for the synthesis of peptide aldehydes A novel oxazolidine linker for the synthesis of peptide aldehydes International Journal of Peptide Research and Therapeutics, 13, 1-2, 271-279 , 13, 1-2, 271-279 International Journal of Peptide Research and Therapeutics, 13, 1-2, 271-279 2007/06 Refereed English Disclose to all
H. Ohno; Y. Ohta; S. Oishi; N. Fujii H. Ohno; Y. Ohta; S. Oishi; N. Fujii Erratum: Direct synthesis of 2-(aminomethyl)-indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions (Angewandte Chemie - International Edition (2007) 46, (2295-2298) DOI: 10.1002/anie.200604342) Erratum: Direct synthesis of 2-(aminomethyl)-indoles through copper(I)-catalyzed domino three-component coupling and cyclization reactions (Angewandte Chemie - International Edition (2007) 46, (2295-2298) DOI: 10.1002/anie.200604342) Angewandte Chemie - International Edition, 46, 18, 3173- , 46, 18, 3173- Angewandte Chemie - International Edition, 46, 18, 3173- 2007 Refereed English Disclose to all
H. Ohno H. Ohno Vinylaziridines in Organic Synthesis Vinylaziridines in Organic Synthesis Aziridines and Epoxides in Organic Synthesis, 37-71 , 37-71 Aziridines and Epoxides in Organic Synthesis, 37-71 2006 Refereed English Disclose to all
T. Tanaka; K. Hiramatsu; Y. Kobayashi; H. Ohno T. Tanaka; K. Hiramatsu; Y. Kobayashi; H. Ohno Chemo- and stereoselectivity in titanium-mediated regioselective ring-opening reaction of epoxides at the more substituted carbon Chemo- and stereoselectivity in titanium-mediated regioselective ring-opening reaction of epoxides at the more substituted carbon Tetrahedron, 61, 28, 6726-6742 , 61, 28, 6726-6742 Tetrahedron, 61, 28, 6726-6742 2005 Refereed English Disclose to all
大野 浩章 大野 浩章 Asymmetric construction of quaternary carbon centers by allyltitanium-mediated stereospecific ring-opening reaction of 2,3-epoxy alcohols. Asymmetric construction of quaternary carbon centers by allyltitanium-mediated stereospecific ring-opening reaction of 2,3-epoxy alcohols. Tetrahedron Lett. 45/1, 75–78, 45, 1, 75-78 , 45, 1, 75-78 Tetrahedron Lett. 45/1, 75–78, 45, 1, 75-78 2004 Refereed English Disclose to all
H. Ohno; K. Hiramatsu; T. Tanaka H. Ohno; K. Hiramatsu; T. Tanaka Asymmetric construction of quaternary carbon centers by titanium-mediated stereospecific allylation of 2,3-epoxy alcohol derivatives Asymmetric construction of quaternary carbon centers by titanium-mediated stereospecific allylation of 2,3-epoxy alcohol derivatives Tetrahedron Letters, 45, 1, 75-78 , 45, 1, 75-78 Tetrahedron Letters, 45, 1, 75-78 2004 Refereed English Disclose to all
H. Ohno; M. Okumura; S.-I. Maeda; H. Iwasaki; R. Wakayama; T. Tanaka H. Ohno; M. Okumura; S.-I. Maeda; H. Iwasaki; R. Wakayama; T. Tanaka Samarium(II)-promoted radical spirocyclization onto an aromatic ring Samarium(II)-promoted radical spirocyclization onto an aromatic ring Journal of Organic Chemistry, 68, 20, 7722-7732 , 68, 20, 7722-7732 Journal of Organic Chemistry, 68, 20, 7722-7732 2003/10/03 Refereed English Disclose to all
H. Ohno; R. Wakayama; S.-I. Maeda; H. Iwasaki; M. Okumura; C. Iwata; H. Mikamiyama; T. Tanaka H. Ohno; R. Wakayama; S.-I. Maeda; H. Iwasaki; M. Okumura; C. Iwata; H. Mikamiyama; T. Tanaka Radical cyclization by Ipso substitution of the methoxy group: Considerable effect of HMPA on samarium-mediated cyclization Radical cyclization by Ipso substitution of the methoxy group: Considerable effect of HMPA on samarium-mediated cyclization Journal of Organic Chemistry, 68, 15, 5909-5916 , 68, 15, 5909-5916 Journal of Organic Chemistry, 68, 15, 5909-5916 2003/07/25 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; M. Ohata; T. Tanaka H. Ohno; H. Hamaguchi; M. Ohata; T. Tanaka Bromoallenes as synthetic equivalents of allyl dications: Synthesis of medium-sized nitrogen heterocycles through the cyclization of bromoallenes in the presence of a palladium(0) catalyst and an alcohol Bromoallenes as synthetic equivalents of allyl dications: Synthesis of medium-sized nitrogen heterocycles through the cyclization of bromoallenes in the presence of a palladium(0) catalyst and an alcohol Angewandte Chemie - International Edition, 42, 15, 1749-1753 , 42, 15, 1749-1753 Angewandte Chemie - International Edition, 42, 15, 1749-1753 2003 Refereed English Disclose to all
H. Ohno; K. Miyamura; Y. Takeoka; T. Tanaka H. Ohno; K. Miyamura; Y. Takeoka; T. Tanaka Palladium(0)-catalyzed tandem cyclization of allenenes Palladium(0)-catalyzed tandem cyclization of allenenes Angewandte Chemie - International Edition, 42, 23, 2647-2650 , 42, 23, 2647-2650 Angewandte Chemie - International Edition, 42, 23, 2647-2650 2003 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka H. Ohno; H. Hamaguchi; M. Ohata; S. Kosaka; T. Tanaka Novel synthesis of azocine, azepine, oxocine, and oxepine derivatives by palladium-catalyzed medium-ring formation from bromoallenes Novel synthesis of azocine, azepine, oxocine, and oxepine derivatives by palladium-catalyzed medium-ring formation from bromoallenes Heterocycles, 61, 65-68 , 61, 65-68 Heterocycles, 61, 65-68 2003 Refereed English Disclose to all
H. Ohno; K. Ando; H. Hamaguchi; Y. Takeoka; T. Tanaka H. Ohno; K. Ando; H. Hamaguchi; Y. Takeoka; T. Tanaka A highly cis-selective synthesis of 2-ethynylaziridines by intramolecular amination of chiral bromoallenes: Improvement of stereoselectivity based on the computational investigation A highly cis-selective synthesis of 2-ethynylaziridines by intramolecular amination of chiral bromoallenes: Improvement of stereoselectivity based on the computational investigation Journal of the American Chemical Society, 124, 51, 15255-15266 , 124, 51, 15255-15266 Journal of the American Chemical Society, 124, 51, 15255-15266 2002/12/25 Refereed English Disclose to all
