森﨑一宏

Last Update: 2019/08/07 10:39:21

Name(Kanji/Kana/Abecedarium Latinum)

森﨑一宏/モリサキカズヒロ/Morisaki, Kazuhiro

Primary Affiliation(Org1/Job title)

Institute for Chemical Research (ICR)/Assistant Professor

Affiliated programs (koza)

Org1	Job title
Graduate Schools Pharmaceutical Sciences	Assistant Professor

Academic Degree

Field(Japanese)	Field(English)	University(Japanese)	University(English)	Method
修士（創薬科学）		九州大学
博士（創薬科学）		九州大学

ORCID ID

https://orcid.org/0000-0002-5692-4726

researchmap URL

https://researchmap.jp/7000023080

Research Topics

(Japanese)
有機合成における以下の未解決課題に取り組んでいる。・C-H官能基化反応における選択性制御および遠隔位認識・触媒的遠隔位不斉誘導・超分子の不斉合成・不斉記憶型反応による非天然アミノ酸含有ペプチドの効率的合成
(English)
Site-selective C-H bond functionalization via remote functionality recognition Remote asymmetric induction Asymmetric synthesis of topological chiral molecules Development of facile synthetic methods for unnatural amino acid-containing peptides via Memory Of Chirality

Fields of research (key words)

Key words(Japanese)	Key words(English)
位置選択的反応、 C-H官能基化反応	Site-Selectivity, C-H functionalization
遠隔位不斉誘導	Remote Assymetric Induction