M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka; Y. Takemoto M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka; Y. Takemoto Asymmetric synthesis of β<sup>2,3</sup>-amino acids by InI-Pd(0)-promoted metalation and addition of chiral 2-vinylaziridines Asymmetric synthesis of β<sup>2,3</sup>-amino acids by InI-Pd(0)-promoted metalation and addition of chiral 2-vinylaziridines Tetrahedron, 58, 26, 5231-5239 , 58, 26, 5231-5239 Tetrahedron, 58, 26, 5231-5239 2002/06/24 Refereed English Disclose to all
H. Ohno; S.-I. Maeda; M. Okumura; R. Wakayama; T. Tanaka H. Ohno; S.-I. Maeda; M. Okumura; R. Wakayama; T. Tanaka The first samarium(II)-mediated stereoselective spirocyclization onto an aromatic ring The first samarium(II)-mediated stereoselective spirocyclization onto an aromatic ring Chemical Communications, 4, 316-317 , 4, 316-317 Chemical Communications, 4, 316-317 2002 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka Stereoselective synthesis of chiral 2,3-cis-2-ethynylaziridines by base-mediated intramolecular amination of bromoallenes Stereoselective synthesis of chiral 2,3-cis-2-ethynylaziridines by base-mediated intramolecular amination of bromoallenes Organic Letters, 3, 15, 2269-2271 , 3, 15, 2269-2271 Organic Letters, 3, 15, 2269-2271 2001/07/26 Refereed English Disclose to all
H. Ohno; M. Anzai; A. Toda; S. Ohishi; N. Fujii; T. Tanaka; Y. Takemoto; T. Ibuka H. Ohno; M. Anzai; A. Toda; S. Ohishi; N. Fujii; T. Tanaka; Y. Takemoto; T. Ibuka Stereoselective synthesis of 2-alkenylaziridines and 2-alkenylazetidines by palladium-catalyzed intramolecular amination of α- and β-amino allenes Stereoselective synthesis of 2-alkenylaziridines and 2-alkenylazetidines by palladium-catalyzed intramolecular amination of α- and β-amino allenes Journal of Organic Chemistry, 66, 14, 4904-4914 , 66, 14, 4904-4914 Journal of Organic Chemistry, 66, 14, 4904-4914 2001/07/13 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka 2-Ethynylaziridines as chiral carbon nucleophiles: Stereoselective synthesis of 1,3-amino alcohols with three stereocenters via allenylindium reagents bearing a protected amino group 2-Ethynylaziridines as chiral carbon nucleophiles: Stereoselective synthesis of 1,3-amino alcohols with three stereocenters via allenylindium reagents bearing a protected amino group Journal of Organic Chemistry, 66, 5, 1867-1875 , 66, 5, 1867-1875 Journal of Organic Chemistry, 66, 5, 1867-1875 2001/03/09 Refereed English Disclose to all
Y. Takemoto; M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka Y. Takemoto; M. Anzai; R. Yanada; N. Fujii; H. Ohno; T. Ibuka Stereoselective synthesis of nonracemic 1,3-amino alcohols from chiral 2-vinylaziridines by InI-Pd(0)-promoted metalation Stereoselective synthesis of nonracemic 1,3-amino alcohols from chiral 2-vinylaziridines by InI-Pd(0)-promoted metalation Tetrahedron Letters, 42, 9, 1725-1728 , 42, 9, 1725-1728 Tetrahedron Letters, 42, 9, 1725-1728 2001/02/26 Refereed English Disclose to all
S.M. Abdur Rahman; H. Ohno; H. Yoshino; N. Satoh; M. Tsukaguchi; K. Murakami; C. Iwata; N. Maezaki; T. Tanaka S.M. Abdur Rahman; H. Ohno; H. Yoshino; N. Satoh; M. Tsukaguchi; K. Murakami; C. Iwata; N. Maezaki; T. Tanaka A model study for the total synthesis of (±)-scopadulin: Stereoselective construction of the A/B ring system with desired functionalities A model study for the total synthesis of (±)-scopadulin: Stereoselective construction of the A/B ring system with desired functionalities Tetrahedron, 57, 1, 127-134 , 57, 1, 127-134 Tetrahedron, 57, 1, 127-134 2001 Refereed English Disclose to all
S.M.A. Rahman; H. Ohno; T. Tanaka S.M.A. Rahman; H. Ohno; T. Tanaka Improved method of an unusual conversion of aliphatic amines into alcohols Improved method of an unusual conversion of aliphatic amines into alcohols Tetrahedron Letters, 42, 45, 8007-8010 , 42, 45, 8007-8010 Tetrahedron Letters, 42, 45, 8007-8010 2001 Refereed English Disclose to all
S.M.A. Rahman; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki; T. Tanaka S.M.A. Rahman; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki; T. Tanaka Total synthesis of (±)-scopadulin Total synthesis of (±)-scopadulin Journal of Organic Chemistry, 66, 14, 4831-4840 , 66, 14, 4831-4840 Journal of Organic Chemistry, 66, 14, 4831-4840 2001 Refereed English Disclose to all
T. Tanaka; K. Murakami; A. Kanda; D. Patra; S. Yamamoto; N. Satoh; S.-W. Kim; S.M.A. Rahman; H. Ohno; C. Iwata T. Tanaka; K. Murakami; A. Kanda; D. Patra; S. Yamamoto; N. Satoh; S.-W. Kim; S.M.A. Rahman; H. Ohno; C. Iwata Total synthesis of (±)-stemodinone via an efficient ring-exchange strategy Total synthesis of (±)-stemodinone via an efficient ring-exchange strategy Journal of Organic Chemistry, 66, 21, 7107-7112 , 66, 21, 7107-7112 Journal of Organic Chemistry, 66, 21, 7107-7112 2001 Refereed English Disclose to all
S.M.A. Rahman; T. Tanaka; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki S.M.A. Rahman; T. Tanaka; H. Ohno; T. Murata; H. Yoshino; N. Satoh; K. Murakami; D. Patra; C. Iwata; N. Maezaki The first total synthesis of (±)-scopadulin, an antiviral aphidicolane diterpene The first total synthesis of (±)-scopadulin, an antiviral aphidicolane diterpene Organic Letters, 3, 4, 619-621 , 3, 4, 619-621 Organic Letters, 3, 4, 619-621 2001 Refereed English Disclose to all
H. Ohno; H. Hamaguchi; T. Tanaka H. Ohno; H. Hamaguchi; T. Tanaka Umpolung of chiral 2-ethynylaziridines: Indium(I)-mediated stereoselective synthesis of nonracemic 1,3-amino alcohols bearing three chiral centers, catalyzed by palladium(0) Umpolung of chiral 2-ethynylaziridines: Indium(I)-mediated stereoselective synthesis of nonracemic 1,3-amino alcohols bearing three chiral centers, catalyzed by palladium(0) Organic Letters, 2, 14, 2161-2163 , 2, 14, 2161-2163 Organic Letters, 2, 14, 2161-2163 2000/07/13 Refereed English Disclose to all