Published Papers

Author	Author(Japanese)	Author(English)	Title	Title(Japanese)	Title(English)	Bibliography	Bibliography(Japanese)	Bibliography(English)	Publication date	Refereed paper	Disclose
Ryohei Yonesaki, Yuta Kondo, Walaa Akkad, Masanao Sawa, Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	Ryohei Yonesaki, Yuta Kondo, Walaa Akkad, Masanao Sawa, Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	Ryohei Yonesaki, Yuta Kondo, Walaa Akkad, Masanao Sawa, Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	3-Mono-Substituted BINOL Phosphoric Acids as Effective Organocatalysts in Direct Enantioselective Friedel–Crafts-Type Alkylation of N-Unprotected α-Ketiminoester	3-Mono-Substituted BINOL Phosphoric Acids as Effective Organocatalysts in Direct Enantioselective Friedel–Crafts-Type Alkylation of N-Unprotected α-Ketiminoester	3-Mono-Substituted BINOL Phosphoric Acids as Effective Organocatalysts in Direct Enantioselective Friedel–Crafts-Type Alkylation of N-Unprotected α-Ketiminoester	Chemistry - A European Journal, 24, 15211-15214	Chemistry - A European Journal, 24, 15211-15214	Chemistry - A European Journal, 24, 15211-15214	2018/10/12		Disclose to all
Kenta Arai, Yoshihiro Ueda, Kazuhiro Morisaki, Takumi Furuta, Takahiro Sasamori, Norihiro Tokitoh, Takeo Kawabata	Kenta Arai, Yoshihiro Ueda, Kazuhiro Morisaki, Takumi Furuta, Takahiro Sasamori, Norihiro Tokitoh, Takeo Kawabata	Kenta Arai, Yoshihiro Ueda, Kazuhiro Morisaki, Takumi Furuta, Takahiro Sasamori, Norihiro Tokitoh, Takeo Kawabata	Intermolecular Chemo- and Regioselective Aromatic C-H Amination of Alkoxyarenes Promoted by Rhodium Nitrenoids	Intermolecular Chemo- and Regioselective Aromatic C-H Amination of Alkoxyarenes Promoted by Rhodium Nitrenoids	Intermolecular Chemo- and Regioselective Aromatic C-H Amination of Alkoxyarenes Promoted by Rhodium Nitrenoids	Chemical Communications	Chemical Communications	Chemical Communications	2018	Refereed	Disclose to all
Kazuhiro Morisaki, Hiroyuki Morimoto, Kazushi Mashima, Takashi Ohshima	Kazuhiro Morisaki, Hiroyuki Morimoto, Kazushi Mashima, Takashi Ohshima	Kazuhiro Morisaki, Hiroyuki Morimoto, Kazushi Mashima, Takashi Ohshima	Development of Direct Enantioselective Alkynylation of α-Ketoester and α-Ketiminoesters Catalyzed by Phenylbis(oxazoline)Rh(III) Complexes	Development of Direct Enantioselective Alkynylation of α-Ketoester and α-Ketiminoesters Catalyzed by Phenylbis(oxazoline)Rh(III) Complexes	Development of Direct Enantioselective Alkynylation of α-Ketoester and α-Ketiminoesters Catalyzed by Phenylbis(oxazoline)Rh(III) Complexes	Journal of Synthetic Organic Chemistry, Japan, 76, 3, 226	Journal of Synthetic Organic Chemistry, Japan, 76, 3, 226	Journal of Synthetic Organic Chemistry, Japan, 76, 3, 226	2018	Refereed	Disclose to all
Masanao Sawa, Kazuhiro Morisaki, Yuta Kondo, Hiroyuki Morimoto, Takashi Ohshima	Masanao Sawa, Kazuhiro Morisaki, Yuta Kondo, Hiroyuki Morimoto, Takashi Ohshima	Masanao Sawa, Kazuhiro Morisaki, Yuta Kondo, Hiroyuki Morimoto, Takashi Ohshima	Direct Access to N-Unprotected α- and/or β-Tetrasubstituted Amino Acid Esters via Direct Catalytic Mannich-Type Reactions Using N-Unprotected Trifluoromethyl Ketimines	Direct Access to N-Unprotected α- and/or β-Tetrasubstituted Amino Acid Esters via Direct Catalytic Mannich-Type Reactions Using N-Unprotected Trifluoromethyl Ketimines	Direct Access to N-Unprotected α- and/or β-Tetrasubstituted Amino Acid Esters via Direct Catalytic Mannich-Type Reactions Using N-Unprotected Trifluoromethyl Ketimines	Chemistry - A European Journal	Chemistry - A European Journal	Chemistry - A European Journal	2017/09	Refereed	Disclose to all
Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	Kazuhiro Morisaki, Hiroyuki Morimoto, Takashi Ohshima	Direct access to N-unprotected tetrasubstituted propargylamines via direct catalytic alkynylation of N-unprotected trifluoromethyl ketimines	Direct access to N-unprotected tetrasubstituted propargylamines via direct catalytic alkynylation of N-unprotected trifluoromethyl ketimines	Direct access to N-unprotected tetrasubstituted propargylamines via direct catalytic alkynylation of N-unprotected trifluoromethyl ketimines	Chem. Commun., 53, 47, 6319	Chem. Commun., 53, 47, 6319	Chem. Commun., 53, 47, 6319	2017	Refereed	Disclose to all