H. Ohno; A. Toda; S. Oishi; T. Tanaka; Y. Takemoto; N. Fujii; T. Ibuka H. Ohno; A. Toda; S. Oishi; T. Tanaka; Y. Takemoto; N. Fujii; T. Ibuka Novel synthesis of chiral terminal allenes via palladium(o)catalyzed reduction of mesylates of 2-bromoalk-2-en-1-ols bearing a protected amino group, using diethylzinc Novel synthesis of chiral terminal allenes via palladium(o)catalyzed reduction of mesylates of 2-bromoalk-2-en-1-ols bearing a protected amino group, using diethylzinc Tetrahedron Letters, 41, 26, 5131-5134 , 41, 26, 5131-5134 Tetrahedron Letters, 41, 26, 5131-5134 2000/06/24 Refereed English Disclose to all
H. Ohno; A. Toda; N. Fujii; Y. Takemoto; T. Tanaka; T. Ibuka H. Ohno; A. Toda; N. Fujii; Y. Takemoto; T. Tanaka; T. Ibuka Stereoselective synthesis of chiral amino allenes by organocopper- mediated anti-S(N)2\\'-substitution reaction of chiral ethynylaziridines Stereoselective synthesis of chiral amino allenes by organocopper- mediated anti-S(N)2\\'-substitution reaction of chiral ethynylaziridines Tetrahedron, 56, 18, 2811-2820 , 56, 18, 2811-2820 Tetrahedron, 56, 18, 2811-2820 2000/04/28 Refereed English Disclose to all
S.M.A. Rahman; H. Ohno; N. Maezaki; C. Iwata; T. Tanaka S.M.A. Rahman; H. Ohno; N. Maezaki; C. Iwata; T. Tanaka Efficient one-step conversion of primary aliphatic amines into primary alcohols: Application to a model study for the total synthesis of (±)-scopadulin Efficient one-step conversion of primary aliphatic amines into primary alcohols: Application to a model study for the total synthesis of (±)-scopadulin Organic Letters, 2, 18, 2893-2895 , 2, 18, 2893-2895 Organic Letters, 2, 18, 2893-2895 2000 Refereed English Disclose to all
K. Ando; T. Oishi; M. Hirama; H. Ohno; T. Ibuka K. Ando; T. Oishi; M. Hirama; H. Ohno; T. Ibuka Z-selective Horner-Wadsworth-Emmons reaction of ethyl (diarylphosphono)acetates using sodium iodide and DBU Z-selective Horner-Wadsworth-Emmons reaction of ethyl (diarylphosphono)acetates using sodium iodide and DBU Journal of Organic Chemistry, 65, 15, 4745-4749 , 65, 15, 4745-4749 Journal of Organic Chemistry, 65, 15, 4745-4749 2000 Refereed English Disclose to all
T. Tanaka; R. Wakayama; S.-I. Maeda; H. Mikamiyama; N. Maezaki; H. Ohno T. Tanaka; R. Wakayama; S.-I. Maeda; H. Mikamiyama; N. Maezaki; H. Ohno Unusual radical ipso-substitution reaction of an aromatic methoxy group induced by tris(trimethylsilyl)silane-AIBN or SmI<sub>2</sub> Unusual radical ipso-substitution reaction of an aromatic methoxy group induced by tris(trimethylsilyl)silane-AIBN or SmI<sub>2</sub> Chemical Communications, 14, 1287-1288 , 14, 1287-1288 Chemical Communications, 14, 1287-1288 2000 Refereed English Disclose to all
Ohno, H; Toda, A; Takemoto, Y; Fujii, N; Ibuka, T Ohno, H; Toda, A; Takemoto, Y; Fujii, N; Ibuka, T Convenient syntheses of chiral 3-substituted 2-ethynylaziridines Convenient syntheses of chiral 3-substituted 2-ethynylaziridines JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 20, 2949-2962 , 20, 2949-2962 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 20, 2949-2962 1999/10/21 Refereed English Disclose to all
M. Anzai; A. Toda; H. Ohno; Y. Takemoto; N. Fujii; T. Ibuka M. Anzai; A. Toda; H. Ohno; Y. Takemoto; N. Fujii; T. Ibuka Palladium-catalyzed regio- and stereoselective synthesis of N-protected 2,4-dialkylated azacyclobutanes from amino allenes Palladium-catalyzed regio- and stereoselective synthesis of N-protected 2,4-dialkylated azacyclobutanes from amino allenes Tetrahedron Letters, 40, 41, 7393-7397 , 40, 41, 7393-7397 Tetrahedron Letters, 40, 41, 7393-7397 1999/10/08 Refereed English Disclose to all
Ishii, K; Ohno, H; Takemoto, Y; Osawa, E; Yamaoka, Y; Fujii, N; Ibuka, T Ishii, K; Ohno, H; Takemoto, Y; Osawa, E; Yamaoka, Y; Fujii, N; Ibuka, T Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N arylsulfonylaminoalk-2-en-1-ols Selective synthesis of cis-2-vinyl-3-alkylaziridines and 3-pyrrolines from common intermediates (Z)-4-N arylsulfonylaminoalk-2-en-1-ols JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 15, 2155-2163 , 15, 2155-2163 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 15, 2155-2163 1999/08/07 Refereed English Disclose to all
H. Ohno; A. Toda; Y. Miwa; T. Taga; E. Osawa; Y. Yamaoka; N. Fujii; T. Ibuka H. Ohno; A. Toda; Y. Miwa; T. Taga; E. Osawa; Y. Yamaoka; N. Fujii; T. Ibuka First palladium-catalyzed aziridination reaction of amino allenes First palladium-catalyzed aziridination reaction of amino allenes Journal of Organic Chemistry, 64, 9, 2992-2993 , 64, 9, 2992-2993 Journal of Organic Chemistry, 64, 9, 2992-2993 1999/04/30 Refereed English Disclose to all
H. Ohno; A. Toda; N. Fujii; Y. Miwa; T. Taga; Y. Yamaoka; E. Osawa; T. Ibuka H. Ohno; A. Toda; N. Fujii; Y. Miwa; T. Taga; Y. Yamaoka; E. Osawa; T. Ibuka Sterically congested chiral activated aziridines: Synthesis of both 2,3- cis-and 2,3-Trans-2-alkenyl-3-alkylaziridines from common intermediates Sterically congested chiral activated aziridines: Synthesis of both 2,3- cis-and 2,3-Trans-2-alkenyl-3-alkylaziridines from common intermediates Tetrahedron Letters, 40, 7, 1331-1334 , 40, 7, 1331-1334 Tetrahedron Letters, 40, 7, 1331-1334 1999/02/12 Refereed English Disclose to all
Ishii, K; Ohno, H; Takemoto, Y; Ibuka, T Ishii, K; Ohno, H; Takemoto, Y; Ibuka, T Selective synthesis of nonracemic 3-pyrrolines and 2,3-cis-2-vinylaziridines from (Z)-amino allylic alcohols: A new synthetic route to chiral 3,4-dehydroproline Selective synthesis of nonracemic 3-pyrrolines and 2,3-cis-2-vinylaziridines from (Z)-amino allylic alcohols: A new synthetic route to chiral 3,4-dehydroproline SYNLETT, 2, 228-230 , 2, 228-230 SYNLETT, 2, 228-230 1999/02 Refereed English Disclose to all
H. Ohno; A. Toda; Y. Miwa; T. Taga; N. Fujii; T. Ibuka H. Ohno; A. Toda; Y. Miwa; T. Taga; N. Fujii; T. Ibuka Synthesis of chiral amino allenes via an organocyanocuprate-mediated ring-opening reaction of enantiopure ethynylaziridines Synthesis of chiral amino allenes via an organocyanocuprate-mediated ring-opening reaction of enantiopure ethynylaziridines Tetrahedron Letters, 40, 2, 349-352 , 40, 2, 349-352 Tetrahedron Letters, 40, 2, 349-352 1999/01/08 Refereed English Disclose to all
H. Tamamura; M. Yamashita; Y. Nakajima; K. Sakano; A. Otaka; H. Ohno; T. Ibuka; N. Fujii H. Tamamura; M. Yamashita; Y. Nakajima; K. Sakano; A. Otaka; H. Ohno; T. Ibuka; N. Fujii Regiospecific ring-opening reactions of β-aziridinyl ct, β-enoates with acids: Application to the stereoselective synthesis of a couple of diastereoisomeric (Zi)-alkene dipeptide isosteres from a single β-aziridinyl a, β-enoate and to the convenient prepa Regiospecific ring-opening reactions of β-aziridinyl ct, β-enoates with acids: Application to the stereoselective synthesis of a couple of diastereoisomeric (Zi)-alkene dipeptide isosteres from a single β-aziridinyl a, β-enoate and to the convenient prepa Journal of the Chemical Society - Perkin Transactions 1, 20, 2983-2996 , 20, 2983-2996 Journal of the Chemical Society - Perkin Transactions 1, 20, 2983-2996 1999 Refereed English Disclose to all
H. Ohno; A. Toda; N. Fujii; T. Ibuka H. Ohno; A. Toda; N. Fujii; T. Ibuka A convenient synthesis of activated enantiomerically pure 2- ethynylaziridines A convenient synthesis of activated enantiomerically pure 2- ethynylaziridines Tetrahedron Asymmetry, 9, 22, 3929-3933 , 9, 22, 3929-3933 Tetrahedron Asymmetry, 9, 22, 3929-3933 1998/11/27 Refereed English Disclose to all
Ohno, H; Ishii, K; Honda, A; Tamamura, H; Fujii, N; Takemoto, Y; Ibuka, T Ohno, H; Ishii, K; Honda, A; Tamamura, H; Fujii, N; Takemoto, Y; Ibuka, T A 2,3-cis-selective synthesis of aziridines bearing a vinyl group from allyl methyl carbonates and allyl mesylates A 2,3-cis-selective synthesis of aziridines bearing a vinyl group from allyl methyl carbonates and allyl mesylates JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 22, 3703-3716 , 22, 3703-3716 JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1, 22, 3703-3716 1998/11/21 Refereed English Disclose to all
A. Honda; H. Ohno; N. Mimura; T. Ibuka A. Honda; H. Ohno; N. Mimura; T. Ibuka Rhodium(I)- or iridium(I)-mediated equilibrated reactions of activated 2,3-cis- and trans-3-alkyl-2-vinylaziridines Rhodium(I)- or iridium(I)-mediated equilibrated reactions of activated 2,3-cis- and trans-3-alkyl-2-vinylaziridines Synlett, 9, 969-+ , 9, 969-+ Synlett, 9, 969-+ 1998/09 Refereed English Disclose to all
A. Toda; H. Aoyama; N. Mimura; H. Ohno; N. Fujii; T. Ibuka A. Toda; H. Aoyama; N. Mimura; H. Ohno; N. Fujii; T. Ibuka Reactions of n-arylsulfonyl-2,3-cis- and n-arylsulfonyl-2,3-frans-3-alkyl-2-vinylaziridines with organocopper reagents: importance of 2,3-cis-stereochemistry in controlling regio- and stereoselectivity Reactions of n-arylsulfonyl-2,3-cis- and n-arylsulfonyl-2,3-frans-3-alkyl-2-vinylaziridines with organocopper reagents: importance of 2,3-cis-stereochemistry in controlling regio- and stereoselectivity Journal of Organic Chemistry, 63, 20, 7053-7061 , 63, 20, 7053-7061 Journal of Organic Chemistry, 63, 20, 7053-7061 1998 Refereed English Disclose to all
T. Ibuka; N. Mimura; H. Ohno; K. Nakai; M. Akaji; H. Habashita; H. Tamamura; Y. Miwa; T. Taga; N. Fujii; Y. Yamamoto T. Ibuka; N. Mimura; H. Ohno; K. Nakai; M. Akaji; H. Habashita; H. Tamamura; Y. Miwa; T. Taga; N. Fujii; Y. Yamamoto Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an α,β-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsvdfonyl) 2-Enoates over the Other Three Stereoisomers Palladium(0)-Catalyzed Isomerization Reactions of Aziridines Bearing an α,β-Unsaturated Ester Group: A Thermodynamic Preference for Chiral Alkyl (2E)-4,5-cis-4,5-Epimino-N-(alkyl- or arylsvdfonyl) 2-Enoates over the Other Three Stereoisomers Journal of Organic Chemistry, 62, 9, 2982-2991 , 62, 9, 2982-2991 Journal of Organic Chemistry, 62, 9, 2982-2991 1997/05/02 Refereed English Disclose to all
H. Ohno; N. Mimura; A. Otaka; H. Tamamura; N. Fujii; T. Ibuka; I. Shimizu; A. Satake; Y. Yamamoto H. Ohno; N. Mimura; A. Otaka; H. Tamamura; N. Fujii; T. Ibuka; I. Shimizu; A. Satake; Y. Yamamoto Palladium-catalyzed reductive ring opening with formic acid of aziridines bearing an α,β-unsaturated ester group Palladium-catalyzed reductive ring opening with formic acid of aziridines bearing an α,β-unsaturated ester group Tetrahedron, 53, 38, 12933-12946 , 53, 38, 12933-12946 Tetrahedron, 53, 38, 12933-12946 1997 Refereed English Disclose to all
T. Ibuka; N. Mimura; H. Aoyama; M. Akaji; H. Ohno; Y. Miwa; T. Taga; K. Nakai; H. Tamamura; N. Fujii; Y. Yamamoto T. Ibuka; N. Mimura; H. Aoyama; M. Akaji; H. Ohno; Y. Miwa; T. Taga; K. Nakai; H. Tamamura; N. Fujii; Y. Yamamoto A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres A Thermodynamic Preference of Chiral N-Methanesulfonyl and N-Arenesulfonyl 2,3-cis-3-Alkyl-2-Vinylaziridines over Their 2,3-Trans-Isomers: Useful Palladium(0)-Catalyzed Equilibration Reactions for the Synthesis of (E)-Alkene Dipeptide Isosteres Journal of Organic Chemistry, 62, 4, 999-1015 , 62, 4, 999-1015 Journal of Organic Chemistry, 62, 4, 999-1015 1997 Refereed English Disclose to all