Morisaki K, Morimoto H, Mashima K, Ohshima T.	Morisaki K, Morimoto H, Mashima K, Ohshima T.	Morisaki K, Morimoto H, Mashima K, Ohshima T.	Direct enantioselective alkynylation of α-ketoesters and α-ketiminoesters catalyzed by [bis(oxazoline)phenyl]rhodium(III) complexes	Direct enantioselective alkynylation of α-ketoesters and α-ketiminoesters catalyzed by [bis(oxazoline)phenyl]rhodium(III) complexes	Direct enantioselective alkynylation of α-ketoesters and α-ketiminoesters catalyzed by [bis(oxazoline)phenyl]rhodium(III) complexes	Heterocycles, 95, 2, 637-661	Heterocycles, 95, 2, 637-661	Heterocycles, 95, 2, 637-661	2017	Refereed	Disclose to all
Morisaki K, Kondo Y, Sawa M, Morimoto H, Ohshima T.	Morisaki K, Kondo Y, Sawa M, Morimoto H, Ohshima T.	Morisaki K, Kondo Y, Sawa M, Morimoto H, Ohshima T.	Synthesis of 1-tetrasubstituted 2,2,2-trifluoroethylamine derivatives via palladium-catalyzed allylation of sp<sup>3</sup>C–H bonds	Synthesis of 1-tetrasubstituted 2,2,2-trifluoroethylamine derivatives via palladium-catalyzed allylation of sp<sup>3</sup>C–H bonds	Synthesis of 1-tetrasubstituted 2,2,2-trifluoroethylamine derivatives via palladium-catalyzed allylation of sp<sup>3</sup>C–H bonds	Chemical and Pharmaceutical Bulletin, 65, 11, 1089-1092	Chemical and Pharmaceutical Bulletin, 65, 11, 1089-1092	Chemical and Pharmaceutical Bulletin, 65, 11, 1089-1092	2017	Refereed	Disclose to all
Morisaki K, Sawa M, Yonesaki R, Morimoto H, Mashima K, Ohshima T.	Morisaki K, Sawa M, Yonesaki R, Morimoto H, Mashima K, Ohshima T.	Morisaki K, Sawa M, Yonesaki R, Morimoto H, Mashima K, Ohshima T.	Mechanistic Studies and Expansion of the Substrate Scope of Direct Enantioselective Alkynylation of α-Ketiminoesters Catalyzed by Adaptable (Phebox)Rhodium(III) Complexes	Mechanistic Studies and Expansion of the Substrate Scope of Direct Enantioselective Alkynylation of α-Ketiminoesters Catalyzed by Adaptable (Phebox)Rhodium(III) Complexes	Mechanistic Studies and Expansion of the Substrate Scope of Direct Enantioselective Alkynylation of α-Ketiminoesters Catalyzed by Adaptable (Phebox)Rhodium(III) Complexes	Journal of the American Chemical Society, 138, 19, 6194-6203	Journal of the American Chemical Society, 138, 19, 6194-6203	Journal of the American Chemical Society, 138, 19, 6194-6203	2016	Refereed	Disclose to all
T. Ohshima, H. Morimoto, K. Morisaki	T. Ohshima, H. Morimoto, K. Morisaki	T. Ohshima, H. Morimoto, K. Morisaki	Catalytic Asymmetric 1,2-Alkynylation☆	Catalytic Asymmetric 1,2-Alkynylation☆	Catalytic Asymmetric 1,2-Alkynylation☆	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	2015	Refereed	Disclose to all
Morimoto H, Fujiwara R, Shimizu Y, Morisaki K, Ohshima T.	Morimoto H, Fujiwara R, Shimizu Y, Morisaki K, Ohshima T.	Morimoto H, Fujiwara R, Shimizu Y, Morisaki K, Ohshima T.	Lanthanum(III) triflate catalyzed direct amidation of esters	Lanthanum(III) triflate catalyzed direct amidation of esters	Lanthanum(III) triflate catalyzed direct amidation of esters	Organic Letters, 16, 7, 2018-2021	Organic Letters, 16, 7, 2018-2021	Organic Letters, 16, 7, 2018-2021	2014	Refereed	Disclose to all
Morisaki K, Sawa M, Nomaguchi J.-Y, Morimoto H, Takeuchi Y, Mashima K, Ohshima T.	Morisaki K, Sawa M, Nomaguchi J.-Y, Morimoto H, Takeuchi Y, Mashima K, Ohshima T.	Morisaki K, Sawa M, Nomaguchi J.-Y, Morimoto H, Takeuchi Y, Mashima K, Ohshima T.	Rh-catalyzed direct enantioselective alkynylation of α-ketiminoesters	Rh-catalyzed direct enantioselective alkynylation of α-ketiminoesters	Rh-catalyzed direct enantioselective alkynylation of α-ketiminoesters	Chemistry - A European Journal, 19, 26, 8417-8420	Chemistry - A European Journal, 19, 26, 8417-8420	Chemistry - A European Journal, 19, 26, 8417-8420	2013	Refereed	Disclose to all
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Conference Activities & Talks

Title	Title(Japanese)	Title(English)	Conference	Conference(Japanese)	Conference(English)	Date	Language	Disclose
Remote Asymmetric Induction by Chemoselective C–H Amination	Remote Asymmetric Induction by Chemoselective C–H Amination	Remote Asymmetric Induction by Chemoselective C–H Amination	11th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for young Scientists	11th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for young Scientists	11th Seoul-Kyoto-Osaka Joint Symposium on Pharmaceutical Sciences for young Scientists	2019/06/12	English	Disclose to all
触媒的化学選択的C(sp2)–H結合アミノ化による遠隔位不斉誘導	触媒的化学選択的C(sp2)–H結合アミノ化による遠隔位不斉誘導		第17回次世代を担う有機化学シンポジウム	第17回次世代を担う有機化学シンポジウム		2019/05/31	Japanese	Disclose to all
触媒的化学選択的C(sp2)–H結合アミノ化による遠隔位不斉誘導	触媒的化学選択的C(sp2)–H結合アミノ化による遠隔位不斉誘導		第139回薬学会年会	第139回薬学会年会		2019/03/23	Japanese	Disclose to all
ロジウム触媒を用いたC(sp2)-Hアミノ化による遠隔位不斉非対称化	ロジウム触媒を用いたC(sp2)-Hアミノ化による遠隔位不斉非対称化		第68回日本薬学会近畿支部総会・大会	第68回日本薬学会近畿支部総会・大会		2018/10/13	Japanese	Disclose to all
N無保護トリフルオロメチルケチミンに対する直接的触媒的アルキニル化反応	N無保護トリフルオロメチルケチミンに対する直接的触媒的アルキニル化反応		第137回薬学会年会	第137回薬学会年会		2017		Disclose to all
亜鉛触媒を用いたN無保護トリフルオロメチルケトイミンに対する直接的アルキニル化反応	亜鉛触媒を用いたN無保護トリフルオロメチルケトイミンに対する直接的アルキニル化反応		第63回有機金属化学討論会	第63回有機金属化学討論会		2016		Disclose to all
Development and Mechanistic Studies of Rh-Catalyzed Direct Enantioselective Alkynylation of α-Ketiminoesters	Development and Mechanistic Studies of Rh-Catalyzed Direct Enantioselective Alkynylation of α-Ketiminoesters		the 252nd ACS National Meeting in Philadelphia	the 252nd ACS National Meeting in Philadelphia		2016		Disclose to all
Direct Catalytic Enantioselective Alkynylation of Ketimines	Direct Catalytic Enantioselective Alkynylation of Ketimines		5th Junior International Symposium of Cutting-Edge of Organic Chemistry Asia	5th Junior International Symposium of Cutting-Edge of Organic Chemistry Asia		2015		Disclose to all
ロジウム触媒を用いたα-ケチミノエステルに対する直接的触媒的不斉アルキニル化反応の開発	ロジウム触媒を用いたα-ケチミノエステルに対する直接的触媒的不斉アルキニル化反応の開発		第13回次世代シンポジウム	第13回次世代シンポジウム		2015		Disclose to all
ケチミンに対する直接的触媒的不斉アルキニル化反応の開発	ケチミンに対する直接的触媒的不斉アルキニル化反応の開発		第31回有機合成化学セミナー	第31回有機合成化学セミナー		2014		Disclose to all
Rh(III)/Phebox-Catalyzed Direct Enantioselective Alkynylation of α-Ketiminoesters	Rh(III)/Phebox-Catalyzed Direct Enantioselective Alkynylation of α-Ketiminoesters		XXVI International Conference on Organometallic Chemistry (ICOMC 2014)	XXVI International Conference on Organometallic Chemistry (ICOMC 2014)		2014		Disclose to all
ロジウム触媒によるα-ケチミノエステルに対する直接的触媒的不斉アルキニル化反応の開発及びメカニズム解析	ロジウム触媒によるα-ケチミノエステルに対する直接的触媒的不斉アルキニル化反応の開発及びメカニズム解析		第105回有機合成シンポジウム【春】	第105回有機合成シンポジウム【春】		2014		Disclose to all
α-ケト及びケチミノエステルに対する直接的触媒的不斉アルキニル化反応の反応機構解析	α-ケト及びケチミノエステルに対する直接的触媒的不斉アルキニル化反応の反応機構解析		第134回薬学会年会	第134回薬学会年会		2014		Disclose to all
ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応の開発	ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応の開発		第22回福岡万有シンポジウム	第22回福岡万有シンポジウム		2013		Disclose to all
Rh-Catalysed Direct Enantioselective Alkynylation of α-Ketiminoesters	Rh-Catalysed Direct Enantioselective Alkynylation of α-Ketiminoesters		Twenty-third French-Japanese Symposium on Medicinal and Fine Chemistry	Twenty-third French-Japanese Symposium on Medicinal and Fine Chemistry		2013		Disclose to all
α-ケトイミノエステルの直接的触媒的不斉アルキニル化反応の開発	α-ケトイミノエステルの直接的触媒的不斉アルキニル化反応の開発		第133回薬学会年会	第133回薬学会年会		2013		Disclose to all
ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応	ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応		第29回日本薬学会九州支部大会	第29回日本薬学会九州支部大会		2012		Disclose to all
Rh-Catalyzed Direct Asymmetric Alkynylation of α-Ketoiminoesters	Rh-Catalyzed Direct Asymmetric Alkynylation of α-Ketoiminoesters		第59回有機金属化学討論会	第59回有機金属化学討論会		2012		Disclose to all
ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応の開発	ロジウム触媒によるα-ケトイミノエステルの直接的不斉アルキニル化反応の開発		第29回有機合成化学セミナー	第29回有機合成化学セミナー		2012		Disclose to all
ロジウム触媒を用いたα-ケトイミノエステルの直接的触媒的不斉アルキニル化反応の開発	ロジウム触媒を用いたα-ケトイミノエステルの直接的触媒的不斉アルキニル化反応の開発		第49回化学関連支部合同九州支部大会	第49回化学関連支部合同九州支部大会		2012		Disclose to all
Rh-Catalyzed Direct Catalytic Asymmetric Alkynylation of α-Ketoiminoesters	Rh-Catalyzed Direct Catalytic Asymmetric Alkynylation of α-Ketoiminoesters		Symposium on Molecular Chirality ASIA 2012	Symposium on Molecular Chirality ASIA 2012		2012		Disclose to all
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Books etc