H. Aoyama; N. Mimura; H. Ohno; K. Ishii; A. Toda; H. Tamamura; A. Otaka; N. Fujii; T. Ibuka H. Aoyama; N. Mimura; H. Ohno; K. Ishii; A. Toda; H. Tamamura; A. Otaka; N. Fujii; T. Ibuka Regio- and stereoselectivity in reactions of 2,3-cis- and trans-3-alkyl-2-vinylaziridines with organocopper reagents: Importance of 2,3-cis-stereochemistry in controlling selectivity Regio- and stereoselectivity in reactions of 2,3-cis- and trans-3-alkyl-2-vinylaziridines with organocopper reagents: Importance of 2,3-cis-stereochemistry in controlling selectivity Tetrahedron Letters, 38, 42, 7383-7386 , 38, 42, 7383-7386 Tetrahedron Letters, 38, 42, 7383-7386 1997 Refereed English Disclose to all
H. Tamamura; M. Yamashita; H. Muramatsu; H. Ohno; T. Ibuka; A. Otaka; N. Fujii H. Tamamura; M. Yamashita; H. Muramatsu; H. Ohno; T. Ibuka; A. Otaka; N. Fujii Regiospecific ring-opening reactions of aziridines bearing an α,β-unsaturated ester group with trifluoroacetic acid or methanesulfonic acid: Application to the stereoselective synthesis of (E)-alkene dipeptide isosteres Regiospecific ring-opening reactions of aziridines bearing an α,β-unsaturated ester group with trifluoroacetic acid or methanesulfonic acid: Application to the stereoselective synthesis of (E)-alkene dipeptide isosteres Chemical Communications, 23, 2327-2328 , 23, 2327-2328 Chemical Communications, 23, 2327-2328 1997 Refereed English Disclose to all

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Title language:
Conference Activities & Talks
Title Title(Japanese) Title(English) Conference Conference(Japanese) Conference(English) Promotor Promotor(Japanese) Promotor(English) Date Language Assortment Disclose
⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤[Invited] ⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤ [Invited] 千葉大学大学院 薬学研究院 特別講義 千葉大学大学院 薬学研究院 特別講義 2018/06/08 Japanese Oral presentation(invited, special) Disclose to all
⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤[Invited] ⾦触媒を⽤いたアルカロイド型⾻格の構築と応⽤ [Invited] 岡山大学医歯薬学総合研究科 特別講演会 岡山大学医歯薬学総合研究科 特別講演会 2017/09/29 Japanese Oral presentation(invited, special) Disclose to all
⾦触媒を⽤いた複素環⾻格構築法の開発と応⽤[Invited] ⾦触媒を⽤いた複素環⾻格構築法の開発と応⽤ [Invited] 中外製薬 講演会 中外製薬 講演会 2017/09/13 Japanese Oral presentation(invited, special) Disclose to all
金触媒によるアルカロイド型骨格の構築と全合成研究[Invited] 金触媒によるアルカロイド型骨格の構築と全合成研究 [Invited] 第37回有機合成若手セミナー 第37回有機合成若手セミナー 2017/08/09 Japanese Oral presentation(invited, special) Disclose to all
Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations[Invited] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations [Invited] Direct Construction of Fused Nitrogen Heterocycles by Gold-Catalyzed Cascade Cyclizations [Invited] Nordic/Kyoto OMCOS 2017 Nordic/Kyoto OMCOS 2017 Nordic/Kyoto OMCOS 2017 2017/06/24 English Oral presentation(invited, special) Disclose to all
金触媒によるアルキンの活性化を基盤とした骨格構築反応の開発と応用[Invited] 金触媒によるアルキンの活性化を基盤とした骨格構築反応の開発と応用 [Invited] 明治薬科大学 特別講義 明治薬科大学 特別講義 2016/12/19 Japanese Oral presentation(invited, special) Disclose to all
金触媒を用いた反応の開発と応用[Invited] 金触媒を用いた反応の開発と応用 [Invited] 塩野義製薬(株) 創薬化学研究所セミナー 塩野義製薬(株) 創薬化学研究所セミナー 2016/10/03 Japanese Oral presentation(invited, special) Disclose to all
多重結合の連続活性化を用いた骨格構築反応の開発と応用[Invited] 多重結合の連続活性化を用いた骨格構築反応の開発と応用 [Invited] 近畿大学薬学研究科 大学院特別講義 近畿大学薬学研究科 大学院特別講義 2016/04/23 Japanese Oral presentation(invited, special) Disclose to all
Efficient Construction of Heterocyclic Scaffolds and Its Application[Invited] Efficient Construction of Heterocyclic Scaffolds and Its Application [Invited] Efficient Construction of Heterocyclic Scaffolds and Its Application [Invited] AGORA Bayer Meeting 2016 AGORA Bayer Meeting 2016 AGORA Bayer Meeting 2016 2016/04/15 English Oral presentation(invited, special) Disclose to all
Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles[Invited] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles [Invited] Gold-Catalyzed Cascade Cyclizations of Alkynes for Construction of Nitrogen Heterocycles [Invited] Pacifichem Pacifichem Pacifichem 2015/12/15 English Oral presentation(invited, special) Disclose to all
金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用[Invited] 金触媒によるアルキンの活性化を用いた骨格構築反応の開発と応用 [Invited] 名城大学特別講演会 名城大学特別講演会 2015/12/04 Japanese Oral presentation(invited, special) Disclose to all
アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用[Invited] アルキンの活性化を基盤とする複素環骨格構築反応の開発と応用 [Invited] 京大有機金属化学若手勉強会 京大有機金属化学若手勉強会 2015/10/31 Japanese Oral presentation(invited, special) Disclose to all
アルキンの活性化を基盤とする連続反応の開発と応用[Invited] アルキンの活性化を基盤とする連続反応の開発と応用 [Invited] 日本薬学会東海支部特別講演会 日本薬学会東海支部特別講演会 2015/05/29 Japanese Oral presentation(invited, special) Disclose to all
π結合の活性化を基盤とする連続反応の開発と応用[Invited] π結合の活性化を基盤とする連続反応の開発と応用 [Invited] 東京医科歯科大学 生材研セミナー 東京医科歯科大学 生材研セミナー 2015/01/26 Japanese Oral presentation(invited, special) Disclose to all
Gold-Catalyzed Annulations and Their Medicinal Applications[Invited] Gold-Catalyzed Annulations and Their Medicinal Applications [Invited] Gold-Catalyzed Annulations and Their Medicinal Applications [Invited] DPhG Annual Meeting 2014 DPhG Annual Meeting 2014 DPhG Annual Meeting 2014 2014/09/25 English Oral presentation(invited, special) Disclose to all
アレンやアルキンを合成素子とする連続反応の開発と応用[Invited] アレンやアルキンを合成素子とする連続反応の開発と応用 [Invited] 金沢大学 医歯薬保健研究域薬学系 講演会 金沢大学 医歯薬保健研究域薬学系 講演会 2014/06/13 Japanese Oral presentation(invited, special) Disclose to all
金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用[Invited] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用 [Invited] 京都府立大学 鴨叡会・生命分子化学科セミナー 京都府立大学 鴨叡会・生命分子化学科セミナー 2013/12/17 Japanese Oral presentation(invited, special) Disclose to all
金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用[Invited] 金触媒を用いた骨格構築反応の開発と生物活性化合物合成への応用 [Invited] 立命館大学 創薬基盤科学若手セミナー 立命館大学 創薬基盤科学若手セミナー 2013/12/09 Japanese Oral presentation(invited, special) Disclose to all
付加反応を用いて中心骨格を構築する天然物合成[Invited] 付加反応を用いて中心骨格を構築する天然物合成 [Invited] 第12回化学系薬学若手研究者セミナー 第12回化学系薬学若手研究者セミナー 2013/08/24 Japanese Oral presentation(invited, special) Disclose to all
高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究[Invited] 高い原子効率を有する遷移金属触媒反応を用いた天然物の合成研究 [Invited] 天然物ケミカルバイオロジー:分子標的と活性制御地区シンポジウム 天然物ケミカルバイオロジー:分子標的と活性制御地区シンポジウム 新学術領域「天然物ケミカルバイオロジー:分子標的と活性制御」 新学術領域「天然物ケミカルバイオロジー:分子標的と活性制御」 2013/03/16 Japanese Oral presentation(invited, special) Disclose to all
Gold-Catalyzed Reactions for Construction of Heterocycles[Invited] Gold-Catalyzed Reactions for Construction of Heterocycles [Invited] Gold-Catalyzed Reactions for Construction of Heterocycles [Invited] Dortmund University Special Lecture Dortmund University Special Lecture Dortmund University Special Lecture 2013/03/06 English Oral presentation(invited, special) Disclose to all
Gold-Catalyzed Reactions for Construction of Heterocycles[Invited] Gold-Catalyzed Reactions for Construction of Heterocycles [Invited] Gold-Catalyzed Reactions for Construction of Heterocycles [Invited] Heidelberg University Special Lecture Heidelberg University Special Lecture Heidelberg University Special Lecture 2013/03/04 English Oral presentation(invited, special) Disclose to all
触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用[Invited] 触媒的連続結合形成反応による縮環型複素環骨格の一挙構築と天然物合成への応用 [Invited] 6th Organic Syntheses Lectureship 6th Organic Syntheses Lectureship 東京大学薬学研究科 東京大学薬学研究科 2011/02/22 Japanese Oral presentation(invited, special) Disclose to all
触媒的連続結合形成反応による複素環骨格構築法の開発研究[Invited] 触媒的連続結合形成反応による複素環骨格構築法の開発研究 [Invited] 京都大学グローバルCOE プログラム有機若手ワークショップ 京都大学グローバルCOE プログラム有機若手ワークショップ 京都大学グローバルCOE プログラム 京都大学グローバルCOE プログラム 2010/09/14 Japanese Oral presentation(invited, special) Disclose to all
触媒的連続結合形成反応の開発とErgotアルカロイド全合成への応用[Invited] 触媒的連続結合形成反応の開発とErgotアルカロイド全合成への応用 [Invited] 第43回天然物化学談話会 第43回天然物化学談話会 天然物化学談話会 天然物化学談話会 2008/07/10 Japanese Oral presentation(invited, special) Disclose to all
アレンを合成素子とする触媒的連続結合形成反応の開発[Invited] アレンを合成素子とする触媒的連続結合形成反応の開発 [Invited] 有機合成協会関西支部賞受賞講演 有機合成協会関西支部賞受賞講演 有機合成協会関西支部 有機合成協会関西支部 2006/11/08 Japanese Oral presentation(invited, special) Disclose to all
アレン系化合物の新しい反応性に基づく有用反応の開発と連続環化反応への展開[Invited] アレン系化合物の新しい反応性に基づく有用反応の開発と連続環化反応への展開 [Invited] 日本薬学会第124年会(奨励賞受賞講演) 日本薬学会第124年会(奨励賞受賞講演) 日本薬学会 日本薬学会 2005/03/30 Japanese Oral presentation(invited, special) Disclose to all
アレンとパラジウム触媒の新しい反応性を利用した複素環合成[Invited] アレンとパラジウム触媒の新しい反応性を利用した複素環合成 [Invited] 日本薬学会第124年会ミニシンポジウム「有機合成化学の若い力」 日本薬学会第124年会ミニシンポジウム「有機合成化学の若い力」 日本薬学会 日本薬学会 2004/03/29 Japanese Oral presentation(invited, special) Disclose to all
パラジウム(0)を触媒としたアミノアレンの環化反応[Invited] パラジウム(0)を触媒としたアミノアレンの環化反応 [Invited] 第51回日本薬学会近畿支部総会・大会(受賞講演) 第51回日本薬学会近畿支部総会・大会(受賞講演) 日本薬学会近畿支部 日本薬学会近畿支部 2001/10/27 Japanese Oral presentation(invited, special) Disclose to all
From amino acids to peptide isosteres and heterocycles: implications to vinylaziridines and amino allene chemistry From amino acids to peptide isosteres and heterocycles: implications to vinylaziridines and amino allene chemistry 11th Akabori conference 11th Akabori conference Akabori Society Akabori Society 2006/09/11 English Oral presentation(invited, special) Disclose to all

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Title language:
Books etc
Author Author(Japanese) Author(English) Title Title(Japanese) Title(English) Publisher Publisher(Japanese) Publisher(English) Publication date Language Type Disclose
Hiroaki Ohno Hiroaki Ohno Intramolecular C−X Bond Formation between C=X or X−H and Alkynes (in Transition-Metal-Mediated Aromatic Ring Construction) Intramolecular C−X Bond Formation between C=X or X−H and Alkynes (in Transition-Metal-Mediated Aromatic Ring Construction) Wiley Wiley 2013 English Disclose to all
Hiroaki Ohno and Kiyoshi Tomioka Hiroaki Ohno and Kiyoshi Tomioka Synthesis by Substitution (in Science of Synthesis) Synthesis by Substitution (in Science of Synthesis) Thieme Thieme 2007 English Disclose to all
Hiroaki Ohno Hiroaki Ohno Vinylaziridines in Organic Synthesis (in Aziridines and Epoxides in Organic Synthesis) Vinylaziridines in Organic Synthesis (in Aziridines and Epoxides in Organic Synthesis) Wiley-VCH Wiley-VCH 2005 English Disclose to all
Hiroaki Ohno, Yasuo Nagaoka, and Kiyoshi Tomioka Hiroaki Ohno, Yasuo Nagaoka, and Kiyoshi Tomioka Enantioselective Synthesis of Allenes (in Modern Allene Chemistry) Enantioselective Synthesis of Allenes (in Modern Allene Chemistry) Wiley-VCH Wiley-VCH 2004 English Disclose to all
Title language:
Patents
Inventor(s) Inventor(s) (Japanese) Inventor(s) (English) Title Title(Japanese) Title(English) Stage Patent number Date Disclose
前田 英樹, 加藤 貴之, 松岡 雅雄, 志村 和也, 藤井 信孝, 大野 浩章, 大石 真也, 水原 司 前田 英樹, 加藤 貴之, 松岡 雅雄, 志村 和也, 藤井 信孝, 大野 浩章, 大石 真也, 水原 司 ピリミドベンゾチアジン−6−イミン誘導体またはその塩を含有するウイルス感染症の治療および/または予防のための薬剤 ピリミドベンゾチアジン−6−イミン誘導体またはその塩を含有するウイルス感染症の治療および/または予防のための薬剤 特許公開 特開2012-250973 2012/12/20 Disclose to all
辻本 豪三, 平澤 明, 村田 克美, 藤井 信孝, 大野 浩章, 大石 真也, 鈴木 大和, ゾンイェ ホウ, 仲西 功, 木下 誉富, 高倉 喜信, 西川 元也 辻本 豪三, 平澤 明, 村田 克美, 藤井 信孝, 大野 浩章, 大石 真也, 鈴木 大和, ゾンイェ ホウ, 仲西 功, 木下 誉富, 高倉 喜信, 西川 元也 キナーゼ阻害剤 キナーゼ阻害剤 特許公開 WO2012-121168 2012/09/13 Disclose to all
藤井 信孝, 大野 浩章, 大石 真也, 井ノ口 恵利子, 久保 達彦, 松岡 雅雄, 志村 和也 藤井 信孝, 大野 浩章, 大石 真也, 井ノ口 恵利子, 久保 達彦, 松岡 雅雄, 志村 和也 新規ケモカイン受容体拮抗剤 新規ケモカイン受容体拮抗剤 特許公開 WO2012-118124 2012/09/07 Disclose to all
藤井 信孝, 大野 浩章, 大石 真也, 渡部 敏明, 浅井 章良, 澤田 潤一 藤井 信孝, 大野 浩章, 大石 真也, 渡部 敏明, 浅井 章良, 澤田 潤一 Eg5阻害剤 Eg5阻害剤 特許公開 特開2012-051804 2012/03/15 Disclose to all
Title language:
Awards
Title(Japanese) Title(English) Organization name(Japanese) Organization name(English) Date