Author	Author(Japanese)	Author(English)	Title	Title(Japanese)	Title(English)	Publisher	Publisher(Japanese)	Publisher(English)	Publication date	Language	Type	Disclose
Morisaki, K.; Morimoto, H.; Ohshima, T	森﨑一宏、森本浩之、大嶋孝志	Morisaki, K.; Morimoto, H.; Ohshima, T	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	Reference Module in Chemistry, Molecular Sciences and Chemical Engineering	Elsevier Inc.	Elsevier Inc.	Elsevier Inc.			Joint Work	Disclose to all
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Awards

Title(Japanese)	Title(English)	Organization name(Japanese)	Organization name(English)	Date
第137回　薬学会年会　優秀発表賞		日本薬学会		2017/03/28
5th Junior International Conference of Cutting-Edge of Organic Chemistry Asia Outstanding Oral Presentation Award		Asian Core Program		2015/11/01
第31回有機合成化学セミナー　ポスター賞		有機合成化学協会		2014/09/17
九州大学学生表彰(学術研究表彰)		九州大学		2014/03/27
第35回井上研究奨励賞	35th Inoue Research Award for Young Scientists	井上科学振興財団	Inoue Foundation for Science	2019/02/04

External funds: competitive funds and Grants-in-Aid for Scientific Research (Kakenhi)

Type	Position	Title(Japanese)	Title(English)	Period
特別研究員奨励費	Representative	不斉四置換炭素含有アミン類の立体選択的合成		2014/04/25-2017/03/31
特別研究員奨励費	Representative	化学選択性の逆転を指向した触媒反応の開発		2017/04/26-2018/03/31
若手	Representative	位置選択的C-H結合官能基化	Site-selective C-H bond functionalization	2019/04/01-2022/03/31

Teaching subject(s)

Name(Japanese)	Name(English)	Term	Department	Period
基盤精密有機合成化学実習	Laboratory Practice in Basic Fine Organic Synthesis	通年不定	薬学研究科	2019/04-2020/03
基盤精密有機合成化学実験	Research in Basic Fine Organic Synthesis	通年不定	薬学研究科	2019/04-2020/03
基盤精密有機合成化学演習	Basic Organic Chemistry Seminar	通年不定	薬学研究科	2019/04-2020/03
基礎化学実験	Fundamental Chemical Experiments	後期	全学共通科目	2019/04-2020/03

森﨑 一宏

森﨑一宏