近畿支部奨励賞 Kinki Branch Award for Encouragement of Research 日本薬学会 The Pharmaceutical Society of Japan 2001/01/
奨励賞 Award for Young Scientists 日本薬学会 The Pharmaceutical Society of Japan 2005/03/
研究企画賞 Meiji Seika Award in Synthetic Organic Chemistry, Japan 有機合成化学協会 The Society of Synthetic Organic Chemistry, Japan 2005/12/
関西支部賞 Kansai Branch Award 有機合成化学協会関西支部 Kansai Branch, The Society of Synthetic Organic Chemistry, Japan 2006/11/
Banyu Chemist Award Banyu Chemist Award 万有生命科学振興国際交流財団 Banyu Life Science Foundation 2013/11/
Thieme Chemistry Journals Award Thieme Chemistry Journals Award Thieme Thieme 2014/02/
最優秀教員賞 Best Teacher Award 京都大学薬学部 Faculty of Pharmaceutical Sciences, Kyoto University 2014/10/24
External funds, competitive funds and Grants-in-Aid for Scientific Research(kaken)
Type Position Title(Japanese) Title(English) Period
奨励研究(A) Representative 高活性な降圧剤及びプロテアーゼ阻害剤の開発を指向したアミノアレンの合成研究 2000-2001
若手研究(B) Representative 生物活性を有する含窒素複素環の自在な合成を指向した新規環形成反応の開発研究 2003-2004
若手研究(B) Representative 複雑な構造を有する生物活性複素環の一挙合成法の開発と環境調和型連続反応への展開 2005-2006
若手研究(A) Representative 触媒的連続多点制御反応を基盤とする高原子効率分子構築法の開発と機能性分子への応用 2007-2009
基盤研究(C) Representative 触媒的連続環化反応を基盤とした生物活性天然物の多様性指向型全合成研究 2010-2012
新学術領域研究 Representative 触媒的多成分反応・高原子効率反応の高度集積化と創薬展開 2010-2011
若手研究(A) Representative π結合の連続活性化を基軸とする革新的分子変換法の開発と創薬リードの創出 Development of Inovative Molecular Transformations Based on Consecutive pai-Activation and Its Application to Drug Discovery 2012-2015
新学術領域研究 Representative 原子移動型反応の高度集積化による多環式芳香族化合物の合成と創薬展開 Integration of Atom-Transfer Reactions for the Synthesis of Polycyclic Arenes and Its Application to Drug Discovery 2012-2013
基盤研究(B) Representative 近接効果を利用した遷移状態制御による選択的活性化法の開発と創薬展開 Selective Activation Based on Control of Transition States by the Neighboring Effect and Its Medicinal Applications 2015-2018
基盤研究(B) Representative 多環式骨格構築反応を基軸とする生物活性インドールアルカロイドの全合成と創薬展開 Synthetic and Medicinal Studies on Bioactive Indole Alkaloids Based on Direct Construction of Polycyclic Ring Systems 2017-2020
基盤研究(B) Representative 近接効果を利用した遷移状態制御による選択的活性化法の開発と創薬展開 (平成29年度分) 2017/04/01-2018/03/31
基盤研究(B) Representative 多環式骨格構築反応を基軸とする生物活性インドールアルカロイドの全合成と創薬展開 (平成29年度分) 2017/04/01-2018/03/31
新学術領域研究 Representative 反応集積化によるアルカロイドの全合成と中分子化戦略 Syntheses and Middle Molecular Strategy of Alkaloids Based on Reaction Integration 2018/04/01-2019/03/31

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Teaching subject(s)
Name(Japanese) Name(English) Term Department Period
有機化学I(化学結合論) 前期 薬学部 2011/04-2012/03
特別実習(ケモゲノミクス・薬品有機製造学) 通年 薬学部 2011/04-2012/03
基礎有機化学A Basic Organic Chemistry A 前期 全学共通科目 2011/04-2012/03
特別実習[ケモゲノミクス・薬品有機製造学 通年 薬学部 2011/04-2012/03
創薬リード探索技術 Drug Discovery & Development II: 後期不定 薬学研究科 2011/04-2012/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2011/04-2012/03
リード化合物探索スキル(秋入学用) Skill Development for Lead Discovery 後期前期 薬学研究科 2011/04-2012/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2011/04-2012/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 前期不定 薬学研究科 2011/04-2012/03
基盤有機化学実験技術(秋入学用) Basic Laboratory Techniques in Organic Chemistry 後期不定 薬学研究科 2011/04-2012/03
基盤有機化学概論 Introduction to Basic Organic Chemistry 前期不定 薬学研究科 2011/04-2012/03
基盤有機化学特論Ⅰ Advanced Basic Organic Chemistry I 後期不定 薬学研究科 2011/04-2012/03
基盤薬品創製化学実習 Laboratory Practice in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04-2012/03
基盤薬品創製化学実験 Research in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04-2012/03
基盤薬品創製化学演習 Seminar in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems 通年不定 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系コンテンツ制作(秋入学) Advanced Methods in Systems 後期前期 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系研究 Research in Systems 通年不定 薬学研究科 2011/04-2012/03
システム生物学・医薬創成系研究(秋入学用) Research in Systems 後期前期 薬学研究科 2011/04-2012/03
薬学専門実習II 前期 薬学部 2011/04-2012/03
薬学専門実習2 前期 薬学部 2011/04-2012/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2012/04-2013/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2012/04-2013/03
博士後期課程特論 doctoral program 前期集中 薬学研究科 2012/04-2013/03
博士後期課程特論 doctoral program 後期集中 薬学研究科 2012/04-2013/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 前期不定 薬学研究科 2012/04-2013/03
基盤有機化学実験技術 Basic Laboratory Techniques in Organic Chemistry 後期不定 薬学研究科 2012/04-2013/03
基盤有機化学概論 Introduction to Basic Organic Chemistry 前期不定 薬学研究科 2012/04-2013/03
基盤有機化学特論II Advanced Basic Organic Chemistry II 後期不定 薬学研究科 2012/04-2013/03
基盤薬品創製化学実習 Laboratory Practice in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04-2013/03
基盤薬品創製化学実験 Research in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04-2013/03
基盤薬品創製化学演習 Seminar in Basic Medicinal and Organic Chemistry 通年不定 薬学研究科 2012/04-2013/03
基礎有機化学A Basic Organic Chemistry A 前期 全学共通科目 2012/04-2013/03
有機化学I(化学結合論) Organic Chemistry I(Bonding in Organic Chemistry) 前期 薬学部 2012/04-2013/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2012/04-2013/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2012/04-2013/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2012/04-2013/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2012/04-2013/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2012/04-2013/03
薬学専門実習II Pharmaceutical Laboratory II:Organic Chemistry 前期 薬学部 2012/04-2013/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2012/04-2013/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2013/04-2014/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2013/04-2014/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2013/04-2014/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2013/04-2014/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2013/04-2014/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2013/04-2014/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2013/04-2014/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2013/04-2014/03
博士後期課程特論 doctoral program 前期集中 薬学研究科 2013/04-2014/03
博士後期課程特論 doctoral program 後期集中 薬学研究科 2013/04-2014/03
基礎有機化学B Basic Organic Chemistry B 後期 全学共通科目 2013/04-2014/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2013/04-2014/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2014/04-2015/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2014/04-2015/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2014/04-2015/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2014/04-2015/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2014/04-2015/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2014/04-2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2014/04-2015/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2014/04-2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2014/04-2015/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2014/04-2015/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2014/04-2015/03
基礎有機化学B Basic Organic Chemistry B 後期 全学共通科目 2014/04-2015/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2014/04-2015/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2015/04-2016/03
くすりの化学 Organic Chemistry of Pharmaceuticals 前期 全学共通科目 2015/04-2016/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2015/04-2016/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2015/04-2016/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2015/04-2016/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2015/04-2016/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2015/04-2016/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2015/04-2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2015/04-2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2015/04-2016/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2015/04-2016/03
薬学専門実習2 Pharmaceutical Laboratory 2 : Organic Chemistry 前期 薬学部 2015/04-2016/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2016/04-2017/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2016/04-2017/03
医薬創成プロセス概論 Introduction to Drug Discovery Sciences 前期不定 薬学研究科 2016/04-2017/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2016/04-2017/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2016/04-2017/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2016/04-2017/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2016/04-2017/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2016/04-2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2016/04-2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2016/04-2017/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2016/04-2017/03
創薬有機化学概論 Introduction to Organic Chemistry for Drug Discovery 前期不定 薬学研究科 2017/04-2018/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2017/04-2018/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2017/04-2018/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2017/04-2018/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2017/04-2018/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2017/04-2018/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2017/04-2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2017/04-2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2017/04-2018/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2017/04-2018/03
創薬リード探索技術 Drug Discovery & Development II: Lead Discovery Technology 後期不定 薬学研究科 2018/04-2019/03
創薬有機化学概論 Introduction to Organic Chemistry for Drug Discovery 前期不定 薬学研究科 2018/04-2019/03
リード化合物探索スキル Skill Development for Lead Discovery 通年不定 薬学研究科 2018/04-2019/03
基盤有機化学特論II Advanced Basic Organic Chemistry II 後期不定 薬学研究科 2018/04-2019/03
基礎有機化学II Basic Organic Chemistry II 後期 全学共通科目 2018/04-2019/03
特別実習(ケモゲノミクス・薬品有機製造学) Research Training(Chemogenomics) 通年 薬学部 2018/04-2019/03
特別実習[ケモゲノミクス・薬品有機製造学] Research Training(Chemogenomics) 通年 薬学部 2018/04-2019/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 後期前期 薬学研究科 2018/04-2019/03
システム生物学・医薬創成系コンテンツ制作 Advanced Methods in Systems Biology & Drug Discovery 通年不定 薬学研究科 2018/04-2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 後期前期 薬学研究科 2018/04-2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Dicovery 通年不定 薬学研究科 2018/04-2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 後期前期 薬学研究科 2018/04-2019/03
システム生物学・医薬創成系研究 Research in Systems Biology & Drug Discovery 通年不定 薬学研究科 2018/04-2019/03
生理化学概論 Outline of Physiological Chemistry 後期集中 全学共通科目 2018/04-2019/03
臨床薬学概論 Introduction to Clinical Pharmacy 前期不定 薬学研究科 2018/04-2019/03

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School management (title, position)
Title Period
外国語教育専門委員会 委員 2008/04/01-2011/03/31
国際高等教育院 企画評価専門委員会 委員 2015/04/01-2017/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2013/07/05-2014/06/30
国際高等教育院 企画評価専門委員会 化学部会 委員 2015/05/01-2016/04/30
国際高等教育院 企画評価専門委員会 化学部会 委員 2016/05/01-2017/04/30
学生生活委員会 委員 2016/04/01-2018/03/31
学生生活委員会第一小委員会 委員 2016/04/01-2018/03/31
京都大学奨学金返還免除候補者選考委員会 4号委員 2016/04/01-2018/03/31
オープンキャンパス委員会 委員 2016/01/01-2016/12/31
図書館協議会 協議員 2017/04/01-2019/03/31
学生生活委員会第一小委員会 委員長 2016/04/01-2018/03/31
京都大学奨学金返還免除候補者選考委員会 委員長 2016/04/01-2018/03/31
学生表彰選考委員会 委員 -
国際高等教育院 企画評価専門委員会 委員 2017/04/01-2019/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2017/05/01-2018/03/31
学生表彰選考委員会 2018/01/01-2018/03/31
国際高等教育院 企画評価専門委員会 化学部会 委員 2018/04/01-2019/03/31
国際高等教育院 基盤企画評価専門委員会 委員 2017/04/01-2019/03/31

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Faculty management (title, position)
Title Period
薬学研究科 就職委員 2017/04/01-2019/03/31
薬学研究科 学生委員(先任教員) 2017/04/01-2018/03/31
薬学研究科 環境・安全衛生委員会委員長 2016/04/01-2018/03/31
薬学研究科 図書委員会委員長 2017/04/01-2019/03/31